4 bromo 2 tert butyl phenol 4 4 cyano 2 methoxyphenyl 5 ethoxy 2 8 dimethyl 1 4 dihydro 1 6 naphthyridine 3 carboxylic acid 4 bromo 2 phenylthiazole 3 methoxyisonicotinaldehyde 2 cyanoethyl 4 4 cyano 2 methoxyphenyl 2 8 dimethyl 5 oxo 1 4 5 6 tetrahydro 1 6 naphthyridine 3 carboxylate 2 bromo 5 methylnicotinonitrile 3 Bromopropionaldehydedimethylacetal 4 CYANO 2 METHOXYBENZALDEHYDE 2 fluoro 3 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 4 6 Trimethylaniline 2 hydroxy 6 methoxybenzaldehyde 2 chloro N MesitylpyriMidin 4 aMine 2 6 dimethoxybenzaldehyde 6 hydroxy N 2 dimethylbenzofuran 3 carboxamide 3 bromo 6 chloropicolinaldehyde 2 3 4 6 7 11b hexahydro 1H pyrazino 2 1 a isoquinoline 4 hydroxy 3 methoxyphenylboronic acid 5 fluoro 2 methoxyisonicotinaldehyde 6 4 Fluoro phenyl pyridine 3 carbaldehyde 6 furan 2 yl 1H indole 1 4 dimethylamino phenyl ethanone 4 Chloromethyl 2 4 fluorophenyl pyridine 5 methyl 1H 1 2 3 triazole 4 carboxylic acid 3 AMINO 4 5 DIHYDRONAPHTHO 1 2 B THIOPHENE 2 CARBOXYLIC ACID METHYL ESTER 2 4 dipropoxyphenyl boronic acid 4 bromophenyl 4 1 4 dioxa 8 azaspiro 4 5 decan 8 ylmethyl phenyl methanone 4 4 5 5 tetramethyl 2 3 methylthiophen 2 yl 1 3 2 dioxaborolane 4 chloro 2 3 dimethylpyridine 5 Fluoro 2 methoxybenzoic acid 4 bromo 2 cyclopropoxypyridine

1 4 methoxypyridin 2 yl ethanone 2 fluoro 3 nitrobenzaldehyde 1 5 chloro 2 methoxyphenyl ethanone 1 6 chloropyridin 3 yl ethanone 2 Methyloxazole 4 carboxaldehyde 1 amino 2 3 4 dimethoxyphenyl ethyl boronic acid 4 Formylbenzoic acid 1 2 methylamino ethyl piperidin 4 yl 1 1 biphenyl 2 ylcarbamate 1 amino 2 3 4 dihydroxyphenyl ethyl boronic acid 4 2 amino 2 boronoethyl benzoic acid 1 2 3 4 carbamoylpiperidin 1 yl methyl N methylbenzamido ethyl piperidin 4 yl 1 1 biphenyl 2 ylcarbamate 2 BIPHENYLYL ISOCYANATE 1 amino 3 phenylpropyl boronic acid 2 benzyl methyl amino acetaldehyde 1 amino 3 phenylpropyl boronic acid 1 amino 2 phenylethyl boronic acid 1 aminoethyl boronic acid 4 4 4 trifluoro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 1 Pyrrolidinecarboxylic acid 2 8 amino 1 bromoimidazo 1 5 a pyrazin 3 yl phenylmethyl ester 2S 2 phenyl 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl ethanamine 2S 1 phenylmethoxycarbonylpyrrolidine 2 carboxylic acid 5 chloro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pentan 1 amine 4 methoxy 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 5 bromo 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pentan 1 amine 3 3 difluoro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl propan 1 amine 3 3 difluoro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl propan 1 amine 4 Chloro 1H pyrrolo 2 3 b pyridine 3 carbaldehyde 4 chloro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 4 4 5 6 trifluoromethyl pyridin 3 ylamino pyridin 2 yl phenyl cyclohexyl 4 bromo 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine

4 fluoro 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 5 amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pentan 1 ol 3 Pyridinecarboximidamide N hydroxy 1 oxide 9CI 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl but 3 en 1 amine 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl but 3 en 1 amine 4 4 Hydroxyphenyl cyclohexanone 2 methyl 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 3 methyl 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 3 methyl 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 3 methyl 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl butan 1 amine 1 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl propan 1 amine 2 amino 5 ethylbenzoic acid 4 chloro 3 methylpicolinonitrile 2 bromo 5 chloropyrimidine 3 5 diethoxyaniline 5 chloropyridin 3 yl boronic acid 31 trimethylsilylether rapamycin 4 iodopyrimidine 2 furan 2 carbonyl benzoic acid 1 2 3 difluoro 4 trifluoromethyl phenyl ethanone 5 boronothiophene 2 carboxylic acid 3 formylisonicotinonitrile 2 ethyl naphtho 1 2 b furan 4 5 quinone 6 formylnicotinonitrile 3 E but 1 enyl 4 hydroxynaphthalene 1 2 dione 6 methyl 2 nitropyridin 3 ol 6 methoxybenzo b thiophene 2 ethyl naphtho 2 3 b furan 4 9 quinone 1 methyl 1H pyrazol 3 yl boronic acid

2 1 hydroxyethyl benzo f 1 benzofuran 4 9 dione 4 chloro 2 isopropylpyridine 2 bromo 3 chlorothiophene 5 methoxypyridin 2 amine 2 Hydroxy 1 4 naphthoquinone 4 chloro 3 methylpicolinaldehyde 1 2 4 benzotriazin 3 amine 2 amino 4 phenyl 1H pyrrole 3 carbonitrile 2 bromo 1 4 ethylphenyl ethanone 1 methyl 1H 1 2 3 triazole 3 hydroxy 6 methylpicolinaldehyde 1S 5R 6S 7R 8S 9S 7 acetoxy 9 benzyloxy methoxy 5 tert butoxycarbonyl amino 6 S 2 2 dimethyl 1 3 dioxolan 4 yl 8 hydroxy 2 oxabicyclo 3 3 1 non 3 en 8 yl methyl benzoate 5 chloro 2 methoxypyridin 3 yl boronic acid 1S 5R 8S 8aR 5 benzyloxy methoxy 7 tert butyldiphenylsilyl oxy methyl 3 hydroxy 1 hydroxymethyl 3 5 8 8a tetrahydro 1H isochromen 8 yl benzoate 5 bromo 1 methylpyridin 2 1H one 1S 2R 3S 4R 5S 6R 2 acetoxy 5 benzyloxy methoxy 4 tert butoxycarbonyl amino 3 S 2 2 dimethyl 1 3 dioxolan 4 yl 4 2 oxoethyl 7 oxabicyclo 4 1 0 heptan 1 yl methyl benzoate 4 trifluoromethyl pyrimidin 2 ol 5 bromo 6 chloropyrimidin 4 amine 2 chloro 5 fluorobenzene 1 3 diamine 1S 4R 6R E 4 benzyloxy methoxy 2 tert butyldiphenylsilyl oxy methyl 6 S 2 2 dimethyl 1 3 dioxolan 4 yl 5 2 hydroxyethylidene cyclohex 2 en 1 ol 6 bromo 1 2 3 4 tetrahydroquinoxaline 1 2 4 5 Dianhydro cis inosit 1 6 naphthyridine 8 bromo 1 6 naphthyridine 2 3 anhydro 1 4 di O benzyl myo inositol 1 chloro 7 nitroisoquinoline 7 nitroisoquinolin 1 2H one 5 nitroisoquinolin 1 amine 1 bromo 2 7 naphthyridine 2R 3R 4S 5R 6S 6 methoxy 3 4 5 tris phenylmethoxy oxan 2 yl methanol