1 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 1 yl ethanone 3 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 1 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 1 yl ethanone 7 trifluoromethyl benzo b thiophen 2 yl boronic acid 2 7 fluoro 3 methylbenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 3 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 1 yl ethanone 5 trifluoromethyl benzo b thiophen 2 yl boronic acid 4 4 5 5 tetramethyl 2 5 trifluoromethyl benzo b thiophen 2 yl 1 3 2 dioxaborolane 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo b thiophene 3 carbaldehyde 2 butyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 4 trifluoromethyl phenyl thiazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 4 trifluoromethyl phenyl 1H pyrazole 1 benzyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl pyridine 1 tetrahydro 2H pyran 4 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl piperidine 1 2 pyrrolidin 1 yl ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 trimethylsilyl ethoxy methyl 1H pyrazole 1 tetrahydrofuran 3 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 cyclohexyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl acetic acid 1 cyclopentyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl ethanol 1 isobutyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 propyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 4 dimethoxypyrimidin 5 yl boronic acid

2 chloro 4 6 dimethoxypyrimidin 5 yl boronic acid 2 4 bis benzyloxy pyrimidin 5 yl boronic acid 2 phenoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 1H pyrazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 4 methylpiperazin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 isobutoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 pyrrolidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 4 methyl N 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl benzenesulfonamide 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl oxy acetonitrile 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl oxy acetonitrile 2 1H pyrazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 1H pyrrol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 2 5 dimethyl 1H pyrrol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 isopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 isopropyl 1H pyrazol 4 yl boronic acid 1 cyclopentyl 1H pyrazol 4 yl boronic acid 1 tert butyl 1H pyrazol 4 yl boronic acid 1 ethyl 1H pyrazol 4 yl boronic acid 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 2 morpholinoethyl 1H pyrazol 4 yl boronic acid 2 benzyloxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 diethoxymethyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 chlorothieno 3 2 b pyridine 5 bromothieno 3 2 b pyridine 4 chloro 3 methyl 1H pyrazolo 3 4 b pyridine 3 iodo 6 nitro 1H indazole 3 bromo 5 nitro 1H indazole 6 chloro 3 iodo 1H indazole 3 iodo 5 nitro 1H indazole 3 bromo 4 chloro 1H indazole

3 bromo 7 chloro 1H indazole 3 bromo 6 chloro 1H indazole 5 fluoro 3 iodo 1H indazole 4 fluoro 3 iodo 1H indazole 7 bromo 3 chloro 1H indazole 6 bromo 3 chloro 1H indazole 5 bromo 3 iodo 1H indazole 3 bromo 5 fluoro 1H indazole 6 fluoro 3 iodo 1H indazole 7 fluoro 3 iodo 1H indazole 3 bromo 6 fluoro 1H indazole 7 bromothieno 2 3 c pyridine 5 trifluoromethyl benzo b thiophene 2 carboxylic acid 7 bromo 3 methylbenzo b thiophene 5 fluoro 3 methylbenzo b thiophene 7 bromo 1H pyrazolo 3 4 c pyridine 4 bromo 1H pyrazolo 3 4 c pyridin 3 amine 5 7 dichloro 1H pyrazolo 3 4 c pyridine 5 trifluoromethyl 1H pyrazolo 3 4 c pyridine 7 trifluoromethyl 1H pyrazolo 3 4 c pyridine 3 bromo 1H pyrazolo 4 3 b pyridine 5 bromo 1H pyrazolo 4 3 b pyridine 6 chloro 1H pyrazolo 4 3 b pyridine 3 bromo 1H pyrazolo 3 4 c pyridine 7 bromo 1H pyrazolo 4 3 c pyridin 3 amine 1H pyrazolo 4 3 c quinolin 3 amine 6 chloro 1H pyrazolo 4 3 c pyridin 3 amine 3 bromo 1H pyrazolo 4 3 c pyridine 3 phenyl 1H pyrazolo 4 3 c pyridine 5 bromo 6 trifluoromethyl 1H pyrazolo 3 4 b pyridin 3 amine

5 bromo 1 methyl 1H pyrazolo 3 4 b pyridine 4 6 dimethyl 1H pyrazolo 3 4 b pyridin 3 amine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methyl acetate 3 chloro 5 trifluoromethyl 1H indazole 3 bromo 5 trifluoromethyl 1H indazole 3 iodo 5 trifluoromethyl 1H indazole 5 iodo 1 methyl 1H pyrazolo 3 4 b pyridin 3 amine 2 propoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 piperidin 1 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl morpholine 1 methyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 2 ethoxy 6 methylpyridin 3 yl boronic acid 3 chloro 2 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinic acid 2 3 dimethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrido 2 3 b pyrazine 2 methoxy 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 3 2 b pyridine 6 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 3 iodo 6 trifluoromethyl 1H indazole 4 fluoro 1H indazole 6 carboxylic acid 3 methyl 1H indazol 7 amine 5 chloro 3 trifluoromethyl 1H indazole 3 bromo 6 trifluoromethyl 1H indazole 2 2 chloro 6 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 fluoro 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 chloro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol