4 Bromomethyl biphenyl 3 Amino 2 4 dichloropyridine 5 6 Dichloro 1 ethyl 2 methylbenzimidazole 4 Amino 1 Boc piperidine 4 carboxylic acid 3 Amino 5 bromo 2 chloropyridine 3 Fluoro 2 nitropyridine 2 Bromo 4 nitrotoluene 2 5 dihydro 1H Pyrrole 1 sulfonyl fluoride 2 fluoro 4 methoxy 1 propan 2 yl benzene 3 1 fluoropropyl azetidine 4 Phenoxy 2 6 Diisopropyl Aniline 1R 2 tert butyldimethylsilyl oxy 1 4 chloro 3 fluorophenyl ethan 1 ol 3 fluorooxetan 3 yl methanamine 1 5 chloro 6 fluoro 1H indol 3 yl ethan 1 ol 2 6 Difluoropyridin 4 yl boronic acid 2R 3S 3 hydroxypyrrolidine 2 carboxylic acid trifluoroacetic acid 6 fluoropyridazin 3 amine 4 cyanobenzohydrazide 2 chloromethyl oxazolo 5 4 b pyridine 2 methylpropane 1 2 diamine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrole 6 bromo 1H imidazo 4 5 b pyridine 2 methylbenzo d oxazol 5 ol 4 Butyryl benzonitrie 3 4 Difluorobenzenesulfonyl chloride 7 fluorobenzo b thiophene 2 carboxylic acid 4 fluorobenzofuran 2 carboxylic acid 2 chloro 5 cyanophenylboronic acid 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol

2 6 difluoropyridin 3 amine 2 Bromo 6 methylpyridine N oxide 5 Aminobenzimidazole 2 Cyclohexen 1 one 2 Bromo 3 methylaniline 2 Chloro 4 5 difluorobenzaldehyde 2 Chloro 4 methoxyphenol 2 Trifluoromethyl benzophenone 1 Bromo 2 fluorobenzene 2 Chlorobenzimidazole 2 Bromo 5 trifluoromethoxy aniline 3 Nitro benzenesulfonyl chloride 2 Amino 3 iodo 6 methylpyridine 5 6 Dihydro 6 oxo 11H pyrido 2 3 b 1 4 benzodiazepine 3 Fluorophenyl isothiocyanate 4 Trifluoromethyl benzyl amine 2 Fluoro 6 trifluoromethyl benzonitrile 3 Bromo 5 methylbenzoic acid 4 Bromo 2 3 5 6 tetrafluorobenzaldehyde 2 4 Dibromopyridine 2 Bromo 5 nitrobenzoic acid 2 Bromo 6 picoline 4 Piperidinecarboxylic acid 1 fluorosulfonyl ethyl ester 3 4 5 triethoxybenzoic acid 4 Methyl 2 oxopentanoic acid methyl ester 3 1 fluoroethyl azetidine 3 fluoropyrazine 2 carboxylic acid 2 4 trifluoromethyl phenyl piperazine dihydrochloride 3 5 difluoro 4 4 4 fluorophenyl piperidin 1 yl aniline 3 fluorooxetan 3 yl methanol

5 chloro 6 fluoro 1H indole 2‐ tert‐butoxy carbonyl amino ‐3‐ 3 3‐difluorocyclobutyl propanoic acid 3 Fluoropyridin 4 yl boronic acid 2R 3R 4R 5R 5 2 amino 6 chloro 9H purin 9 yl 2 4 chlorobenzoyloxy methyl 4 fluoro 4 methyloxolan 3 yl 4 chlorobenzoate 1 tert butoxycarbonyl 2 oxospiro indoline 3 4 piperidine 5 carboxylic acid 6 chloroisoquinolin 1 amine 4 4 dimethylimidazolidin 2 one 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 2 2 difluoro 1 pyridin 2 yl ethanone 3 fluoropicolinaldehyde 1H imidazo 4 5 b pyridin 2 amine 4 bromobenzo b thiophene 2 carboxylic acid 4 bromobenzofuran 2 carboxylic acid 2 chloro 5 formylphenylboronic acid 2 1H pyrazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 chloro 6 trifluoromethyl nicotinonitrile 5 Bromo 2 trifluoromethyl benzonitrile 3 Chloro 2 methylbenzenesulfonyl chloride 3 amino 9 ethylcabazole 4 Bromo 3 trifluoromethyl benzaldehyde 2 Bromo 4 iodoaniline 2 Bromomethyl 6 methylpyridine 1 Bromo 2 6 difluoro 4 iodobenzene 4 Chloro 3 fluorophenol 2 Ethoxyphenyl isothiocyanate 3 Trifluoromethyl benzyl amine 2 AMINO 3 BROMOBENZONITRILE 3 Bromo 2 methylbenzoic acid 2 Fluoro 5 trifluoromethyl benzonitrile 3 Chloro 2 hydroxybenzaldehyde

6 Bromoisoquinoline 5 5‘ Bis 2H tetrazole diammonium salt 2 3 5 6 tetrafluorobenzene 1 4 dicarboxylic acid 3 Cyano 4 isopropoxybenzoic acid 2 4 Dibromo 3 nitropyridine 2 Amino 6 nitrobenzimidazole 3 3 difluorocyclobutoxy methyl benzene 4 methoxy 2 6 dimethyl aniline 1 Bromo 3 nitrobenzene 2 5 Dimethoxybenzaldehyde 2 5 Dibromo 3 picoline 1 fluorosulfonyl 4 Piperidinecarboxylic acid 2 4 trifluoromethyl phenyl piperazine 2 chloro 5 fluoropyridine 3 carboxylic acid 3 4 methyl 1H imidazol 1 yl 5 trifluoromethyl aniline 4 fluoro 1H indazol 5 amine 2R 3R 4R 5R 2 4 chlorobenzoyloxy methyl 4 fluoro 5 hydroxy 4 methyloxolan 3 yl 4 chlorobenzoate 4 Difluoro cyclohexylidene acetic acid 3R 3 fluoropiperidine hydrochloride 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrazolo 1 5 a pyrimidine 4 amino 2 4 4 dimethyl 2 oxoimidazolidin 1 yl N 3 trifluoromethyl phenyl pyrimidine 5 carboxamide 5 bromo 1 methyl 1H pyrazole 3 carboxylic acid 7H spiro furo 3 4 b pyridine 5 4 piperidin 7 one 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 phenyloxazolo 5 4 b pyridine 3 hydroxyisonicotinaldehyde 6 bromo 3 methyl 2 trifluoromethyl pyridine 2 borono 4 fluorobenzoic acid 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl piperidin 4 one 2 Chloro 6 fluorophenyl methanesulfonyl chloride