6 Isobutoxy 2 methylpyridine 3 boronic acid 3 hydroxy 4 5 6 7 tetrahydro 2H pyrazolo 3 4 c pyridine 5 carboxylic acid hydrochloride 2 4 Difluoro 3 iodophenylboronic acid 2 Fluoro 4 formyl 6 methoxyphenylboronic acid 4 Methoxy 2 trifluoromethoxy phenylboronic acid 4 4 bromophenyl piperidine 4 carbonitrile 6 Isopropoxynaphthalene 2 boronic acid 1 tert butyl 2 ethyl 3 oxopiperidine 1 2 dicarboxylate 3 5 Dichloro 2 6 difluorophenylboronic acid 1 benzyl 4 3 phenylpropyl 1 2 3 6 tetrahydropyridine 2 Bromo 4 methylphenylboronic acid 7 Chloro 1H indazole 4 boronic acid 1 benzyl 3 1 benzyl 2 oxo piperidin 4 ylidene piperidine 2 4 dione 6 Isopropoxy 2 methylpyridine 3 boronic acid 2 3 Dimethoxypyridine 5 boronic acid 3 3 difluoropiperidin 4 ol 2 Fluoro 3 isopropoxypyridine 5 boronic acid 5 Fluoro 2 morpholin 4 ylmethyl phenyl boronic acid 5 Chloro 2 methylsulfanyl pyridine 3 boronic acid 1 tert butyl 3 methyl 5 oxopiperidine 1 3 dicarboxylate 4 Bromo 2 Chloro 5 trifluoromethyl phenylboronic acid 3 Bromo 5 methylsulfanyl phenylboronic acid 2 Ethoxy 4 methylphenylboronic acid 2 Chloro 3 5 dimethylphenylboronic acid 4 Bromo 5 chloro 2 methylphenylboronic acid 1 HYDROXYMETHYL 3 OXO 2 AZABICYCLO 2 2 2 OCTANE 4 Bromo 2 fluoro 5 trifluoromethyl phenylboronic acid 4 Amino 3 5 dimethylphenylboronic acid pinacol ester 1 benzyl 3 hydroxymethyl piperidin 4 ol 2 6 Dimethoxybiphenyl 2 ylboronic acid

2 Tert butylcarbonylamino phenylboronic acid pinacol ester 2 Amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 8 benzyl 3 hydroxyimino 8 AZA BICYCLO 3 2 1 OCTANE 2 Fluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid methyl ester 4 Chloro 3 isopropoxyphenylboronic acid 2 Phenoxypyridine 5 boronic acid 8 benzyl 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octane 6 Fluoro 2 methylsulfanyl phenylboronic acid 4 4 bromophenyl piperidine 4 carbonitrile hydrochloride 2 Bromo 4 chlorophenylboronic acid 5 Fluoro 2 morpholinomethyl phenylboronic acid hydrochloride 5 tert butyl 3a ethyl hexahydro 1H pyrrolo 3 2 c pyridine 3a 5 6H dicarboxylate 1 methyl 4 phenylpiperidine 2 Methoxy 4 methylthio pyridine 5 boronic acid 2 Methoxy 4 methylthio pyridine 5 boronic acid pinacol ester 2 Methylthio thiophene 3 boronic acid 2 Methylthio thiophene 4 boronic acid 4 Fluoro 3 methanesulfonyl phenylboronic acid 4 Isopropoxy 3 trifluoromethyl phenylboronic acid 2 Phenoxypyridine 4 boronic acid 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 PYRIDINAMINE 2 Benzyloxy 4 methylpyridine 5 boronic acid 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 3 Bromo 2 formylthiophene 5 boronic acid 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 3 Bromo 5 carboxythiophene 2 boronic acid 2 CHLORO 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 4 N Boc piperazino pyridine 5 boronic acid 2 CHLORO 3 METHYL 5 PHENYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 3 Methoxy 2 methylphenylboronic acid

5 BROMO 2 TRIFLUOROMETHYL PYRIDIN 4 YLBORONIC ACID 2 CARBOXYPYRIDINE 4 BORONIC ACID 2 Isopropoxy 4 methylpyridine 5 boronic acid 2 Isopropoxy 4 methylpyridine 5 boronic acid pinacol ester 2 CHLORO 5 METHOXYPYRIDINE 4 BORONIC ACID 6 Ethoxy 2 fluoro 3 methylphenylboronic acid 5 Methyl 1H indazole 4 boronic acid 2 CHLORO 3 FLUORO 5 PICOLINE 4 BORONIC ACID 4 Benzyloxy 2 chlorophenylboronic acid 2 4 Difluoro 3 hydroxymethyl phenylboronic acid 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID 4 Piperazin 1 ylmethyl phenylboronic acid 2 CHLORO 3 FLUOROPYRIDINE 4 BORONIC ACID 4 2 methylpropyl amino methyl phenylboronic acid 6 Fluoro 2 hydroxy 3 methylphenylboronic acid pinacol ester 4 BORONO 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIETHYL ESTE 2 6 DIMETHYL PYRIDINE 4 BORONIC ACID 2 N BOC AMINO 6 ETHOXYCARBONYL 4 PYRIDINE BORONIC ACID PINACOL ESTER 5 Methoxy 4 methylpyridine 3 boronic acid 5 hexylpicolinic acid 4 Isobutoxyphenylboronic acid 2 4 Difluoro 3 isopropoxyphenylboronic acid 5 BROMO 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 PYRIDINECARBONITRILE 5 Diethylamino methyl 2 fluorophenylboronic acid 2 Fluoro 4 5 dimethoxyphenylboronic acid 2 Fluoro 4 morpholinomethyl phenylboronic acid 2 CYANOPYRIDIN 4 YL BORONIC ACID 5 Hydroxymethylthiophene 2 boronic acid pinacol ester 2 HYDROXY PYRIDINE 4 BORONIC ACID 2 Fluoro 4 morpholinomethyl phenylboronic acid pinacol ester

2 TERT BUTYLDIMETHYLSILYLOXY METHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 3 N N Dimethylaminomethyl phenylboronic acid pinacol ester 2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 4 Bromo 3 fluorophenylboronic acid pinacol ester 1 3 DIHYDRO 1 HYDROXY 1 2 OXABOROLO 4 3 C PYRIDINE 3 4 Dichloropyridine 5 boronic acid pinacol ester 4 Methoxy 2 6 dimethylphenylphenylboronic acid pinacol ester 2 Chloro 5 trifluoromethyl phenylboronic acid pinacol ester 3 Fluoro 4 piperidin 1 ylmethyl phenylboronic acid 2 PYRIDINECARBOXAMIDE 6 METHYL N 4 METHYL 2 THIAZOLYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 Fluoro 4 methoxycarbonylphenylboronic acid pinacol ester 3 FLUORO 2 4 MORPHOLINO PYRIDINE 4 BORONIC ACID PINACOL ESTER 6 Azaindole 4 boronic acid 1 ISOPROPYLPIPERAZINE 1 Boc 4 3 NITRO PYRIDIN 2 YL PIPERAZINE 4 Hydroxy 3 methoxyphenylboronic acid pinacol ester 1 BOC 4 BUTYLPIPERAZINE 2 Fluoro 3 piperidin 1 ylmethyl phenylboronic acid 1 BENZYL 4 3 NITROPYRIDIN 2 YL PIPERAZINE 3 Bromo 2 fluoro 6 methoxyphenylboronic acid 2 3 Difluoro 6 chlorophenylboronic acid 1 BOC 4 ISOPROPYLPIPERAZINE 4 Bromo 3 trifluoromethyl phenylboronic acid pinacol ester 4 BENZYL 3 OXOPIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 3 Fluoro 5 pyrrolidinophenylboronic acid 4 Trifluoromethylphenylboronic acid pinacol ester 2 CARBOXYMETHYL 3 OXO PIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 5 Chloro 2 propoxy 4 pyridinyl boronic acid 4 benzylpiperazin 1 amine 3 Cyano 5 methylphenylboronic acid pinacol ester