1 3 Bromophenyl 1H pyrazole 1H PYRROLO 2 3 B PYRIDINE 3 CARBONITRILE 4 CHLORO 1 PHENYLSULFONYL 8 Chloro 2 methoxy 1 5 naphthyridine 4 Piperidin 1 yl benzoic acid 1H PYRROLO 2 3 B PYRIDINE 3 BROMO 4 CHLORO 1 PHENYLSULFONYL 1H PYRROLO 2 3 B PYRIDINE 5 CARBONITRILE 4 CHLORO 1 TRIS 1 METHYLETHYL SILYL 4 Chloro 2 pyridinemethanamine 7 Methyl 1 2 3 4 tetrahydroisoquinoline 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXALDEHYDE 4 CHLORO 1 TRIS 1 METHYLETHYL SILYL 3 IODO 4 METHOXY 1H PYRROLO 2 3 B PYRIDINE 2 Chloro 6 methoxyquinoline 5 FLUORO PYRROLO 2 3 B PYRIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1H PYRROLO 2 3 B PYRIDINE 4 CHLORO 5 METHOXY 1 TRIS 1 METHYLETHYL SILYL 1 Isopropylpiperidin 4 amine 1 Piperazin 1 yl isoquinoline 5 METHOXY PYRROLO 2 3 B PYRIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID 1 TRIS 1 METHYLETHYL SILYL 2 Methyl 4 5 6 7 tetrahydrothiazolo 5 4 c pyridine 1H PYRROLO 2 3 B PYRIDINE 4 4 PHENYLMETHYL 1 PIPERIDINYL 1H PYRROLO 2 3 B PYRIDINE 4 1 PIPERIDINYL 1H PYRROLO 2 3 B PYRIDINE 4 IODO 1 TRIMETHYLSILYL 2 Pyridin 4 yl 1 p tolyl ethanone 1H PYRROLO 2 3 B PYRIDINE 5 NITRO 1 PHENYLSULFONYL 2 4 Bromophenyl piperazine 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 1H PYRROLO 2 3 B PYRIDINE 4 CHLORO 5 METHYL 1 TRIISOPROPYLSILYL 1H PYRROLO 2 3 B PYRIDINE 1H PYRROLO 2 3 B PYRIDINE 2 CARBOXALDEHYDE 1 PHENYLSULFONYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 6 Bromo 2 methylthiazolo 5 4 b pyridine 5 CHLORO 1 TRIISOPROPYLSILANYL 1H PYRROLO 2 3 B PYRIDINE 1H PYRROLO 2 3 B PYRIDINE 3 PHENYL 1 PHENYLSULFONYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL

5 Chloro 3 trifluoromethyl 1H pyrazole 5 Chloro 2 methoxyisonicotinic acid 1H PYRROLO 2 3 B PYRIDINE 4 BROMO 3 NITRO 1H PYRROLO 2 3 B PYRIDIN 3 AMINE 4 BROMO 4 Chloro 5 methoxypyrimidin 2 amine 5 Bromo 2 pyrazol 1 yl pyrimidine 1H PYRROLO 2 3 B PYRIDINE 2 METHYL 1 PHENYLSULFONYL 3 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 4 4 Bromobenzoyl piperidine hydrochloride 1H PYRROLO 2 3 B PYRIDINE 3 CARBOXYLIC ACID 4 BROMO 1 PHENYLSULFONYL 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID METHOXY METHYL AMIDE 1 1H PYRROLO 2 3 B PYRIDIN 5 YL ETHANONE 2 Bromo 4 chloro 1 nitrobenzene 2 Chloro 6 methoxybenzaldehyde 1 TRIISOPROPYLSILANYL 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID METHOXY METHYL AMIDE 3 1H PYRROLO 2 3 B PYRIDIN 5 YL ACRYLIC ACIDMETHYL ESTER 2 Methoxy 4 nitroaniline 3 Amino 5 bromopyridin 2 yl acetic acid 1H PYRROLO 2 3 B PYRIDINE 2 2 THIENYL 1H PYRROLO 2 3 B PYRIDINE 3 IODO 1 METHYL 2 PHENYL 5 Bromo 2 2 methoxyethylamino pyrimidine 2 Amino 4 picoline 2 Amino 2 phenylethanol 7 Chloro 4 piperazin 1 yl quinoline 4 Methyl 2 nitroaniline 1H PYRROLO 2 3 B PYRIDINE 2 CARBOXYLIC ACID 6 TRIFLUOROMETHYL METHYL ESTER 1 1 Biphenyl 2 amine 1H PYRROLO 2 3 B PYRIDIN 3 OL 1 PHENYLSULFONYL 3 FORMATE 1 Benzyl 7 azaindole 2 4 6 8 Tetrahydroxypyrimido 5 4 d pyrimidine 1 TOSYL 1H PYRROLO 2 3 B PYRIDINE 3 CARBALDEHYDE

3 IODO 1H PYRROLO 2 3 B PYRIDINE 4 CARBONITRILE 7 Methyl 6 azaindole 2 Bromo 5 chloronicotinic acid 3 Hydroxy 4 5 bis hydroxymethyl 2 methylpyridine 1 phenylsulfonyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridine 2 4 Methylphenyl pyrrolidine 4 Bromophenyl hydrazine hydrochloride 1 1 Oxohexadecyl L proline sodium salt 3 1 Methyl 4 piperidinyl indole 8 Ethoxycarbonyl 2 methyl 1 oxa 8 azaspiro 4 5 decan 3 one 3 Bromopropionic acid 5 Bromo 3 1 methyl 4 piperidinyl indole 3 Cyanomethyl benzoic acid 1 Boc 4 piperidin 4 yl piperazine 5 Hydroxy 1H imidazole 4 carboxamide 5 Fluoro 3 1 methyl 4 piperidinyl indole 3 Chloro 4 methoxyaniline 4 Ethyl 6 hydroxy 2 methylpyrimidine 5 Chloro 3 1 methyl 4 piperidinyl indole 1 Methylsulfonyl piperidin 4 amine 6 Chloro 5 methylpyridin 3 amine 1 1 Boc piperidin 4 yl 5 nitro 1 3 dihydro 1H benzoimidazol 2 one 4 Butylpiperidine hydrochloride 6 Bromo 1 2 3 4 tetrahydro 2 quinolinone 1 3 4 Dichloro phenyl 3 aza bicyclo 3 1 0 hexane HCl 1 TERT BUTOXYCARBONYL 4 3 CHLOROPHENYL PIPERIDINE 4 CARBOXYLIC ACID 4 Dimethylamino phenyl boronic acid hydrochloride 1 ISOPROPYL 1 METHYL 4 PHENYLPIPERIDINIUM IODIDE 5 6 Diaminopyrimidine 2 4 1H 3H dione 4 1H imidazol 1 yl benzonitrile

4 3 3 BROMO PHENYL 3 OXO PROPIONYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 4 3 4 BROMO PHENYL 3 OXO PROPIONYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 3R 4R 3 Amino 4 hydroxypentanoic acid hydrochloride 3 FLUORO 3 METHYL 1 4 NITROPHENYL METHYL PIPERIDINE 2 Nitrobenzenesulfonyl chloride 3 TRIFLUOROMETHYL 1 4 6 7 TETRAHYDRO PYRAZOLO 4 3 C PYRIDINE 5 CARBOXYLIC ACID TERT BUTYL ESTER 2 Bromo 6 fluorobenzothiazole 1 TERT BUTOXYCARBONYL 4 3 FLUOROPHENYL PIPERIDINE 4 CARBOXYLIC ACID 1H Imidazol 2 amine sulfate 1 N BOC 2R 4S 4 HYDROXY 2 HYDROXYMETHYL PIPERIDINE 2 Chloro 4 nitroaniline 2 2 4 Dichlorophenoxy propionicacid 1 Chloro 2 nitro 4 trifluoromethyl benzene 2S 4R 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID HYDROCHLORIDE 2 AZABICYCLO 2 2 2 OCTANE 3 CARBOXYLIC ACID 1 4 Nitrobenzyl 1H pyrazole 1H INDAZOLE 7 CARBOXYLIC ACID 5 BROMO 3 1 1 1 DIMETHYLETHOXY CARBONYL 4 PIPERIDINYL 1 2 Dimethyl 3 nitrobenzene 4 4 AMINOPHENYL PIPERIDINE 1 Benzyl 4 4 nitrobenzyl piperazine 3 FLUORO 1 PHENYLMETHYL 3 PIPERIDINEMETHANAMINE 5 FLUORO 1 METHYL 2 PIPERIDIN 3 YL 1H 1 3 BENZODIAZOLE 1 Boc 4 4 Formylphenyl piperazine 1 nonylpiperidine 4 carboxylic acid 1 N BOC 2 ETHOXYCARBONYLMETHYL PIPERIDINE 4 Trifluoromethyl biphenyl 4 carboxylic acid 4 Trifluoromethyl biphenyl 3 carboxylic acid 2 Trifluoromethyl biphenyl 3 carbaldehyde 4 4 difluoropiperidin 3 ol 2 1 1 Biphenyl 2 yl acetonitrile