3 4 Dihydro 2H pyrido 3 2 b 1 4 oxazine 1 ​ 2 ​ Trifluoromethyl ​pyridin ​4 ​yl ​ethanone 5 5 difluoro octahydrocyclopenta c pyrrole 6 6 difluorobicyclo 3 1 0 hexane 3 carboxylic acid 5 bromothiophen 2 yl trimethylsilane 3 N N dimethylsulfamoyl 4 methylphenylboronic acid 3 3 bis bromomethyl oxetane 2 3 3 difluorocyclopentyl ethan 1 ol 1 tert butyl 2 methyl 2R 4R 4 trifluoromethyl pyrrolidine 1 2 dicarboxylate 3 fluoro 2 methylazetidine hydrochloride 6 methoxypyrazine 2 carbonitrile 2 hydroxy 5 nitrobenzonitrile 3 cyano 2 fluorophenylboronic acid 3 piperazin 1 yl pyridazine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methyl acetate 2 chloro 4 methoxyphenyl boronic acid 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 6 chloro 1H pyrazolo 3 4 b pyridin 3 amine 5 fluoro 2 iodophenol 1 2 Fluorophenyl cyclohexanecarboxylic acid 2 Chloro 4 methylphenylhydrazine HCl 4 bromo 2 5 difluorobenzotrifluoride 3 Fluoro 2 methoxybenzoic acid 3 Chloro 2 6 difluoronitrobenzene 3 methoxy 5 methylsulfonyl aniline 2 Trifluoromethyl pyridine 3 Bromo 6 iodo o xylene 2 4 Bis trifluoromethyl acetophenone 2 5 Dichlorobenzaldehyde 4 Iodo 2 trifluoromethoxy aniline

3 4 Methylenedioxybenzyl alcohol 2 6 Difluorobenzoic acid 2 Chloroethyl benzoate 3 4 Difluorophenylacetic acid 5 Fluoro 2 trifluoromethyl benzoic acid 4 Difluoromethoxy benzyl bromide 2 Amino 4 chloro 5 iodopyridine 3 Nitrophthalic acid 2 6 Difluoro 4 iodoaniline 3 Bromo 2 fluoro 6 picoline 1 Boc 3 hydroxymethyl pyrrolidine 3 Amino 5 chlorobenzotrifluoride 3 bromo 5 fluorobenzaldehyde 1 1 1 trifluoropentan 2 one 4 4 difluoro octahydrocyclopenta c pyrrole 4 4 Dihydroxy 3 3 diformylbiphenyl 3 3 difluorocyclopentane 1 carboxylic acid 6 trifluoromethyl 2 pyridyl methanol 3S 4R 3 fluoro 4 methoxypiperidine 3 3 difluoro 2 methylazetidine hydrochloride 2 3 chloro 4 fluorophenyl 4 4 dimethyl 1 2 3 4 tetrahydroquinoline 6 carboxylic acid 6 boc 4 4 difluoro 2 6 diazabicyclo 3 2 0 heptane 4 chloro 6 fluoro 1 7 naphthyridine 3 carbonitrile 5 trimethylsilyl thiophen 2 ylboronic acid 4 bromopyridin 3 ol 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 7 carboxylic acid 2 6 dimethoxyphenyl boronic acid 3 chloro 4 iodophenol 2 4 6 trifluoro 3 methoxyphenylboronic acid 5 bromo 1H pyrazolo 3 4 b pyridin 3 amine

5 Bromothiophene 3 carboxylic acid 3 Iodobenzotrifluoride 5 Chloro 2 fluorophenylhydrazine HCl 4 Benzyloxy 3 methoxyacetophenone 4 Iodo 1 2 dimethoxybenzene 5 Bromo 2 fluoro m xylene 4 Tert butylpyridine 2 hydroxy 9H thioxanthen 9 one 2 Butene 1 4 diol 2 6 bis trifluoromethyl aniline 4 Chloro 2 5 difluorobromobenzene 2 Fluoro 4 methoxybenzoic acid 4 Iodo 2 nitroaniline 2 4 Dichlorobenzaldehyde 3 Difluoromethoxy benzyl bromide 4 Methoxybenzyl alcohol 2 5 Difluorobenzoic acid 2 6 Difluorophenylacetic acid 4 Fluoro 3 trifluoromethyl benzoic acid 3 Chlorophthalic anhydride 2 4 Difluoro 3 5 dimethoxybenzoic acid 2 3 Pyrazinedicarboxylic acid 4 Bromo 2 8 bis trifluoromethyl quinoline 2 3 Difluorochlorobenzene 5 amino 3 bromo 2 fluoropyridine 3 Amino 4 iodobenzotrifluoride 2 Bromo 5 fluorobenzaldehyde 1 1 1 3 3 Pentafluorobutane 5 methoxy 2 phenyl 1H indole 2 Amino 3 trifluoromethyl benzoic acid

4 chloro 3 5 difluoropyridine hydrochloride 4 6 difluoro 1H indazole 3 carboxylic acid 1R 2S 2 amino 1 3 5 bis trifluoromethyl phenyl propan 1 ol 3 fluoropyrazolo 1 5 a pyridin 5 amine 2 1 2 fluorophenyl methyl 1H pyrazolo 3 4 b pyridin 3 yl pyrimidine 4 5 6 triamine trihydrochloride 2 chloro 5 6 7 8 tetrahydroquinoxaline 4 chloro 5 fluoro 1H pyrrolo 2 3 b pyridine 5 chloro 3 trifluoromethyl pyridin 2 amine 3r 4s rel 4 fluoro 3 piperidinol hydrochloride 5 bromo 4 trifluoromethyl pyrimidine 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl benzaldehyde 3 cyano 4 propoxyphenylboronic acid 2 fluoro 4 iodo 6 methoxypyridine 2 bromopyrimidine 4 carbonitrile 4 chloro 2 methoxyphenyl boronic acid 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 4 methoxypyrimidin 2 amine 5 fluoro 1H pyrazolo 3 4 b pyridin 3 amine 2 Fluoro 3 chloro phenylhydrazine HCl 3 4 5 Trichlorobenzotrifluoride 4 Chloro 2 6 dibromonitrobenzene 4 Bromo 2 fluoroacetanilide 8 Chloro 6 trifluoromethyl imidazo 1 2 a pyridine 2 carboxylic acid hydrate 3 Fluoro 1 2 diethoxybenzene 5 Bromo 2 chloro m xylene 5 Amino 2 fluoroacetophenone 2 3 Dichlorobenzaldehyde 2 Iodobenzyl alcohol 2 4 Difluorophenylacetic acid 4 Fluoro 2 trifluoromethyl benzoic acid