1H PYRROLO 2 3 B PYRIDINE 4 CHLORO 3 NITRO 4 Acetyl 2 methylpyridine 1 3 Bromophenyl 1H pyrazole 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXALDEHYDE 1 TRIS 1 METHYLETHYL SILYL 6 Bromo 1H indole 2 carboxylic acidmethylester 1 boc 4 5 bromopyrimidin 2 yl piperazine 1H PYRROLO 2 3 B PYRIDINE 5 CARBONITRILE 4 CHLORO 1 TRIS 1 METHYLETHYL SILYL 4 Piperidin 1 yl benzoic acid 8 Chloro 2 methoxy 1 5 naphthyridine 1H PYRROLO 2 3 B PYRIDINE 3 CARBONITRILE 4 CHLORO 1 PHENYLSULFONYL 1H PYRROLO 2 3 B PYRIDINE 3 BROMO 4 CHLORO 1 PHENYLSULFONYL 7 Methyl 1 2 3 4 tetrahydroisoquinoline 2 Chloro 6 methoxyquinoline 1H PYRROLO 2 3 B PYRIDINE 4 CHLORO 5 METHOXY 1 TRIS 1 METHYLETHYL SILYL 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXALDEHYDE 4 CHLORO 1 TRIS 1 METHYLETHYL SILYL 4 Chloro 2 pyridinemethanamine 3 IODO 4 METHOXY 1H PYRROLO 2 3 B PYRIDINE 5 FLUORO PYRROLO 2 3 B PYRIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID 1 TRIS 1 METHYLETHYL SILYL 5 METHOXY PYRROLO 2 3 B PYRIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1 Piperazin 1 yl isoquinoline 1 Isopropylpiperidin 4 amine 2 Methyl 4 5 6 7 tetrahydrothiazolo 5 4 c pyridine 2 Pyridin 4 yl 1 p tolyl ethanone 2 4 Bromophenyl piperazine 1H PYRROLO 2 3 B PYRIDINE 5 NITRO 1 PHENYLSULFONYL 1H PYRROLO 2 3 B PYRIDINE 4 IODO 1 TRIMETHYLSILYL 1H PYRROLO 2 3 B PYRIDINE 4 4 PHENYLMETHYL 1 PIPERIDINYL 1H PYRROLO 2 3 B PYRIDINE 4 1 PIPERIDINYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 1H PYRROLO 2 3 B PYRIDINE

4 CHLORO 5 METHYL 1 TRIISOPROPYLSILYL 1H PYRROLO 2 3 B PYRIDINE 1H PYRROLO 2 3 B PYRIDINE 2 CARBOXALDEHYDE 1 PHENYLSULFONYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 5 CHLORO 1 TRIISOPROPYLSILANYL 1H PYRROLO 2 3 B PYRIDINE 6 Bromo 2 methylthiazolo 5 4 b pyridine 1H PYRROLO 2 3 B PYRIDINE 3 PHENYL 1 PHENYLSULFONYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 5 Chloro 3 trifluoromethyl 1H pyrazole 1H PYRROLO 2 3 B PYRIDINE 4 BROMO 3 NITRO 5 Chloro 2 methoxyisonicotinic acid 1H PYRROLO 2 3 B PYRIDIN 3 AMINE 4 BROMO 5 Bromo 2 pyrazol 1 yl pyrimidine 1 1H PYRROLO 2 3 B PYRIDIN 5 YL ETHANONE 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID METHOXY METHYL AMIDE 4 4 Bromobenzoyl piperidine hydrochloride 1H PYRROLO 2 3 B PYRIDINE 3 CARBOXYLIC ACID 4 BROMO 1 PHENYLSULFONYL 1H PYRROLO 2 3 B PYRIDINE 2 METHYL 1 PHENYLSULFONYL 3 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 4 Chloro 5 methoxypyrimidin 2 amine 2 Bromo 4 chloro 1 nitrobenzene 2 Chloro 6 methoxybenzaldehyde 3 1H PYRROLO 2 3 B PYRIDIN 5 YL ACRYLIC ACIDMETHYL ESTER 1 TRIISOPROPYLSILANYL 1H PYRROLO 2 3 B PYRIDINE 5 CARBOXYLIC ACID METHOXY METHYL AMIDE 1H PYRROLO 2 3 B PYRIDINE 3 IODO 1 METHYL 2 PHENYL 5 Bromo 2 2 methoxyethylamino pyrimidine 1H PYRROLO 2 3 B PYRIDINE 2 2 THIENYL 3 Amino 5 bromopyridin 2 yl acetic acid 1H PYRROLO 2 3 B PYRIDIN 3 OL 1 PHENYLSULFONYL 3 FORMATE 1H PYRROLO 2 3 B PYRIDINE 2 CARBOXYLIC ACID 6 TRIFLUOROMETHYL METHYL ESTER 1 TOSYL 1H PYRROLO 2 3 B PYRIDINE 3 CARBALDEHYDE 2 Amino 4 picoline 7 Chloro 4 piperazin 1 yl quinoline 2 Amino 2 phenylethanol

1 phenylsulfonyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridine 3 Hydroxy 4 5 bis hydroxymethyl 2 methylpyridine 2 Bromo 5 chloronicotinic acid 7 Methyl 6 azaindole 2 4 6 8 Tetrahydroxypyrimido 5 4 d pyrimidine 2 4 Methylphenyl pyrrolidine 4 Bromophenyl hydrazine hydrochloride 8 Ethoxycarbonyl 2 methyl 1 oxa 8 azaspiro 4 5 decan 3 one 5 Bromo 3 1 methyl 4 piperidinyl indole 3 1 Methyl 4 piperidinyl indole 1 1 Oxohexadecyl L proline sodium salt 5 Hydroxy 1H imidazole 4 carboxamide 1 Boc 4 piperidin 4 yl piperazine 3 Cyanomethyl benzoic acid 4 Ethyl 6 hydroxy 2 methylpyrimidine 5 Chloro 3 1 methyl 4 piperidinyl indole 6 Bromo 1 2 3 4 tetrahydro 2 quinolinone 1 Methylsulfonyl piperidin 4 amine 1 1 Boc piperidin 4 yl 5 nitro 1 3 dihydro 1H benzoimidazol 2 one 6 Chloro 5 methylpyridin 3 amine 4 3 3 BROMO PHENYL 3 OXO PROPIONYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1 3 4 Dichloro phenyl 3 aza bicyclo 3 1 0 hexane HCl 5 6 Diaminopyrimidine 2 4 1H 3H dione 1 ISOPROPYL 1 METHYL 4 PHENYLPIPERIDINIUM IODIDE 4 Dimethylamino phenyl boronic acid hydrochloride 4 1H imidazol 1 yl benzonitrile 3R 4R 3 Amino 4 hydroxypentanoic acid hydrochloride 4 3 4 BROMO PHENYL 3 OXO PROPIONYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 3 FLUORO 3 METHYL 1 4 NITROPHENYL METHYL PIPERIDINE 3 TRIFLUOROMETHYL 1 4 6 7 TETRAHYDRO PYRAZOLO 4 3 C PYRIDINE 5 CARBOXYLIC ACID TERT BUTYL ESTER

2 Bromo 6 fluorobenzothiazole 1H Imidazol 2 amine sulfate 1 N BOC 2R 4S 4 HYDROXY 2 HYDROXYMETHYL PIPERIDINE 2S 4R 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID HYDROCHLORIDE 1 4 Nitrobenzyl 1H pyrazole 2 AZABICYCLO 2 2 2 OCTANE 3 CARBOXYLIC ACID 1H INDAZOLE 7 CARBOXYLIC ACID 5 BROMO 3 1 1 1 DIMETHYLETHOXY CARBONYL 4 PIPERIDINYL 4 4 AMINOPHENYL PIPERIDINE 1 Benzyl 4 4 nitrobenzyl piperazine 1 nonylpiperidine 4 carboxylic acid 1 Boc 4 4 Formylphenyl piperazine 5 FLUORO 1 METHYL 2 PIPERIDIN 3 YL 1H 1 3 BENZODIAZOLE 3 FLUORO 1 PHENYLMETHYL 3 PIPERIDINEMETHANAMINE 2 Amino 5 bromo 2 fluorobenzophenone 6 FLUORO 2 3 DIHYDRO 1 H SPIRO CYCLOPROPANE 1 4 ISOQUINOLINE 2 1 1 Biphenyl 2 yl acetonitrile 1 Boc 4 5 Aminopyridin 2 yl piperazine 2 Trifluoromethyl biphenyl 3 carbaldehyde 4 4 difluoropiperidin 3 ol 4 Trifluoromethyl biphenyl 3 carboxylic acid 1 N BOC 2 ETHOXYCARBONYLMETHYL PIPERIDINE 4 Trifluoromethyl biphenyl 4 carboxylic acid 8 FLUORO 2 3 DIHYDRO 1 H SPIRO CYCLOPROPANE 1 4 ISOQUINOLINE 3 1 tert Butoxycarbonyl piperidin 4 yl propanoic acid 4 BENZYLOXY METHYL 3 3 DIFLUOROPIPERIDINE 4 4 Ethylpiperazin 1 yl benzaldehyde 1 3 3 DIFLUORO 4 4 DIHYDROXY PIPERIDIN 1 YL 2 2 2 TRIFLUORO ETHANONE 3 TRIFLUOROMETHYL 4 5 6 7 TETRAHYDRO ISOXAZOLO 4 5 C PYRIDINE 1 Methyl 3 piperidin 4 yl 1H benzo d imidazol 2 3H one 8 3 CHLORO 5 FLUOROBENZYL 3 METHYLAMINO METHYL 8 AZA BICYCLO 3 2 1 OCTAN 3 OL