1 N BOC 4 4 METHYLCARBAMOYLPHENYL PIPERIDINE 1 BUTYL 4 FORMYL 1 METHYL 4 PHENYLPIPERIDINIUM IODIDE 2 Chloro 6 4 3 4 dichloro 5 methyl 1H pyrrol 2 yl carbonyl amino piperidin 1 yl isonicotinamide 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octane 4 methylbenzenesulfonate 4 SPIRO 1 3 4 DIHYDRO NAPHTHALENE PIPERIDINE HCL 4 AMINO 4 4 BROMO PHENYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 2 2 6 6 tetramethylpiperidin 1 ol 2 Amino dodecanoic acid 3 Methylamino L Alanine 1 Amino 3 benzyloxy cyclobutanecarboxylic acid 3S 5S 5 2 Propen 1 yl 3 morpholinecarboxylic acid methyl ester 3 Methyl L Valine Methyl ester 1 N Boc 1 7 diaza spiro 4 5 decan 6 one 1 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 1 benzyl 3 5 dimethyl piperidine 1 3 5 tricarboxylate 4 bromo 1 propyl 1 2 3 6 tetrahydropyridine 2S 4S 1 tert Butyl 2 methyl 4 aminopyrrolidine 1 2 dicarboxylate 8 Boc 2 8 DIAZA SPIRO 5 5 UNDECAN 1 ONE 3 Hydroxy pyrrolidin 1 yl acetic acid 7 Boc 2 7 DIAZA SPIRO 5 5 UNDECAN 1 ONE 10 10 DIFLUORO 2 7 DIAZA SPIRO 4 5 DECAN 1 ONE HYDROCHLORIDE 1 tert butylpiperidin 4 one 8 Boc 2 8 DIAZA SPIRO 5 4 DECAN 1 ONE 4R 1 Boc 4 Methyl D proline 1 tert butoxycarbonyl 2 methoxycarbonyl piperidine 4 carboxylic acid 4R 1 Boc 4 Methyl L proline 2S 1 tert butoxycarbonyl 4 hydroxypiperidine 2 carboxylic acid 4 bromomethyl piperidine hydrochloride 2 Phenoxymethyl morpholine 1 2 bis 1 benzylpiperidin 4 ylidene hydrazine

2 Amino 1 4 methylphenyl ethanol 2R 6R 2 6 Mimethyl piperazine 4 5 6 7 tetrahydro 1H pyrazolo 3 4 c pyridin 3 ol hydrochloride 3S 4R 4 4 Fluorophenyl 3 piperidinemethanol 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 4 tetrahydroisoquinoline 1 tert butoxycarbonyl octahydro 1H pyrrolo 3 2 c pyridine 3a carboxylic acid 2 3 4 5 Tetrahydro 8 methyl pyrido 3 2 f 1 4 oxazepine 1 HYDROXYMETHYL 2 AZABICYCLO 2 2 2 OCTANE 2 N methyl 1 HYDROXYMETHYL 2 AZABICYCLO 2 2 2 OCTANE 3 OXO 2 AZABICYCLO 2 2 2 OCTANE 1 CARBOXYLIC ACID METHYL ESTER 7 N BENZYL 1 OXO 2 7 DIAZA SPIRO 4 5 DECAN 10 ONE ETHYLENE KETAL 4 Pyridinemethaneamine 3 Dimethylaminopiperidine 1 tert butyl 3 3 dimethyl 4 oxopiperidine 1 3 3 tricarboxylate 1 1 dibenzyl 1 1 2 2 5 5 6 6 octahydro 3 3 bipyridine 1 benzyl 4 hydroxypiperidin 3 yl methyl acetate 1 4 Boc aminobutyl piperazine 4 Oxa 7 azaspiro 2 5 octane 5 6 7 8 Tetrahydro 2 6 naphthyridin 1 2H one HCl 3 oxa 9 aza bicyclo 3 3 1 nonan 7 one hydrochloride 4 Methyl 3 morpholinemethanamine 1 tert butyl 4 ethyl 4 methyl 3 oxopiperidine 1 4 dicarboxylate 6 Amino 3 4 dihydroquinolin 2 1H one 3aR 7aS 5 Boc octahydro pyrrolo 3 4 c pyridine 4 bromo 1 propyl 1 2 3 6 tetrahydropyridine hydrochloride 3aR 7aR 5 Boc octahydro pyrrolo 3 4 c pyridine 3S 5S 5 1 methylethyl 3 morpholinemethanol 2 6 DICHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 3 FLUOROPYRIDINE 4 BORONIC ACID HYDRATE 6 BROMO 2 CHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE

1R 3S 3 Aminocyclopentanol 2 ETHOXYPYRIDINE 4 BORONIC ACID 3 BROMO 2 METHOXYPYRIDINE 4 BORONIC ACID 3 Aminocyclopentanol 4 Spiroindane piperidine hydrochloride 3 5 DIMETHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 3 DIMETHOXYPYRIDINE 4 BORONIC ACID 3 Amino 2 oxazolidone hydrochloride 3 PICOLINE 4 BORONIC ACID HCL 3 Methyl 3 phenylmorpholine 3 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID 3 Methyl 5 phenylmorpholine 3 CHLORO 2 METHOXYPYRIDINE 4 BORONIC ACID PINACOL ESTER 5 pentylpicolinic acid 3R 6S tert Butyl 6 methylpiperidin 3 ylcarbamate 3 Ethenylmorpholine 3 BROMO 2 FLUOROPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 Oxa 7 azaspiro 4 5 decane 3 BROMO 5 METHOXY 4 PYRIDINYL BORONIC ACID 5 BROMO 2 ETHOXYPYRIDINE 4 BORONIC ACID 2 3 FLUOROPHENYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 2 Oxa 8 azaspiro 4 5 decane 1 4 Diazabicyclo 3 2 2 nonane 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIMETHYL ESTER 2 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 PICOLINE 4 BORONIC ACID HCL 2 ETHOXYCARBONYL PYRIDIN 4 YL BORONIC ACID 3 CYANOPYRIDINE 4 BORONIC ACID 2 3 pyridinyl morpholine 2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID

3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 3 3 Pyridinyl morpholine 2 Furan 2 yl morpholine 2 Thiophen 2 yl morpholine 2 AMINO 4 PYRIDYL BORONIC ACID 2 3 Furanyl morpholine 2 PYRIDINECARBOXAMIDE N 2 CHLORO 4 PYRIDINYL 6 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 Furan 3 yl morpholine 3 CHLORO 4 5 5 DIMETHYL 1 3 2 DIOXABORINAN 2 YL PYRIDINE 3 CHLORO 2 MORPHOLINOPYRIDINE 4 BORONIC ACID 2 Cyclohexylmethyl morpholine 2 Cyclopentylmethyl morpholine 3 CHLORO 2 4 MORPHOLINO PYRIDINE 4 BORONIC ACID PINACOL ESTER 1 ETHYL 4 TERT BUTYLOXYCARBONYL PIPERAZIN 2 ONE 5 6 7 8 tetrahydroimidazo 1 2 a pyrazine 2 carboxylic acid 2 Cyclopropylmethyl morpholine 3 Cyclopropylmethyl morpholine 2 METHYL 3 OXOPIPERAZINE HYDROCHLORIDE 2 2 Oxetanyl morpholine 2 Tetrahydro 3 furanyl morpholine 2 4 Pyridinyl morpholine 3 4 Pyridinyl morpholine 4 4 Difluoro L prolinamide hydrochloride 2 Oxetan 3 yl morpholine 3 Cyclopentylmorpholine 1 benzyl 3 methylpyrrolidin 3 ol 2 Cyclohexyl morpholine 3 ACETAMIDOPYRROLIDINE 3aR 6aS octahydrocyclopenta c pyrrole 1S tert butyl 6 oxo 5 oxa 2 aza bicyclo 2 2 1 heptane 2 carboxylate