1 1 dibenzyl 1 1 2 2 5 5 6 6 octahydro 3 3 bipyridine 1 benzyl 4 hydroxypiperidin 3 yl methyl acetate 1 4 Boc aminobutyl piperazine 4 Oxa 7 azaspiro 2 5 octane 4 Methyl 3 morpholinemethanamine 3 oxa 9 aza bicyclo 3 3 1 nonan 7 one hydrochloride 5 6 7 8 Tetrahydro 2 6 naphthyridin 1 2H one HCl 3S 5S 5 1 methylethyl 3 morpholinemethanol 1 tert butyl 4 ethyl 4 methyl 3 oxopiperidine 1 4 dicarboxylate 4 bromo 1 propyl 1 2 3 6 tetrahydropyridine hydrochloride 3aR 7aR 5 Boc octahydro pyrrolo 3 4 c pyridine 3aR 7aS 5 Boc octahydro pyrrolo 3 4 c pyridine 3 Methyl 5 phenylmorpholine 6 Amino 3 4 dihydroquinolin 2 1H one 2 6 DICHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 6 BROMO 2 CHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 3 FLUOROPYRIDINE 4 BORONIC ACID HYDRATE 3 Amino 2 oxazolidone hydrochloride 3 5 DIMETHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 3 DIMETHOXYPYRIDINE 4 BORONIC ACID 4 Spiroindane piperidine hydrochloride 3 Aminocyclopentanol 3 BROMO 2 METHOXYPYRIDINE 4 BORONIC ACID 2 ETHOXYPYRIDINE 4 BORONIC ACID 1R 3S 3 Aminocyclopentanol 3 PICOLINE 4 BORONIC ACID HCL 3 Methyl 3 phenylmorpholine 3 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID 3 CHLORO 2 METHOXYPYRIDINE 4 BORONIC ACID PINACOL ESTER 3 BROMO 2 FLUOROPYRIDINE 4 BORONIC ACID PINACOL ESTER

3R 6S tert Butyl 6 methylpiperidin 3 ylcarbamate 3 Ethenylmorpholine 3 BROMO 5 METHOXY 4 PYRIDINYL BORONIC ACID 5 pentylpicolinic acid 2 Oxa 7 azaspiro 4 5 decane 5 BROMO 2 ETHOXYPYRIDINE 4 BORONIC ACID 2 3 FLUOROPHENYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 2 Oxa 8 azaspiro 4 5 decane 1 4 Diazabicyclo 3 2 2 nonane 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIMETHYL ESTER 2 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 ETHOXYCARBONYL PYRIDIN 4 YL BORONIC ACID 2 3 pyridinyl morpholine 2 PICOLINE 4 BORONIC ACID HCL 3 3 Pyridinyl morpholine 2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID 3 CYANOPYRIDINE 4 BORONIC ACID 3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 AMINO 4 PYRIDYL BORONIC ACID 2 Thiophen 2 yl morpholine 2 Furan 2 yl morpholine 3 CHLORO 4 5 5 DIMETHYL 1 3 2 DIOXABORINAN 2 YL PYRIDINE 3 Furan 3 yl morpholine 2 PYRIDINECARBOXAMIDE N 2 CHLORO 4 PYRIDINYL 6 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 Cyclohexylmethyl morpholine 3 CHLORO 2 MORPHOLINOPYRIDINE 4 BORONIC ACID 2 3 Furanyl morpholine 3 CHLORO 2 4 MORPHOLINO PYRIDINE 4 BORONIC ACID PINACOL ESTER 1 ETHYL 4 TERT BUTYLOXYCARBONYL PIPERAZIN 2 ONE 2 Cyclopentylmethyl morpholine

5 6 7 8 tetrahydroimidazo 1 2 a pyrazine 2 carboxylic acid 2 Cyclopropylmethyl morpholine 2 2 Oxetanyl morpholine 3 Cyclopropylmethyl morpholine 2 METHYL 3 OXOPIPERAZINE HYDROCHLORIDE 3 Cyclopentylmorpholine 2 Oxetan 3 yl morpholine 2 4 Pyridinyl morpholine 4 4 Difluoro L prolinamide hydrochloride 3 4 Pyridinyl morpholine 2 Cyclohexyl morpholine 3 ACETAMIDOPYRROLIDINE 2 Tetrahydro 3 furanyl morpholine 1 benzyl 3 methylpyrrolidin 3 ol 3aR 6aS octahydrocyclopenta c pyrrole 1S tert butyl 6 oxo 5 oxa 2 aza bicyclo 2 2 1 heptane 2 carboxylate 4 1 Piperazinylmethyl benzoicacid 1 tert butyl 2 methyl 2 ethyl 4 oxopyrrolidine 1 2 dicarboxylate 3 Azaspiro 5 5 undecan 9 one 4 Amino 3 Pyrrolidinol 3 methylpyrrolidin 3 ol hydrochloride 7 Azaspiro 3 5 nonane 3 Azabicyclo 3 1 0 hexane 5 Bromo 1 2 3 4 tetrahydro 1 7 naphthyridine 7 3 TRIFLUOROMETHYL PHENYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXAMIDE 3 2 Bromoethyl Pyridine 5 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 OL 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDIN 2 AMINE 3 Hydroxymethylmorpholine 7 Chloro 3 quinolinamine

6 2 CARBOXYBIPHENYL 4 YL METHYL 7 HYDROXY 5 PROPYLPYRAZOLO 1 5 A PYRIMIDINE 1 2 4 CHLOROPHENYL 7 METHYLPYRAZOLO 1 5 A PYRIMIDIN 6 YL ETHAN 1 ONE 2 Amino N cyclopropyl acetamide 2 TERT BUTYL 7 CHLORO 5 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 5 7 BIS TRIFLUOROMETHYL 2 METHYLTHIO PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXAMIDE 3 Maleimidopropionicacidhydrazide 5 Maleimidovaleric acid hydrazide 5 7 BIS TRIFLUOROMETHYL 3 CYANOPYRAZOLO 1 5 A PYRIMIDINE 6 4 METHOXY PHENYL 3 PHENYL PYRAZOLO 1 5 A PYRIMIDINE 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 2 3 DIAMINE 6 Maleimidocaproic acid hydrazide Trifluoroacetic Acid 2 Maleimidoacetic acid hydrazide 7 AMINO 2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 5 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 AMINE 2 Ethyl morpholine 2 Isobutylmorpholine 6 BROMO PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 2 4 BROMOPHENYL 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 5 ISOPROPYL 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE 7 Methyl 5 azaspiro 2 4 heptan 7 amine 5 1 METHYL CYCLOPROPYL 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 5 Azaspiro 2 4 heptan 1 amine dihydrochloride 9CI 6 BROMO 3 CHLOROPYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 5 Azaspiro 2 4 hept 1 yl carbamic acid tert butyl ester 6 TERT BUTYLSULFONYL 2 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 AMINE 2R 6R 2 6 Dimethyl piperazine 6 NITROPYRAZOLO 1 5 A PYRIMIDINE 5 METHYL 3 PHENYL PYRAZOLO 1 5 A PYRIMIDIN 7 YL HYDRAZINE 7 CHLORO 5 6 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE