6 methoxyindoline 6 Ethyl 5 fluoro 4 hydroxypyrimidine 4 5 Diaminopyrimidine 5 fluoro 2 methylbenzaldehyde 5 Fluoro 1 indanone 2 4 5 Trifluoroaniline 4 Fluoro 3 nitrobenzenesulfonamide 3 Bromo 2 chloropyridine 4 5 Dichloro 1 2 benzenediamine 2 Methyl 3 nitroaniline 4 Amino 3 5 dichloroacetophenone 2 amino 4 trifluoromethyl benzoic acid 1 Methyl 1H imidazole 4 carboxylic acid 5 Bromo 2 methoxy 4 methyl 3 nitropyridine 2 Methoxy 5 pyridineboronic acid 3 Iodo 4 methoxyaniline 2 Chloro 3 cyanopyridine 3 Bromo 4 methoxypyridine 2 4 Dichloro 5 nitropyridine 2 Fluoro 5 methoxyaniline 2 Chloro 5 fluoro 3 nitropyridine 1S 2S 3R 5S Pinanediol 2 Trifluoromethyl benzaldehyde 9 3 Bromophenyl 10 2 naphthyl anthracene 4 Pentynoic acid 2 Chloro 4 methylpyridine 3 carbonitrile 2 2 Diphenylglycine 2 Amino 4 5 difluorobenzoic acid 5 Methyl 1H pyrrolo 2 3 b pyridine 3 Fluoro 4 methoxyaniline

4 5 Difluorophthalic acid 2 Chloro 6 cyanopyridine 2 6 Difluorobenzotrifluoride 4 Hydroxymethyl phenylboronic acid 3 Bromo 2 fluoroanisole 5 Bromo 2 chlorophenol 4 2 Aminoethyl tetrahydropyran 1 N Boc pyrrolidin 2 ylboronic acid 3 Formylphenylboronic acid 1 hydroxymethyl cyclopropaneactetonitrile 3 Fluoro 4 trifluoromethoxy aniline 1 Bromo 3 chloro 2 5 difluorobenzene 1 Methylcyclopropene 3 nitro 4 trifluoromethyl aniline 2 4 5 trifluorophenylacetic acid 4 Bromobenzamidine 1 2 4 5 Tetrafluoro 3 nitrobenzene 3 Aminopropylphosphate 2 Chloro 5 cyanomethyl pyridine 5 Methyl 3 2H pyridazinone 2 Chloro 5 nitropyridine 4 amine 4 Methoxy 2 trifluoromethyl benzaldehyde 4 Bromo 3 5 dimethylphenol 3 Chloro 2 iodoaniline 3 Nitrophthalic acid 2 Nitro 4 trifluoromethyl aniline 2 4 Dibromo 3 fluoro nitrobenzene 2 Amino 4 bromopyridine 2 Chloro 4 methylaniline 3 chloro 4 fluorocinnamic acid

3 Bromo 4 fluorotoluene 3 Fluoro 2 nitropyridine 3 4 Dimethylphenylaceticacid 2 4 Difluoro 3 trifluoromethyl benzoic acid 4 chloro 3 nitrophenol 5 Cyano 2 fluoro 3 picoline 4 chloro 2 trifluoromethyl phenylboronic acid 5 Fluoro 2 methylbenzoic acid 5 Bromo 2 chloropyrimidine 1 Bromo 2 chloro 4 iodobenzene 2 Pyridineethanol 2 Methyl 4 trifluoromethyl aniline 3 Fluoro 4 methyl 5 hydroxybenzoic acid 4 Bromo 3 methylthiophenecarboxylic acid 4 Bromo 3 fluorotoluene 4 Bromo Thiazole 3 Cyclopropyl 3 oxopropanenitrile 3 4 Dihydro 7 methoxy 4 oxoquinazolin 6 yl acetate 5 Chloro 3 n methoxy carbonyl methyl sulfamoyl 2 thiophene carboxylic acid methyl ester 6 Chloromethyl uracil 2 Chloro 4 trifluoromethyl aniline 5 Bromo 3 methyl 1H indazole 5 Chloro 1H pyrrolo 2 3 b pyridine 4 Amino 2 chloropyridine 3 Chloro 2 fluoroaniline 3 Hydroxypyrazine 2 carboxylic acid 2 Amino 2 fluoro 5 bromobenzophenone 2R 2 Aminopropanamide hydrochloride 1 Bromonapthalene 6 Trifluoromethyl indole

3 Chloro 4 bromotoluene 3 4 Difluorotoluene 1 Aminomethyl adamantane 5 bromofuran 2 carbonyl chloride 2 amino 3 chloro 4 fluoronitrobenzene 5 Chloro 2 fluoro 3 hydroxypyridine 5 Chloro 3 fluorobenzene 1 2 diol 1 4 5 8 tetrahydro 2 7 dimethoxy Naphthalene 2 Fluoro 5 hydroxy 3 picoline 3 Amino 4 picoline 2 Chloro 6 phenylnicotinonitrile 2 Fluoro 6 nitrobenzonitrile 1 2 Dimethylaminoethyl 1H Tetrazole 5 Thiol 2 6 10 Trimethylundeca 5 9 dienal Cidalor 2 6 Difluorobenzyl alcohol 3 Isobutylglutaric acid 2 Isopropoxy 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Amino 3 fluoropyridine 3R 4R 1 Benzyl N 4 dimethylpiperidin 3 amine dihydrochloride 2 4 Dichloro 7H pyrrolo 2 3 d pyrimidine 2 Ethylbenzaldehyde 3 S 1 Carbamoyl 1 1 diphenylmethyl pyrrolidine L tartrate 3 5 Dimethoxyaniline 3 Fluoro 4 trifluoromethyl benzonitrile 1 1 1 Trifluoro 3 chloropropane 3 Amino 4 iodopyridine 2 Chloro 4 fluorobenzonitrile 1H Pyrazole 2 Amino 3 5 dibromotoluene 2 3 Pyrazinedicarboxylic anhydride