1 prop 2 ynyl pyrrolidine 3 trifluoromethyl 1H pyrazolo 3 4 b pyridine 7 mercapto 4 methyl 2H chromen 2 one 7 4 chlorobutoxy 3 4 dihydroquinolin 2 1H one 1 2 3 4 tetrahydroisoquinolin 7 amine 5 bromo 2 1H pyrazol 3 yl pyridine 4 bromo 2 3 dimethoxybenzaldehyde 3 bromopyrazine 2 carbonitrile 2 bromonaphthalen 1 ol 2 formyl 5 methylphenylboronic acid 5 ethoxy 1H benzo d imidazole 2 3H thione 4 bromo 2 fluoro 3 methoxybenzoic acid 5 6 dimethylpyrazin 2 ol 1 isopropyl 1H pyrazol 4 amine 2 methoxy 6 methylbenzaldehyde 4 fluoronaphthalen 1 amine 7 methoxybenzo b thiophene 2 carboxylic acid 2 cyclohexyl N 1 isopropylpiperidin 4 yl 6 methoxy 7 3 pyrrolidin 1 yl propoxy quinazolin 4 amine 4 amino 2 4 4 dimethyl 2 oxoimidazolidin 1 yl N 3 trifluoromethyl phenyl pyrimidine 5 carboxamide 1 4 4 3 4 dichloro 2 fluorophenyl amino 7 methoxyquinazolin 6 yl oxy piperidin 1 yl prop 2 en 1 one 2 4 6 7 dimethoxyquinazolin 4 yl oxy phenyl N 1 isopropyl 1H pyrazol 4 yl acetamide 2 bromo 4 6 7 dimethoxyquinazolin 4 yl amino phenol 3 6 7 dimethoxyquinazolin 4 yl amino phenol 1 2 4 bromophenoxy ethyl pyrrolidine 1 tert butyl 3 p tolyl 1H pyrazolo 3 4 d pyrimidin 4 amine 2 4 5 ethylpyrimidin 4 yl piperazin 1 yl methyl 5 trifluoromethyl 1H benzo d imidazole 6 4 3 methylsulfonyl benzyl amino 5 trifluoromethyl pyrimidin 2 yl amino 3 4 dihydroquinolin 2 1H one 4 2 6 difluoro 4 3 1 piperidin 4 yl 1H pyrazol 4 yl quinoxalin 5 yl benzyl morpholine 4 6 7 dimethoxyquinazolin 4 yl amino phenol 1 4 3 amino 1H indazol 4 yl phenyl 3 2 fluoro 5 methylphenyl urea

6 1H indazol 6 yl N 4 morpholinophenyl imidazo 1 2 a pyrazin 8 amine 1 cyclopentyl N 4 6 dimethyl 2 oxo 1 2 dihydropyridin 3 yl methyl 6 4 morpholinomethyl phenyl 1H indazole 4 carboxamide 2 2 3 hydroxyphenyl amino pyrimidin 4 yl amino benzamide 4 4 aminomethyl 1 1 biphenyl 3 yl oxy pyrimidine 2 carbonitrile 2 amino 4 2 4 dichloro 5 2 pyrrolidin 1 yl ethoxy phenyl N ethylthieno 2 3 d pyrimidine 6 carboxamide 5 4 2 3 dimethyl 2H indazol 6 yl methyl amino pyrimidin 2 yl amino 2 methylbenzenesulfonamide 1H pyrrolo 2 3 b pyridin 5 ol 6 2 3 dichlorophenyl N4 methylpyrimidine 2 4 diamine 2 5 dioxopyrrolidin 1 yl 6 2 5 dioxo 2 5 dihydro 1H pyrrol 1 yl hexanoate 2 3 bromo 5 tert butyl 4 hydroxybenzylidene malononitrile 1 ethylpiperidin 3 yl 2 2 diphenylacetate 2 4 tert butyl phenyl 1H benzo d imidazole 1 4 chlorophenyl N 3 cyano 4 4 morpholinopiperidin 1 yl phenyl 5 methyl 1H pyrazole 4 carboxamide 1 2 bromophenyl 3 2 hydroxy 4 nitrophenyl urea 4 amino 2 3 bithiophene 5 carboxamide 1 4 naphthalen 2 yl pyrimidin 2 yl piperidin 4 yl methanamine 2 6 dimethylphenyl 2 4 dimethoxyphenyl 2 4 4 methylpiperazin 1 yl phenyl amino pyrimidin 4 yl carbamate 4 2 5 nitro 1H imidazol 1 yl ethyl morpholine 2 chloro N 2 N cyanosulfamoyl 1 1 biphenyl 4 yl methyl N 4 methylbenzyl benzamide 4 2 4 nitro 1H imidazol 1 yl ethyl morpholine 5 4 amino 1 isopropyl 1H pyrazolo 3 4 d pyrimidin 3 yl benzo d oxazol 2 amine 1 4 6 methyl 5 3 4 5 trimethoxyphenyl pyridin 3 yl phenyl piperazine 1 3 hydroxybenzyl 3 4 pyridin 4 yl thiazol 2 yl urea 2 methyl 2 4 2 methyl 8 pyridin 3 ylethynyl 1H imidazo 4 5 c quinolin 1 yl phenyl propanenitrile 4 1 butyl 3 phenylureido methyl N hydroxybenzamide 1 5 iodonaphthalen 1 yl sulfonyl 1 4 diazepane 2 3 5 bis trifluoromethyl phenyl N 2 dimethyl N 6 4 methylpiperazin 1 yl 4 o tolyl pyridin 3 yl propanamide 2 benzyloxy 5 2 fluoropyridin 4 yl N pyridin 3 yl benzamide 4 3 pyridin 2 yl 1H pyrazol 4 yl quinoline 2 phenyl 4 3 pyridin 2 yl 1H pyrazol 4 yl pyridine

4 4 3 pyridin 2 yl 1H pyrazol 4 yl pyridin 2 yl N tetrahydro 2H pyran 4 yl benzamide 3 6 4 trifluoromethoxy phenyl amino pyrimidin 4 yl benzamide 2 2 hydroxyethoxy ethyl 2 3 trifluoromethyl phenyl amino benzoate 4 methoxy 2 2 dimethyl 4 oxobutanoic acid 4 2 5 ethoxy 1H benzo d imidazol 2 yl thio ethyl morpholine 6 chloro 9 4 methoxy 3 5 dimethylpyridin 2 yl methyl 9H purin 2 amine 4 2 6 dichlorobenzamido N piperidin 4 yl 1H pyrazole 3 carboxamide 3 chlorophenyl 6 7 dimethoxy 1 4 methoxyphenoxy methyl 3 4 dihydroisoquinolin 2 1H yl methanone 4 4 4 3 acrylamidophenyl amino 5 fluoropyrimidin 2 yl amino phenoxy N methylpicolinamide 5 3 chlorophenyl N 4 morpholinomethyl phenyl furan 2 carboxamide 2 1 4 chlorobenzoyl 5 methoxy 2 methyl 1H indol 3 yl 1 morpholinoethanone 3 azepan 1 ylsulfonyl N 3 bromophenyl benzamide 6 bromo 2 iodoquinazoline 2 2 5 5 oxybis ethane 2 1 diyl bis oxy bis pyridine 5 2 diyl bis 6 trifluoromethoxy 1H benzo d imidazole 2 3 4 dihydroxybenzylidene malononitrile 3 6 methylpyridin 2 yl N phenyl 4 quinolin 4 yl 1H pyrazole 1 carbothioamide 4 3 6 methylpyridin 2 yl 1H pyrazol 4 yl quinoline 1 4 morpholinomethyl phenyl ethanone 2 6 dibromo 3 nitrophenol 2 4 dibromo 3 hydroxybenzoic acid 2 7 methoxynaphthalen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 3 bromo 2 hydroxyphenyl ethanone 3 6 dibromo 2 hydroxybenzoic acid 4 bromo 2 3 dihydroxybenzoic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoquinoline 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoxaline 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiophene 2 carbaldehyde 2 2 3 dihydrobenzofuran 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole

2 benzofuran 7 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzo b thiophen 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzo b thiophen 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 triisopropylsilyl 1H pyrrole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyrimidin 2 amine 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 3 dimethylcarbamoyl phenylboronic acid 3 methoxymethyl phenylboronic acid 2 4 boronophenyl acetic acid 5 methoxy 2 methylphenylboronic acid 1 methyl 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 6 dichloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 cyclopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 isopropylthio phenylboronic acid 4 piperidin 1 yl phenylboronic acid hydrochloride 4 bromo 2 6 difluorophenylboronic acid 2 ethylthio phenylboronic acid 4 chloro 2 6 difluorophenylboronic acid 4 pyrrolidin 1 yl phenylboronic acid 3 4 5 trichlorophenylboronic acid 2 3 difluoro 6 methoxyphenylboronic acid 3 amino 4 fluorophenylboronic acid 2 chloro 4 trifluoromethyl phenylboronic acid 4 benzyloxycarbonylamino phenylboronic acid 3 benzyloxycarbonyl phenylboronic acid 4 methoxy 3 methylphenylboronic acid