5 bromo 2 chloro 4 trifluoromethyl pyridine 5 bromo 7 fluoro 2 3 dihydro 1H indole 5 fluorobenzo d oxazol 2 amine 2 4 fluorophenyl ethanimidamide hydrochloride 3 3 difluoro 1H 2H 3H pyrrolo 2 3 b pyridin 2 one 3H spiro isobenzofuran 1 4 piperidine 7 Bromo 2 ethyl 1H benzo d imidazole 5 carboxylic acid 4 chloro 5 fluoro 2 methyl 1H pyrrolo 2 3 b pyridine 5 trifluoromethoxy 2 3 dihydro 1H isoindole hydrochloride 1 4 chlorophenylsulfonyl 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 1 chloro 3 methoxy 5 methylbenzene 2 bromo 6 ethylphenol 2 benzyloxy 5 2 fluoropyridin 4 yl N pyridin 3 yl benzamide 5 nitroisoquinoline 4 chloro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 6 bromo 3 chlorobenzo d isoxazole 3 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 fluoro 4 methoxyphenol 3 tert butyl 4 hydroxybenzaldehyde 8 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 1 3 chlorophenyl 1H pyrazol 4 yl boronic acid 6 chloro 1H pyrazolo 4 3 c pyridin 3 amine 4 5 Difluorophthalic anhydride 3 Bromo 5 trifluoromethyl benzyl acohol 2 4 Difluoro 5 nitroanisole 1 3 Diamino 4 fluorobenzene 5 Amino 2 chloro 4 fluorophenol 5 Bromouracil 2 5 Dibromo p xylene 4 Bromoethylacetophenone

2 3 Dimethoxybenzaldehyde 2 Methyl 3 trifluoromethyl aniline 1 2 6 Dichlorophenyl ethanol 2 Methoxy 5 trifluoromethyl benzyl bromide 4 Iodo 3 trifluoromethoxy benzoic acid 5 Fluoro 2 methylphenylacetic acid 7 Chloro 6 fluoro 1 cyclopropyl 1 4 dihydro 4 oxo 3 quinoline carboxylic acid 4 Amino 2 fluorobenzoic acid 2 Fluoro 5 nitrobenzaldehyde 2 Bromo 4 fluorobenzaldehyde 4 Methylamino benzoic acid 2 Fluoro 5 nitro 6 picoline 3 Bromofuran 6 Chlorobenzo d isoxazol 3 ol 5 Trifluoromethyl pyridine 2 carboxylic acid 1 2 2 3 4 4 hexamethylphosphetane 1 oxide 1 2 2 difluoroethyl piperazine dihydrochloride 2S 4S 1 tert butoxy carbonyl 4 fluoropyrrolidine 2 carboxylic acid 4 trifluoromethyl benzo d thiazol 2 amine 5 trifluoromethoxy 2 3 dihydro 1H isoindole 6 fluoro 1H 2H 3H pyrrolo 2 3 b pyridin 2 one 2 3 trifluoromethyl phenyl ethanimidamide hydrochloride 6 4 4 chlorophenylsulfonyl piperazin 1 yl pyridin 3 ylboronic acid 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiophene 3 carbonitrile 1 benzenesulfonyl 5 bromo 4 fluoro 1H pyrrolo 2 3 b pyridine 3 difluoromethyl pyrrolidine hydrochloride 3 5 dichloro 2 methoxyisonicotinic acid 3 bromobenzene 1 2 diol 4 fluoro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 3 bromo 1 methylpyridin 2 1H one

5 chloro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 bromo 1H pyrazolo 4 3 c pyridin 3 amine 1 2 tert butyldimethylsilyl oxy ethyl 1H pyrazol 4 yl boronic acid 2 methoxy 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoxaline 4 hydroxy 2 iodobenzaldehyde 2 Fluoro 5 nitrobenzoyl chloride 2 Bromo 5 trifluoromethyl benzyl bromide 4 5 Difluorophthalic acid 3 cyano 2 hydroxybenzoic acid 2 3 Diaminobromobenzene 5 amino 2 chlorophenol 1 2 chloro 6 methoxylphenyl ethanone 2 Bromopyrimidine 2 4 Dibromo m xylene 4 Bromo 3 5 dichloro 1 trifluoromethoxy benzene 2 Bromo 2 difluoromethoxyacetophenone 4 Difluoromethoxy 3 methoxybenzaldehyde 1 2 4 Dichlorophenyl ethanol 3 Iodobenzyl bromide 4 Iodobenzoic acid 3 Fluoro 5 methylphenylacetic acid 2 Amino 5 fluorobenzoic acid 1 4 Dihydro 4 oxoquinoline 3 carboxylic acid 2 Hydroxy 3 chloro 5 trifluoromethyl pyridine 2 Bromo 4 methyl 5 nitrobenzaldehyde 1H Pyrazol 3 amine 2 Fluoro 5 iodopyridine 3 Bromo 2 chloro 6 fluorotoluene 3 Chloro 4 fluorothiophenol 1 1 2 2 Tetrafluoroethyl 2 2 3 3 tetrafluoropropylether

5 Fluoro 2 methylbenzaldehyde 3 Methoxy 2 Piperidone 4 fluoro 7 nitro 1H indazole 2 3 fluorophenyl ethanimidamide hydrochloride 5 bromo 6 fluoro 2 3 dimethyl 2H indazole 5 trifluoromethyl 1 3 benzothiazol 2 amine hydrobromide 5 fluoro 6 oxo 1 6 dihydropyridine 3 carbonitrile 3 3‐difluorocyclopentyl hydrazine 3 difluoromethyl pyrrolidine 3 Iodo 1H indazole 6 carboxylic acid 5 bromo 4 fluoro 2 iodo 1H pyrrolo 2 3 b pyridine 2 3 dibromo 6 chloropyridine 2 chloro 4 methylpyridin 3 ylboronic acid 4 3 pyridin 2 yl 1H pyrazol 4 yl quinoline 4 bromo 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 4 methylnicotinaldehyde 3 4 formylphenyl propanoic acid 3 phenyl 1H pyrazolo 4 3 c pyridine 2 hydroxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 1 2 Diamino 3 fluorobenzene 2 Bromo 5 trifluoromethyl benzyl alcohol 3 6 Difluorophthalic acid 1 2 amino 4 fluorophenyl ethanone 2 ethyl 4 hydroxybenzaldehyde 7 chloro 1H pyrazolo 4 3 c pyridine 1 4 fluorophenyl 1H pyrazol 4 yl boronic acid 4 Amino 3 chloroanisole 5 Fluoro 2 nitrobenzoic acid 2 Fluoro 5 methylphenylacetic acid 4 Hydroxy 2 trifluoromethyl benzoic acid