5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 triisopropylsilyl 1H pyrrole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyrimidin 2 amine 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 9 Amino 2 bromoacridine 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5’ 6’ 7’ 8’ tetrahydrospiro cyclohexane 1 2’ 1’h quinazolin 4’ 3’h one 2 cyclopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 6 dichloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Aminophenylboronic acid pinacol ester 1 methyl 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 3 methoxymethyl phenylboronic acid 2 4 boronophenyl acetic acid 2 Chloro 4 6 di morpholin 4 yl 1 3 5 triazine 5 methoxy 2 methylphenylboronic acid 3 dimethylcarbamoyl phenylboronic acid 2 2 2 diethylaminoethylamino ethyl 4 methyl 1H pyrrole 3 carboxylicacid ethyl ester 4 isopropylthio phenylboronic acid 4 piperidin 1 yl phenylboronic acid hydrochloride 2 2 diethylaminoethylcarbamoyl methyl 4 methyl 1H pyrrole 3 carboxylic acid ethyl ester 4 bromo 2 6 difluorophenylboronic acid 2 carboxymethyl 4 methyl 1H pyrrole 3 carboxylic acid ethyl ester 3 4 dichlorobenzoyl chloride 2 ethylthio phenylboronic acid 4 chloro 2 6 difluorophenylboronic acid 4 pyrrolidin 1 yl phenylboronic acid 3 4 5 trichlorophenylboronic acid 3 amino 4 fluorophenylboronic acid 2 3 difluoro 6 methoxyphenylboronic acid

4 cyano N 4 cyanophenyl benzamide 3 3 methoxy 3 oxoprop 1 enyl phenylboronic acid 4 cyanobenzoyl chloride 4 methoxy 3 methylphenylboronic acid 2 tert butyl 4 chloro 5 4 2 hydroxyethoxymethyl benzyloxy 2H pyridazin 3 one 3 benzyloxycarbonyl phenylboronic acid 4 benzyloxycarbonylamino phenylboronic acid 2 tert butyl 4 chloro 5 hydroxypyridazin 3 2H one 3 aminomethyl phenylboronic acid hydrochloride 4 2 tert butyldimethylsilyloxy ethoxy methyl phenyl methanol 3 isopropoxycarbonyl phenylboronic acid 3 tert butoxycarbonyl phenylboronic acid 2 morpholinomethyl phenylboronic acid 4S 5S 5 methyl 2 oxo 1 3 oxazinane 4 carboxylic acid 4 benzyloxy phenylboronic acid 4 aminophenylboronic acid 2 ethynylphenylboronic acid 4 1H imidazol 1 yl phenylboronic acid 2 methylbenzo d oxazol 6 ylboronic acid 4 fluoro 2 formylphenylboronic acid 2S 3S 3 2S 1 4 aminobutylamino 4 methyl 1 oxopentan 4 formyl 3 methoxyphenylboronic acid 1 chloromethyl 4 trifluoromethyl benzene 3 amino 5 trifluoromethyl phenylboronic acid 4 trimethylsilyl ethynyl phenylboronic acid 2S 6 dimethylamino 2 2 methylpropan 2 yl oxycarbonylamino hexanoic acid 2S 3R 3 2 methylpropan 2 yl oxy 2 2 methylpropan 2 yl oxycarbonylamino butanoic acid 2 6 difluoro 4 formylphenylboronic acid 3 cyano 4 methoxyphenylboronic acid 2 tert butoxycarbonylamino 5 fluorophenylboronic acid

2 methoxy 5 nitrophenylboronic acid 4 borono 2 nitrobenzoic acid 4 chloro 2 cyanophenylboronic acid 4 2 2R 3R 3 2 4 difluorophenyl 3 hydroxy 4 1 2 4 triazol 1 yl b utan 2 yl 1 3 thiazol 4 yl benzonitrile 3 benzyloxy 4 methoxyphenylboronic acid 5 2 2 dibromoethenyl 2 methoxyphenol 3 acetyl 4 fluorophenylboronic acid 3 chloro 5 cyanophenylboronic acid 3 cyano 5 fluorophenylboronic acid 2 cyano 6 fluorophenylboronic acid 3 chloro 5 methylphenylboronic acid 2 tert butoxycarbonyl 1 2 3 4 tetrahydroisoquinolin 7 ylboronic acid 3 fluoro 4 trifluoromethyl phenylboronic acid 3 5 difluoro 4 methoxyphenylboronic acid 2 hydroxy 3 methoxyphenylboronic acid 2 hydroxy 3 methylphenylboronic acid 4 trifluoromethyl pyrimidin 2 amine 2 bromo 5 methoxypyridine 2 bromo 4 trifluoromethyl pyrimidine 2 BROMO 5 6 DICHLOROBENZIMIDAZOLE 6 nitropyridin 3 ol 2 nitro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 2 bromopyrimidin 4 amine 2 bromo 5 fluoropyrazine 2 Amino 5 bromobenzoic acid 4 6 dibromopyrimidine 8 Nitroquinoline 1 phenylcyclopropanamine 8 CHLORO 3 IODOQUINOLINE

2 3 4 6 tetra O benzoyl D glucopyranosyl trichloroacetimidate 3 bromo 2 hydroxybenzoic acid 2 bromo 6 isopropylphenol 2 3 6 tribromophenol 2 6 dibromo 3 methylphenol 2 3 4 6 Tetra O benzyl D glucopyranose 2 bromo 6 ethylphenol 3 bromobenzene 1 2 diol 4 6 O benzylidene α D glucopyranosyl 1→1 4 6 O benzylidene α D glucopyranoside 2 3 dihydrobenzofuran 6 yl methanol 2 ​ 1R ​5S ​6R ​ ​6 ​cyano ​3 ​ethylbicyclo 3 2 0 ​hept ​3 ​en ​6 ​yl ​ ​ 1 ​3 ​diethyl ester 8 chloro 1 7 naphthyridine 5 bromo 2 methoxybenzonitrile 5 bromo 2 iodophenol 2​ 1R ​5S ​ ​3 ethylbicyclo 3 2 0 ​hept ​3 ​en ​6 ​ylidene ​ ​ 1 ​3 ​diethyl ester 3 bromo 2 chloroisonicotinic acid 2 bromo 1 4 difluoromethoxy phenyl ethanone 4 ethyl 3 hydroxyhept 6 enoic acid 3 hydroxy 4 methylbenzonitrile 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl benzaldehyde 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 7 carboxylic acid 2 3 dibromo 4 methylpyridine 3 6 dibromopicolinic acid 3 ethynyl 4 methylbenzoic acid 2 3 Dihydrofuran 1 3 bromophenyl 2 phenyl 1H benzo d imidazole 2 5 FLUORO 1H INDOL 3 YL ETHANOL 4 methylimino cyclohexanone ketal 3 5 diethynylbenzoic acid 1 4 dimethylamino phenyl 5 oxopyrrolidine 3 carboxylic acid