2 5 chloro 2 2 methoxy 4 4 methylpiperazin 1 yl phenyl amino pyrimidin 4 yl amino N methylbenzenesulfonamide 4 3 trifluoromethyl benzyl 2H benzo b 1 4 thiazin 3 4H one 3 isobutyryl 1 2 oxo 3 4 phenoxyphenoxy propyl 1H indole 5 carboxylic acid 4 4 4 bromophenyl 4 hydroxypiperidin 1 yl 1 4 fluorophenyl butan 1 one 1 ethylpiperidin 3 yl 2 2 diphenylacetate 3 dimethylamino N 3 4 hydroxybenzamido 4 methylphenyl benzamide 4 3 4 fluorophenyl ureido benzenesulfonamide 2 phenylamino 1 4 phenylene bis 4 pyrrolidin 1 yl piperidin 1 yl methanone 5 bromopyridin 3 yl 4 pyrrolidin 1 yl piperidin 1 yl methanone 2 5 chloro 2 2 methoxy 4 morpholinophenyl amino pyrimidin 4 yl amino N methylbenzamide 3 5 p tolyl thieno 2 3 d pyrimidin 4 yl thio propanoic acid 4 amino 2 1 methylsulfonyl piperidin 4 yl amino pyrimidin 5 yl 2 3 difluoro 6 methoxyphenyl methanone 1 2 methylbenzo d oxazol 6 yl 3 1 5 naphthyridin 4 yl urea 3 4 dimethoxy N 4 3 nitrophenyl thiazol 2 yl benzenesulfonamide 4 benzylpiperazin 1 yl 2 isopentylamino pyridin 3 yl methanone 2 chloro 5 nitro N phenylbenzamide 1 1 4 4 5 chloropyrimidine 2 4 diyl bis azanediyl bis 3 methoxy 4 1 phenylene bis piperazine 4 1 diyl diethanone 2 4 amino 1 isopropyl 1H pyrazolo 3 4 d pyrimidin 3 yl 1H indol 5 ol 4 methyl 2 piperidin 1 yl quinoline 1 4 chlorobenzyl 2 pyrrolidin 1 ylmethyl 1H benzo d imidazole 1 4 chlorobenzyl 2 pyrrolidin 1 ylmethyl 1H benzo d imidazole 2 methyl 2 3 methyl 4 4 methylamino 5 trifluoromethyl pyrimidin 2 yl amino 1H pyrazol 1 yl propanenitrile 2 methyl 1 2 methyl 3 trifluoromethyl benzyl 6 morpholino 1H benzo d imidazole 4 carboxylic acid 3 6 amino 5 3 4 5 trimethoxyphenyl pyridin 3 yl phenol 2 bromo N 3 butyramidophenyl benzamide 4 methyl N1 3 phenylpropyl benzene 1 2 diamine 1 5 chloro 2 methoxyphenyl 3 2 methylquinolin 4 yl urea 4 acetamido N 2 aminophenyl benzamide 3 5 dichloro 2 hydroxy N 4 methoxy 1 1 biphenyl 3 yl benzenesulfonamide 4 tert butyl N 2 methyl 3 4 methyl 6 4 morpholine 4 carbonyl phenyl amino 5 oxo 4 5 dihydropyrazin 2 yl phenyl benzamide

8 2 4 2 methoxyphenyl piperazin 1 yl ethyl 8 azaspiro 4 5 decane 7 9 dione 3 5 dibromo 1 methylpyrazin 2 1H one 6 bromoquinazolin 2 amine 1 3 4 dichlorobenzyl indoline 2 3 dione 1 4 methoxybenzyl 3 5 nitrothiazol 2 yl urea 3 4 dimethylamino 1 1 biphenyl 3 yl 1 1 dimethylurea 4 6 methoxyquinolin 8 yl amino pentanoic acid 4 methyl 3 2 2 morpholinoethyl amino quinazolin 6 yl N 3 trifluoromethyl phenyl benzamide 2 nitro 5 phenylsulfonyl phenyl 4 chlorobenzoate 4 5 5 8 8 tetramethyl 5 6 7 8 tetrahydronaphthalene 2 carboxamido benzoic acid 5 5 8 8 tetramethyl 5 6 7 8 tetrahydronaphthalene 2 carboxylic acid 2 4 benzoylphenoxy N 1 benzylpiperidin 4 yl acetamide 1 2 4 benzyl 4 hydroxypiperidin 1 yl ethyl 3 2 methylquinolin 4 yl urea 4 bromo 3 hydroxy 2 nitrobenzoic acid 4 morpholinomethyl benzonitrile 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl indolin 2 one 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoindolin 1 one 3 bromo 6 fluoro 2 hydroxybenzaldehyde 4 bromo 2 chloro 3 hydroxybenzoic acid 2 bromo 3 methyl 6 nitrophenol 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 3 dihydro 1H inden 1 one 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 methyl 1H indazol 6 yl boronic acid 4 4 5 5 tetramethyl 2 7 nitrobenzofuran 5 yl 1 3 2 dioxaborolane 2 benzofuran 4 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzofuran 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane

2 benzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzo b thiophen 4 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 ethylcarbamoyl phenylboronic acid 4 isobutylcarbamoyl phenylboronic acid 4 methoxymethoxy phenylboronic acid 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 benzo b thiophen 7 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrole 4 benzylcarbamoyl phenylboronic acid 4 diethylcarbamoyl phenylboronic acid 4 tert butoxycarbonyl phenylboronic acid 3 5 difluoro 2 methoxyphenylboronic acid 2 3 dihydrobenzo b 1 4 dioxin 5 ylboronic acid 3 borono 2 fluorobenzoic acid 2 chloro 4 ethoxyphenylboronic acid 2 chloro 4 hydroxyphenylboronic acid 2 3 4 trichlorophenylboronic acid 2 methoxy 5 methylphenylboronic acid 4 3 methoxy 3 oxoprop 1 enyl phenylboronic acid 4 benzyloxy 3 formylphenylboronic acid 2 fluoro 3 methoxyphenylboronic acid 3 trimethylsilyl ethynyl phenylboronic acid 4 benzyloxycarbonylamino methyl phenylboronic acid 3 isopropylphenylboronic acid

3 hydroxy 4 methylphenylboronic acid 2 4 6 trimethoxyphenylboronic acid 2 boronobenzoic acid 4 dimethylamino methyl phenylboronic acid 2 3 5 trichlorophenylboronic acid 2 4 6 trifluorophenylboronic acid 3 fluoro 2 formylphenylboronic acid 1 acetylindolin 5 ylboronic acid 4 cyano 3 trifluoromethyl phenylboronic acid 3 cyano 4 methylphenylboronic acid 2 cyanomethyl phenylboronic acid 5 chloro 2 cyanophenylboronic acid 4 4 dimethylamino butyl phenylboronic acid 3 1H imidazol 2 yl phenylboronic acid 4 octyloxy phenylboronic acid 2 3 boronophenyl acetic acid 3 4 difluoro 5 methoxyphenylboronic acid 4 cyano 3 methoxyphenylboronic acid 2 hydroxy 3 trifluoromethyl phenylboronic acid 3 chloro 2 hydroxyphenylboronic acid 4 ethynylphenylboronic acid 4 chloro 3 ethoxyphenylboronic acid 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 bromo 2 cyclopropylpyrimidine 2 cyclopropyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 bromo 2 ethylpyridine 5 bromobenzo b thiophene 2 carbonitrile 6 bromo 2 methoxypyridin 3 amine 5 bromo 2 chloro 4 methylthio pyrimidine 4 bromopyrimidin 2 amine