5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridin 2 3H one 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 1 yl ethanone 2 7 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 7 trifluoromethyl benzo b thiophen 2 yl 1 3 2 dioxaborolane 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H imidazo 4 5 b pyridine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 trityl 1H pyrazolo 3 4 b pyridine 8 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyrimidine 2 5 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 5 methylbenzo b thiophen 2 yl 1 3 2 dioxaborolane 2 6 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 5 5 tetramethyl 2 3 methylbenzo b thiophen 5 yl 1 3 2 dioxaborolane 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazol 2 yl morpholine 2 cyclohexyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 2 isopropyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 trityl 1H pyrazole 1 4 methoxybenzyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 3 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl pyridine 1 methyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl piperidine 2 methyl 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazol 1 yl propan 2 ol 1 isopentyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 2 methoxyethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 cyclopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 6 dimethoxypyrimidin 5 yl boronic acid 2 4 diethoxypyrimidin 5 yl boronic acid 1 tert butyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl piperidin 4 ol 2 1H imidazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 piperazin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine

2 propoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 4 methoxyaniline 3 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 propoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 isopentyl 1H pyrazol 4 yl boronic acid 1 benzyl 1H pyrazol 4 yl boronic acid 1 isobutyl 1H pyrazol 4 yl boronic acid 1 methyl 1H pyrazol 4 yl boronic acid 1 trityl 1H pyrazol 4 yl boronic acid 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyridin 2 amine 2 4 methyl 1H pyrazol 1 yl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 benzyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 1H one 1 3 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 1H one 2 1 1 diethoxyethyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methylthio 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 bromo 6 chloro 1H pyrazolo 3 4 b pyridine 6 chloro 3 trifluoromethyl 1H pyrazolo 3 4 b pyridine 6 methyl 1H pyrazolo 3 4 b pyridine 4 bromo 3 iodo 1H indazole 4 bromo 3 chloro 1H indazole 4 chloro 3 iodo 1H indazole 3 bromo 5 chloro 1H indazole 5 chloro 3 iodo 1H indazole 7 chloro 3 iodo 1H indazole 3 chloro 1H indazol 5 amine

3 bromo 6 nitro 1H indazole 5 bromo 3 chloro 1H indazole 6 bromo 3 iodo 1H indazole 3 bromo 4 fluoro 1H indazole 5 chlorothieno 2 3 c pyridine 3 bromo 7 fluoro 1H indazole 7 chlorothieno 2 3 c pyridine 5 chlorothieno 2 3 b pyridine 4 chloro 3 methylbenzo b thiophene 3 methoxy 2 nitroaniline 5 chloro 3 methylbenzo b thiophene 6 chloro 3 methylbenzo b thiophene 5 bromo 1H pyrazolo 4 3 b pyrazin 3 amine 5 iodo 1H pyrazolo 4 3 b pyrazin 3 amine 5 chloro 1H pyrazolo 4 3 b pyrazine 5 bromo 1H pyrazolo 4 3 b pyrazine 5 bromo 3 methyl 1H pyrazolo 4 3 b pyrazine 5 chloro 3 methyl 1H pyrazolo 4 3 b pyrazine 3 bromo 1H pyrazolo 4 3 b pyrazine 4 bromo 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 4 fluoro 1H pyrazolo 3 4 c pyridin 3 amine 4 chloro 1H pyrazolo 3 4 c pyridin 3 amine 5 chloro 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 7 chloro 5 trifluoromethyl 1H pyrazolo 3 4 c pyridine 3 trifluoromethyl 1H pyrazolo 3 4 c pyridine 7 chloro 1H pyrazolo 4 3 b pyridine 6 bromo 1H pyrazolo 4 3 b pyridine 6 bromo 1H pyrazolo 4 3 b pyridin 3 amine 4 bromo 1H pyrazolo 4 3 c pyridin 3 amine 5 bromo 1H pyrazolo 4 3 b pyridin 3 amine

2 6 dimethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 methyl 1H pyrazolo 3 4 b pyridin 3 amine 2 fluoro 4 iodo 6 methoxypyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 6 trifluoromethyl pyridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 2 butoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 isobutoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 methyl N 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl benzenesulfonamide 2 6 diethoxypyridin 3 yl boronic acid 2 pyrrolidin 1 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 1H imidazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 fluoro N methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile 2 fluoro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 3 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 4 1H 3H dione 3 methyl 4 nitro 1H indazole 3 methyl 5 nitro 1H indazole 3 bromo 7 trifluoromethyl 1H indazole 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 ol 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 5 naphthyridine 2 4 methoxy 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 chloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 2 methoxy 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 4 4 5 5 tetramethyl 2 2 methyl 5 trifluoromethyl phenyl 1 3 2 dioxaborolane 2 4 tert butyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 fluoro 3 methoxyphenyl boronic acid