2 Benzyloxy 6 bromonaphthalene 6 Benzyloxy 2 bromo 5 chloronaphthalene 6 Bromo 1 chloro 2 isopropoxynaphthalene 6 Bromo 1 chloro 2 ethoxynaphthalene 4 2 5 Dibromo 3 pyridinyl carbonyl morpholine 1 4 Bromo 2 chlorobenzyl pyrrolidine hydrochloride 4 Bromo 2 chlorophenyl methyl morpholine 1 2 Bromo 5 trifluoromethyl phenyl methyl pyrrolidine hydrochloride 1 2 Bromo 5 methoxyphenyl methyl pyrrolidine 4 2 Bromo 5 methoxyphenyl methyl morpholine 4 5 bromopyridin 2 yl methyl morpholine 2 Methylthio thiophene 3 carboxylic acid 4 Bromo 2 methylthio thiophene 3 Bromo 2 methylthio thiophene 4 Methyl 2 methylthio thiophene 5 Bromo 2 4 tert butoxycarbonylpiperazin 1 yl pyridine 6 4 Methyl 1 piperazinyl 3 pyridinecarboxaldehyde 1 4 Bromobenzyl pyrrolidine 4 3 Bromobenzyl morpholine 4 Bromo 2 fluorophenyl 1 piperidinomethyl benzen 2 Propan 2 yloxy naphthalene 1 carbaldehyde 1 4 Bromobenzyl piperidine 1 4 Bromo 2 chlorophenyl methyl piperidine 4 4 fluorobenzyl morpholine 4 5 Dibromo 1H indazole 4 5 Dichloro 1 H indazole 4 6 Dichloro 1H indazole 1 Iodoisoquinoline 1 Benzyl 7 bromo 1H indazole 4 Bromo 7 methyl 1H indazole

2 Bromo 6 propoxynaphthalene 2 Bromo 6 2 methylpropoxy naphthalene 5 Bromobenzo 1 3 dioxole 4 carboxylic acid 4 7 Dibromo 1H indazole 4 Fluoro 6 methoxy 1H indazole 4 Methoxydibenzothiophene 3 6 Dimethoxypyridazine 4 carboxylic acid 4 Iodo 3 6 dimethoxy pyridazine 6 Bromo 1 tetrahydro 2H pyran 2 yl 1H indazole 1 1 Ethoxy ethyl 4 iodo 1H pyrazole 5 Bromo 1 3 benzodioxole 4 carboxaldehyde 2 3 Dibromobenzothiophene 6 Bromo 1 chloro 2 naphthol 5 Bromo 1 tetrahydro 2H pyran 2 yl 1H indazole 4 Bromo 5 methylthiophene 2 carbaldehyde 3 6 Dimethoxypyridazine 4 Bromo 1 ethylpyrazole 4 Bromo 1 2 methylpropyl 1H pyrazole 1 tetrahydro 2H pyran 2 yl 1H Imidazole 5 Bromothiophene 2 carboxaldehyde oxime 1 Bromo 4 phenylmethoxy naphthalene 2 Chloro 4 fluorophenetole 4 Cyclobutylphenyl boronic acid pinacol ester 6 Chloro 5 methoxynicotinic acid 1 Bromo 4 fluoro 2 nitrobenzene 6 Chloro 5 methoxypyridin 3 yl methanol 2 Bromo 4 trifluoromethoxy biphenyl 1 6 Bromo 5 methoxypyridin 3 yl ethan 1 one 2 5 Dichloro 3 fluorobenzoic acid 5 Chloropyridine 2 carboxamide

4 Bromo nicotinic acid methyl ester hydrobromide 3 Bromo 2 5 dichlorophenol 2 5 Dichloro 3 methoxybenzoic acid 3 Acetyl 2 6 dimethoxypyridine 4 Benzyloxy 2 chloropyrimidine 5 boronic acid 3 Bromo 2 chloro 6 methoxypyridine 6 Bromo 4 methylpyridin 3 ol 3 Chloro 2 fluoropyridine 4 carboxylic acid 2 Diisopropylamino carbonyl phenylboronic acid 4 Methanesulfonylaminophenylboronic acid pinacol ester 4 Bromo 2 chloro 3 fluoropyridine 5 Bromo 3 methyl 2 methylsulfonyl pyridine 2 4 Dichloro 3 fluoropyridine 2 6 Dimethoxy 3 methoxymethyl pyridine 4 Bromo 1 propyl 1H pyrazole 3 Bromo 2 6 dimethoxy 5 methylpyridine 4 Cyclopropylphenylboronic acid 3 Chloro 2 fluoropyridine 4 boronic acid 5 Bromo 3 iodo 2 6 dimethoxypyridine 4 Chloro 3 isopropylbenzeneboronic acid 5 Bromo 2 6 dimethoxypyridine 3 carbaldehyde 3 Acetyl 5 chlorothiophene 5 Bromo 2 6 dimethoxypyridine 3 carboxylic acid 4 Bromo 2 methoxymethoxy 1 methylbenzene 2 Benzyloxy 1 bromonaphthalene 3 Bromo 5 fluoro 2 propoxyphenylboronic acid 3 Chloro 2 6 dimethoxypyridine 1 3 2 Dioxaborolane 2 2 2 2 bis methoxymethoxy 1 1 binaphthalene 3 3 diyl bis 4 4 5 5 tetramethyl 4 Benzyloxy benzotrifluoride 6 Chlorol 3 fluoro 2 iodopyridine

2 3 Dibromo benzonitrile 2 Phenylmethoxy 3 pyridinecarboxylic acid phenylmethyl ester 4 Chloro 3 5 dibromotoluene 6 Bromo 2 Chloro 3 methylbenzaldehyde 2 Benzyloxy nicotinic acid methyl ester 2 Benzyloxy pyridin 3 yl methanol 2 6 Dichloro 4 toluidine 3 5 Dibromo 4 iodotoluene 2 Benzyloxy 3 pyridinecarbaldehyde 2 6 Dibromo 4 methylbenzaldehyde 5 Bromo 4 chloronicotinic acid 2 Bromo 4 chloro 6 fluorobenzaldehyde 2 6 Fluoropyridin 2 yl acetic acid 3 Chloro 5 methylthio pyridine 3 Fluoro 2 formyl 5 methylphenylboronic acid 1 Bromo 4 ethoxy 2 trifluoromethyl benzene 3 Chloro 5 fluoro 2 methoxybenzaldehyde 1 Bromo 3 chloro 5 trifluoromethoxy benzene 2 Ethoxynicotinic acid 2 6 Difluoro 4 iodopyridine 1 6 Bromopyridin 3 yl ethan 1 ol 2 Bromo 5 chloropyridin 3 yl methanol 2 4 Dichloro 6 fluorobenzoic acid 4 Fluoro 2 methoxymethoxy 1 methylbenzene 2 Bromo 5 chloro 3 iodopyridine 1 2 Difluoro 4 methoxymethoxy benzene 2 4 Dichloro 3 methoxyphenylboronic acid 2 Ethoxypyridine 4 carboxaldehyde 4 Methoxyphenylacetate 2 Dimethylamino pyrimidine 5 carboxylic acid