3 4 Dibromothiophene 2 boronic acid pinacol ester 5 Bromo 2 methoxy 4 methylbenzaldehyde 5 Bromo 2 methoxy 4 methylphenyl methanol 2 Benzyloxy 5 bromo 4 methylphenyl methanol 5 Bromo 2 hydroxy 3 methylbenzyl alcohol 3 Formyl 4 methoxy 5 methylphenyl boronic acid 5 Bromo 2 ethoxy 3 methylbenzaldehyde 5 Bromo 3 methyl 2 propan 2 yloxy benzaldehyde 2 Benzyloxy 5 bromo 3 methylbenzaldehyde 3 Methyl 2 trifluoromethylpyridine 5 boronic acid 3 Chloro 2 methoxy 4 methylbenzaldehyde 3 Chloro 2 methoxy 4 methylbenzyl alcohol 3 Methyl 2 trifluoromethylpyridine 5 boronic acid pinacol ester 5 Methyl 6 trifluoromethyl nicotinic acid 2 Fluoro 4 hydroxymethyl 6 methoxyphenol 3 Fluoro 4 5 dimethoxybenzaldehyde 4 Benzyloxy 5 fluoro 3 methoxybenzyl alcohol 4 Ethoxy 3 5 difluorobenzaldehyde 5 Ethoxy 2 fluoro 4 iodopyridine 5 Benzyloxy 2 fluoro 4 iodopyridine 2 Chloro 5 trifluoromethyl 4 pyridinemethanol 4 Bromo 2 methoxy 5 methylbenzyl alcohol 2 Fluoro 5 hydroxypyridine 4 boronic acid pinacol ester 4 Chloro 2 formylphenylboronic acid pinacol ester 2 6 Difluoro 3 methoxybenzyl alcohol 4 Chloro 2 hydroxymethyl phenyl boronic acid 2 Chloro 6 hydroxy 3 methylanisole 2 Bromo 5 chlorobenzoic acid ethyl ester 5 Bromo 3 N N dimethylaminocarbonyl phenylboronic acid 5 Bromo 3 N N diethylaminocarbonyl phenylboronic acid

5 Bromo 3 pyrrolidine 1 carbonyl phenylboronic acid 5 Bromo 3 piperidine 1 carbonyl phenylboronic acid 5 Bromo 3 morpholine 4 carbonyl phenylboronic acid 5 Bromo 3 4 bromophenylcarbamoyl phenylboronic acid 5 Bromo 3 N propylaminocarbonyl phenylboronic acid 4 Methoxybiphenyl 4 carboxaldehyde 6 Bromo 2 3 dichloroanisole 3 4 Dichloro 2 methoxybenzaldehyde 2 Chloro 6 hydroxymethyl phenol 3 Chloro 2 methoxybenzoic acid methyl ester 4 Iodophenylboronic acid pinacol ester 3 Formyl 2 methoxyphenylboronic acid pinacol ester 3 Benzyloxy 4 fluorophenylboronic acid pinacolester 2 Fluoro 4 methylpyridin 3 ol 3 Chloro 4 methoxy 5 trifluoromethyl benzoic acid 3 5 Dimethoxyphenylboronic acid pinacol ester 2 5 Dimethoxy 4 methylbenzoic acid 2 5 Dimethoxy 4 methylphenylmethanol 4 Bromo 2 fluoro 6 methoxyphenol 3 Bromo 5 methylpyridin 2 yl methanol 1 Cyclopentyl 3 flouro 5 methylbenzene 1 Bromo 3 5 dichloro 4 methoxymethyl benzene 3 4 Dichloro 2 methoxyphenol 2 3 4 Dichloro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 4 Dichloro 2 methoxyphenylboronic acid 3 Bromo 5 methylpyridine 4 methanol 2 5 Fifluoro 4 formylbenzoic acid 4 Chloro 5 fluoro pyridine 3 carbaldehyde hydrochloride 3 4 Difluoro 5 methoxybenzoic acid 3 4 Difluoro 5 methoxyphenylboronic acid pinacol ester

3 4 Difluoro 5 ethoxyphenylboronic acid 9 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl 9H carbazole 2 Isopropyl 4 methoxybenzoic acid 2 Chloro 6 methoxypyridine 4 boronic acid 4 Fluoro 2 methoxy 5 methylbenzoic acid 2 Chloro 1 methoxymethoxy 3 trifluoromethyl benzene 2 Chloro 1 iodo 3 trifluoromethyl benzene 2 Isopropoxypyridin 4 yl methanol 4 Fluoro 3 isopropoxybenzoic acid 4 Fluoro 3 isopropoxybenzoic acid methyl ester 2 Methoxy 4 6 bis trifluoromethyl phenylboronic acid pinacol ester 4 Benzyloxy 3 5 dimethyl benzoic acid methyl ester 4 Methyl 1H indazole 5 boronic acid pinacol ester 3 4 Dichloro 2 formylphenylboronic acid pinacol ester 3 4 Dichloro 2 formylphenylboronic acid 2 Chloro 6 methylthio benzenemethanol 2 Bromo 6 methylsulfanyl phenyl methanol 2 Fluoro 5 propan 2 yloxy phenol 9 3 5 Dibromophenyl 9H carbazole 4 Chloro 2 fluoro 5 methylphenylboronic acid pinacol ester 3 9H Carbazol 9 yl 5 chlorophenylboronic acid 3 9H Carbazol 9 yl 5 chlorophenylboronic acid pinacol ester 3 Bromo 5 9H carbazol 9 yl phenylboronic acid pinacol ester 4 Fluoro 2 methoxy 5 methylbenzyl alcohol 5 Ethyl 2 fluorobenzoic acid 2 3 Dimethyl 4 phenylmethoxy benzaldehyde 4 Benzyloxy 2 3 dimethylphenyl boronic acid pinacol ester 5 Bromo 1 4 difluoro 2 isopropoxybenzene 2 5 Difluoro 4 isopropoxyphenylboronic acid 2 5 Difluoro 4 isopropoxybenzaldehyde

2 5 Difluoro 4 isopropoxyphenyl methanol 2 5 Difluoro 4 isopropoxybenzoic acid 3 5 Dichloropyridine 4 boronic acid pinacol ester 2 Fluoro 4 isopropoxybenzoic acid methyl ester 1 Bromo 8 phenylnaphthalene 3 Bromo 5 ethyl 2 fluorophenylboronic acid pinacol ester 6 Butoxy 5 methylpyridine 3 carboxylic acid 4 Methoxy 3 isopropylbenzyl alcohol 6 Butoxy 5 methylpyridin 3 yl methanol 2 Fluoro 4 propan 2 yloxy phenyl methanol 2 Fluoro 4 isopropoxyphenylboronic acid pinacol ester 3 Ethyl 4 formylphenylboronic acid pinacol ester 3 Bromo 2 methoxy 5 methylbenzoic acid 3 Ethyl 4 hydroxymethyl phenylboronic acid 2 Methoxy 4 methylbenzyl alcohol 2 3 Bromo 2 methoxy 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 5 Difluoro 2 propan 2 yloxy benzoic acid 3 Bromo 2 methoxy 5 methylbenzyl alcohol 4 Methyl 1H indazole 5 carbaldehyde 3 Benzyloxy pyridine 5 boronic acid pinacol ester 2 Bromo 6 fluoro 4 trifluoromethyl phenol 2 Formyl 4 methylphenylboronic acid pinacol ester 3 Chloro 5 fluoro 2 methoxyphenylboronic acid pinacol ester 3 Chloro 5 fluoro 2 methoxyphenol 3 Chloro 2 ethoxy 5 fluorophenylboronicacid pinacol ester 2 Chloro 5 trifluoromethoxy benzaldehyde 2 5 Dichloro 3 fluorophenylboronic acid 2 5 Dichloro 3 fluorophenylboronic acid pinacol ester 2 5 Dichloro 3 methoxybenzyl alcohol 5 Bromo 3 pentyloxyphenylboronic acid