2 3 Chloro 4 phenoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 HYDROXY PIPERIDINE 1 2 DICARBOXYLIC ACID 1 BENZYL ESTER 2 METHYL ESTER 1 BOC 4 4 CHLOROPHENYL 4 PIPERIDINECARBOXYLIC ACID METHYL ESTER 5 n Octylthiophene 2 boronic acid pinacol ester 5 n Octylthiophene 2 boronic acid 1 BOC 4 CYANO 4 3 BROMOPHENYL PIPERIDINE 2 8 DIAZA SPIRO 4 5 DECANE 2 3 8 TRICARBOXYLIC ACID 8 TERT BUTYL ESTER 2 9H FLUOREN 9 YLMETHYL ESTER 4 4 METHYLPHENYL 4 PHENYLPIPERIDINE HYDROCHLORIDE 5 Ethylthiophene 2 boronic acid pinacol ester 5 n Propylthiophene 2 boronic acid pinacol este 4 Trifluoromethoxy phenylboronic acid pinacol ester 2 5 butylthiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 5 Dimethyl 4 formylphenylboronic acid pinacol ester 3 TRIFLUOROMETHYL 4 5 6 7 TETRAHYDRO 1H PYRAZOLO 4 3 B PYRIDINE 4 4 BROMOPHENYL 4 4 CHLOROPHENYL PIPERIDINE 3 Chloro 2 fluorobenzeneboronic acid pinacol ester 1 2 AMINOETHYL PIPERIDIN 2 YL METHANOL 2 Methoxy 4 methoxymethoxyphenylboronic acid 2 3 Ethoxy 5 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 2 NITROPHENYL PIPERIDINE 3 Fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 3 4 trahydroquinoline 1 BOC 4 2 TRIFLUOROMETHYL PHENYL 4 HYDROXYPIPERIDINE 4 Phenylaminocarbonyl benzeneboronic acid pinacol ester 1 BOC 4 1 3 BENZODIOXOL 5 YL 4 HYDROXYPIPERIDINE 2 Benzyloxy 4 trifluoromethyl phenylboronic acid 2 2 2 trifluoro 1 piperidin 4 yl ethanone 4 Hydroxy 2 methoxyphenylboronic acid 6 METHYL 2 PIPERIDINEACETIC ACID 4 Cyclopropyl 3 mehtoxyphenylboronic acid

1 BOC 4 3 METHOXYPHENYL 4 HYDROXYPIPERIDINE 4 2 FLUORO PHENYL PIPERIDIN 4 OL 4 Isopropoxy 3 methoxyphenylboronic acid 2 Bromo 4 methoxyphenylboronic acid 4 5 6 7 Tetrahydro 1H Pyrazolo 3 4 c pyridine 3 Cyano 4 methoxyphenylboronic acid pinacol ester 1H INDAZOLE 7 CARBOXAMIDE 5 BROMO 3 4 PIPERIDINYL 1H INDAZOLE 7 CARBONITRILE 5 BROMO 3 1 ETHYLSULFONYL 4 PIPERIDINYL 4 Phenoxy 2 methoxyphenylboronic acid pinacol ester 4 Benzyloxy 2 isopropylphenylboronic acid 4 Phenoxy 2 trifluoromethyl phenylboronic acid 1 METHYL 4 PIPERIDINEACETIC ACID 5 Ethoxy 2 methylphenylboronic acid 1 BOC BETA OXO 3 PIPERIDINEPROPANOIC ACID ETHYL ESTER 3 Bromo 2 methoxyphenylboronic acid 5 1 METHYL PIPERIDIN 4 YL 1H INDOLE 3 hydroxymethyl 5 methoxyphenyl boronic acid 5 1 METHYL PIPERIDIN 4 YL 1H INDAZOLE 2 Benzyloxy 5 chloropyridine 3 boronic acid 6 1 METHYL PIPERIDIN 4 YL 1H INDAZOLE 2 Fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 AZABICYCLO 2 2 1 HEPTANE 3 CARBOXYLIC ACID 2 Fluoro 4 methylphenylboronic acid pinacol ester 9 Carbazolylbenzeneboronic acid pinacol ester 3 Bromo 2 5 dimethylphenylboronic acid 4 METHYL 3 PIPERIDINEACETIC ACID 3 Fluoro 5 morpholino phenylboronic acid pinacol ester 3 AMINO 3 4 CBZ PIPERIDINE PROPIONIC ACID ETHYL ESTER 4 4 METHANESULFONYL PHENYL PIPERIDINE 6 4 Tert butoxycarbonyl piperazin 1 yl 5 methylpyridin 3 yl boronic acid

4 BROMO METHOXYCARBONYL METHYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 3 pyridin 4 yl phenyl boronic acid 2 METHYL PIPERIDINE 1 2 DICARBOXYLIC ACID 1 BENZYL ESTER 4 Pyrid 4 yl phenylboronic acid 1 3 AMINOPROPYL PIPERIDIN 2 YL METHANOL 4 Piperidin 1 ylmethyl phenylboronic acid 6 PIPERIDIN 4 YL 1H INDOLE 2 4 Difluoro 5 bromophenylboronic acid piancol ester 2 4 chloro 2 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Chloro 6 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 3 3 DIFLUORO PIPERIDIN 1 YLAMINE 3 Cyano 5 fluorophenylboronic acid pinacol ester 2 Fluoro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 3 Formyl 4 hydroxyphenylboronic acid 1 BENZYLSPIRO INDOLE 3 4 PIPERIDIN 2 1H ONE 2 Bromo 5 methylphenylboronic acid 1 BOC 4 2 4 DIFLUOROPHENYL 4 HYDROXYPIPERIDINE 4 Hydroxymethyl 3 methoxyphenylboronic acid pinacol ester 4 2 4 DIMETHYL PHENYL PIPERIDIN 4 OL 2 Methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 2 4 PIPERIDINEDICARBOXYLIC ACID 1 3 ACETYLTHIO 1 OXOPROPYL CIS 4 Fluoro 3 hydroxyphenylboronic acid pinacol ester 2 5 PIPERIDINEDICARBOXYLIC ACID 1 3 MERCAPTO 1 OXOPROPYL CIS 4 Fluoro 3 methoxycarbonylphenylboronic acid pinacol ester 4 HYDROXY PIPERIDINE 1 2 DICARBOXYLIC ACID 1 TERT BUTYL ESTER 4 Methoxy 3 1 methylethyl phenylboronic acid 1H INDAZOLE 6 FLUORO 3 1 METHYL 4 PIPERIDINYL 2 Amino 5 trifluoromethyl phenylboronic acid pinacol ester 3 Chloro 2 methylthiopyridine 5 boronic acid 1S 2R 5R 2 HYDROXYMETHYL 3 AZA BICYCLO 3 1 0 HEXANE 3 CARBOXYLIC ACID TERT BUTYL ESTER

3 Fluorophenylboronic acid pinacol ester 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl aniline 3 Hydroxy 5 methylphenylboronic acid pinacol ester 1 PHENETHYL 4 PHENYL 4 PIPERIDINOL 4 N N Diethylaminomethyl phenylboronic acid pinacol ester 4 Hydroxy 3 isopropylphenylboronic acid pinacol ester 1H INDAZOLE 6 FLUORO 1 2 FLUOROPHENYL 3 1 METHYL 4 PIPERIDINYL 1H INDAZOLE 6 CHLORO 3 1 METHYL 4 PIPERIDINYL 2 Methyl 4 methoxymethoxy phenylboronic acid pinacol ester 4 4 BIS 4 METHOXYPHENYL PIPERIDINE 2 Isoproxy 3 methylpyridine 5 boronic acid pinacol ester 3 Methylindazole 6 boronic acid pinacol ester 5 Methyl 1H indazole 4 boronic acid pinacol ester 3 Cyclopropyl 2 6 difluorophenylboronic acid 2 Amino 5 chlorophenyl boronic acid pinacol ester 4 Cyano 3 fluorophenylboronic acid pinacol ester 2 Chloro 6 hydroxyphenylboronic acid pinacol ester 2 6 Difluoro 3 methylthio phenylboronic acid 1 tert butyl 4 ethyl 3 hydroxy 4 methylpiperidine 1 4 dicarboxylate 4 Ethoxy 2 3 dimethylphenylboronic acid 1 tert butoxycarbonyl 1 2 3 6 tetrahydropyridine 4 carboxylic acid 2 8 tert butoxycarbonyl 8 aza bicyclo 3 2 1 octan 3 yl acetic acid 2 Fluoro 4 methoxycarbonyl phenylboronic acid pinacol ester 4 Biphenyl 4 yl piperidine 4 Bromo 2 5 bifluorophenylboronic acid pinacol ester 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 dioxolan 2 yl pyridine 2 Chloro 5 formylphenylboronic acid pinacol ester 2 3 Dimethyl 4 methoxyphenylboronic acid 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 3 bromo 1 methyl 1 2 5 6 tetrahydropyridine