4 Amino 3 fluorobenzonitrile 4 Fluorobenzyl cyanide 1 3 DIHYDROXYNAPHTHALENE 6 Fluoroindole 2 carboxylic acid 3 Fluoro 4 trifluoromethyl benzonitrile 4 6 Dichloropyrimidine 2 Amino 5 Bromo 3 Hydroxymethyl Pyridine 2 Trifluoromethoxy phenylhydrazine hydrochloride 2 Chloro 4 methylcinnamic acid 1 tert butyl 4 methyl 4 fluoropiperidine 1 4 dicarboxylate 5 bromo 1 2 fluoro 6 trifluoromethyl phenyl methyl 6 methyl 1 2 3 4 tetrahydropyrimidine 2 4 dione 4 chloro 2 iodo 5 trifluoromethyl 1H pyrrolo 2 3 b pyridine 4 fluoro 1H pyrrolo 2 3 b pyridin 6 amine 2S 1 methylazetidin 2 yl methanamine bis trifluoroacetic acid 2R 3R 4R 5R 2 benzoyloxy methyl 5 2 4 dioxo 1 2 3 4 tetrahydropyrimidin 1 yl 4 fluoro 4 methyloxolan 3 yl benzoate 5 bromo 2 piperidin 3 yloxy pyrimidine 2 5 dibromo 3 methoxypyrazine 2 fluoro 5 methoxypyridine 3 cyano 4 methylphenylboronic acid 4 4 4 bromophenyl 4 hydroxypiperidin 1 yl 1 4 fluorophenyl butan 1 one 4 chloro 2 fluoro 6 hydroxybenzaldehyde 5 bromo 2 4 dimethylbenzoic acid 2 amino 3 hydroxybenzoic acid 4 bromo 3 chloro 1H indazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 2 chloro 3 methylphenylboronic acid 3 4 Difluorobenzyl bromide 3 Trifluoromethoxy benzyl chloride 4 Trifluoromethoxy nitrobenzene 4 Trifluoromethyl phenethylamine

2 Trifluoromethoxy benzaldehyde 3 Fluoro 4 hydroxyacetophenone 1 4 Bis difluoromethyl benzene 4 Bromonitrobenzene 2 5 Dibromo 1 ethoxymethyl 4 nitro 1H imidazole 4 Fluoro N hydroxybenzenecarboximidamide 2 Fluoroacetophenone 2 4 Dichloro 5 nitrophenol 2 Chloro 4 hydroxycinnamic acid 2 Amino 6 fluorobenzonitrile 2 2 4 Dimethoxyphenyl acetonitrile 2 Methyl 4 nitrobenzoyl chloride 2 Chloro 5 6 7 8 tetrahydro pyrido 3 4 d pyrimidine hydrochloride 2 CHLORO 6 FLUORO 3 METHYLACETOPHENONE 2 Chloro 4 methylpyridine 3 carbonitrile 1 3 Dihydro 3 3 dimethyl 1 trifluoromethyl 1 2 benziodoxole Tognis Reagent 5 Fluoroindole 2 carboxylic acid 2 Bromo 5 fluorobenzonitrile 4 Fluoro 3 Nitrobenzonitrile 4 6 difluoropyridine 2 carboxylic acid 4H 1 Benzopyran 4 one 6 fluoro 3 3 fluorophenyl 2 1R 1 hydroxyethyl 1 tert butoxy carbonyl 4 fluoropiperidine 4 carboxylic acid 4 chloro 2 iodo 5 trifluoromethyl 1 2 trimethylsilyl ethoxy methyl 1H pyrrolo 2 3 b pyridine 6 chloro 4 fluoro 1H pyrrolo 2 3 b pyridine 3 bromo 2 fluoropyridin 4 amine 1 methylazetidin 2 yl methanamine bis trifluoroacetic acid 3 hydroxy 4 isopropoxybenzoic acid 3 5 DICHLOROPYRIDIN 2 YL METHANOL 3 ethynylphenylboronic acid 4 3 4 fluorophenyl ureido benzenesulfonamide

6 bromomethyl pyridin 2 yl methanol 4 cyano 3 trifluoromethyl phenylboronic acid 2 3 4 6 7 11b hexahydro 1H pyrazino 2 1 a isoquinoline 4 tert butyl 1 2 dichlorobenzene 3 amino 2 methoxybenzoic acid 4 bromo 3 iodo 1H indazole 4 acetyl 3 fluorophenylboronic acid 3 Trifluoromethoxy benzyl alcohol 2 4 Dibromobenzonitrile 3 Trifluoromethylthio benzoic acid 3 Trifluoromethoxy chlorobenzene 3 5 Di tert butylcyclohexane 1 2 dione 3 4 Dimethylacetophenone 2 4 Dichloro 5 nitroanisole 5 Bromo 2 iodonitrobenzene 2 5 Dibromo 4 nitro 1H imidazole 2 Fluoro 6 hydroxyacetophenone 1 4 Bis dichloromethyl benzene 2 2 6 Difluoro 3 nitrophenyl acetonitrile 3 Trifluoromethyl phenethylamine 2 3 4 Trifluorobenzaldehyde 2 Amino 5 fluorobenzonitrile 2 Amino 4 nitrobenzotrifluoride 3 5 Dichloro 4 trifluoromethyl aniline hydrochloride 2 CHLORO 4 FLUOROACETOPHENONE 3 Chlorocinnamic acid 4 Bromo 7 methoxy indan 1 one 2 Chloro 5 nitropyridin 4 amine 2 Chloro 4 methylpyrimidine 4 Fluoro 2 nitrobenzonitrile

5 6 Difluorooxindole 2 Bromo 5 fluoroacetophenone 9 1 1′ Biphenyl 4 yl 9′ 4 6 diphenyl 1 3 5 triazin 2 yl 2 2′ bi 9H carbazole 1 3 DIHYDRO 2H IMIDAZO 4 5 B PYRIDIN 2 ONE 3 5 fluoro 2 methoxyphenyl azetidin 3 ol 4 4 difluorocyclohexyl methanol 1H Pyrazolo 3 4 d pyrimidin 4 amine 3 3 fluoro 4 1 methylethoxy phenyl 5 fluoro 3 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 trimethylsilyl ethoxy methyl 1H pyrrolo 2 3 b pyridine 6 trifluoromethyl 1H pyrrolo 2 3 b pyridin 3 amine 7 trifluoromethyl 1H indazole 5 carboxylic acid 5 trifluoromethyl pyrimidine 2 carboxylic acid 4 chloro 5 fluoro 2 hydroxybenzaldehyde 3 Chloro 5 fluoro benzo d isoxazole 2 chloro 5 fluoro N N dimethylpyrimidin 4 amine 2 fluoro 3 nitrobenzonitrile 4 iodo 1 methylpyridin 2 1H one 2 bromomethyl 5 nitrobenzonitrile 4 tert butyl 1 methyl 2 nitrobenzene 4 4 dimethylamino butyl phenylboronic acid 7 4 4 2 3 dichlorophenyl piperazin 1 yl butoxy 3 4 dihydroquinolin 2 1H one 5 bromo 3 iodo 1H indazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 4 1H pyrazol 1 yl phenylboronic acid 5 bromobenzo b thiophene 2 carbaldehyde 3 Bromocinnamic acid 2 4 6 Trifluorobenzyl bromide 2 3 Dichloroanisole 2 4 6 Trifluoroiodobenzene 2 6 Dimethylacetophenone 2 5 Dimethylphenoxyacetic acid