1 ​tert ​butyl 2 ​Methyl 5 ​5 ​difluoropiperidine ​1 ​2 ​dicarboxylate 6 trifluoromethyl 1h pyrazolo 4 3 b pyridine 5 chloro 3 fluoropyridine 2 carboxylic acid 3 trifluoromethoxy pyridin 2 amine 1 tert butyl 3 methyl 3 fluoropyrrolidine 1 3 dicarboxylate 1 1 1 Trifluoro 5 5 dimethyl 2 4 hexanedione 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 fluoro 4 iodopyridin 2 amine 6 chloro 5 fluoro 4 iodopyridin 3 amine 5 6 difluoropyridine 3 carboxylic acid 1 tert butyl 3 methyl 5 trifluoromethyl piperidine 1 3 dicarboxylate 3 trifluoromethyl 1H pyrrolo 2 3 b pyridin 4 amine 1 tert butoxy carbonyl 3 fluoropiperidine 4 carboxylic acid 1 1 1 Trifluoropropan 2 ol 5 difluoromethyl 1 methyl 1H pyrazole 4 carboxylic acid 1r 3r 4r rel 2 boc 5 5 difluoro 2 azabicyclo 2 2 2 octane 3 carboxylic acid 5 trifluoromethyl benzo b thiophen 2 yl boronic acid 2 5 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 fluorobenzo b thiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 5 fluoro 2 3 dihydro 1H isoindole 1 3 dione 5 bromo 3 3 difluoro 1 methyl 2 3 dihydro 1H indol 2 one 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 4 trifluoromethyl phenyl 1H pyrazole 1 tert butyl 2 methyl 2S 4 4 difluoropyrrolidine 1 2 dicarboxylate 2R 1 tert butoxy carbonyl 4 4 difluoro 2 methylpyrrolidine 2 carboxylic acid 2S 4 4 difluoro 1 methylpyrrolidin 2 yl methanamine 5 bromo 7 fluorobenzofuran 1 1 bis propan 2 yl 3 fluorocyclobutane 1 1 dicarboxylate 2 Fluoropyridine 4 boronic acid

6 bromo 4 fluorobenzo b thiophene 2 carboxylic acid 3 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 1 tert butoxycarbonylamino 4 4 difluoro cyclohexanecarboxylic acid 6 fluorobenzofuran 2 carboxylic acid 5 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 6 difluoro 4 methoxyphenyl boronic acid 3 trifluoromethyl imidazo 1 5 a pyrazine 1R 2R 2 fluorocyclopropanecarboxylic acid 3 3 Difluoropropanoic acid 7 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 6 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 7 fluorobenzofuran 2 carboxylic acid 4 cyano 3 5 difluorophenyl boronic acid 7 trifluoromethyl indolizine 1 carbaldehyde 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl 1h indole 1 tert butoxy carbonyl 4 4 difluoropyrrolidine 3 carboxylic acid 1 2 fluoroethyl cyclobutane 1 carboxylic acid 6 trifluoromethoxy pyridine 2 carboxylic acid 1 2 Dibromo 3 3 3 trifluoropropane 3 chloro 5 fluoro 4 methoxyphenyl boronic acid 3 chloro 5 fluoro 4 hydroxyphenyl boronic acid 2 4 fluorophenyl 5 5 iodo 2 methylphenyl methyl thiophene 2 fluoro 4 methoxyphenyl boronic acid 6 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1h indole 3 3 3 Trifluoropropionic acid 7 fluoroquinolin 6 yl methanol 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 tosyl 5 trifluoromethyl 1h pyrrolo 2 3 b pyridine 4 Nitro Benzenesulfonyl fluoride

3 5 Difluoro 4 trifluoromethyl acetophenone 3 fluorocyclobutane 1 1 dicarboxylic acid 6 bromo 7 fluorobenzofuran 1S 3 3 difluorocyclopentane 1 carboxylic acid 1 methyl 3 trifluoromethyl cyclobutan 1 ol 1 methyl 3 trifluoromethyl cyclobutane 1 carboxylic acid 5 Fluoro 2 pyridinecarboxylic acid 2 3 fluoro 1 methylcyclobutyl acetonitrile 2 6 trifluoromethyl pyridin 2 yl acetic acid 1 1 1 2 2 Pentafluoro 4 iodobutane 3 3 difluorocyclobutan 1 one 5 bromo 2 chloro 4 fluoropyridine 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 4 trifluoromethyl pyridine 3 carboxylic acid 5 nitro 3 trifluoromethyl 1H pyrrolo 2 3 b pyridine 4 chloro 5 trifluoromethyl 7H pyrrolo 2 3 d pyrimidine 5 fluoro 6 methylpyridine 2 carbaldehyde 4 5 Difluoro 2 hydroxybenzaldehyde 3R 3 fluoro 3 methylpyrrolidine 2 Fluoro 4 methoxyphenylhydrazine hydrochloride 4 4 4 Trifluorobutane 1 ol 2 3 methoxy 5 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2R 4 4 difluoropyrrolidine 2 carboxylic acid hydrochloride 1 methyl 5 trifluoromethyl 1H indole 2 carboxylic acid 5 Bromo 2 bromomethyl 1 3 difluorobenzene 2 2 2 Trifluoro 1 4 hydroxyphenyl ethanone 4 4 bis trifluoromethyl 2 2 bipyridine 1S 3 3 difluorocyclopentan 1 amine hydrochloride 2 Bromo 6 fluorobenzaldehyde

1H Indole 7 carbonitrile 2 4 Chlorophenyl acetyl benzoic acid 2 Chloro 4 6 dimethoxy 1 3 5 triazine 3 4 Diethoxyphenyl acetic Acid 4 fluoro 2 methoxypyridine 3 carbonitrile 4 Chloro 3 5 dinitrobenzotrifluoride 4 Amino 3 trifluoromethyl benzonitrile 7R 2 chloro 8 3 3 difluorocyclopentyl 7 ethyl 5 methyl 5 6 7 8 tetrahydropteridin 6 one 4 Fluoro 5 methyl 2 nitrophenol 3 4 Difluorophenol 2 chloro 5 trifluoromethyl pyridin 4 amine 1 Cyclopropyl 6 fluoro 7 chloro 4 oxo 1 4 dihydro 1 8 naphthyridine 3 carboxylic acid 2 Bromo 4 trifluoromethyl pyridine 3 4 Difluoroanisole 1R 3 3 difluorocyclopentane 1 carboxylic acid 2 2 Nitro 4 trifluoromethylbenzoyl cyclohexane 1 3 dione 1S 2R 2 fluorocyclopentan 1 amine hydrochloride 6 Fluoro 4 nitro 3H isobenzofuran 1 one 3 benzyloxy methyl 2 fluorocyclobutan 1 one 2 3 3 difluorocyclobutylidene acetonitrile 4 piperidinol 5 fluoro 3 3 dimethyl hydrochloride 1 1 4r 5s rel 7 fluoro 3 4 dihydroquinazolin 4 one 1 1 methylpiperidin 4 yl 1H pyrazol 4 amine 2 benzofuran 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 5 3 chlorophenyl N 4 morpholinomethyl phenyl furan 2 carboxamide 3 amino 2 chloroisonicotinic acid 3 bromo 5 chloro 1 2 4 triazolo 4 3 a pyridine 2 4 diethoxyphenyl boronic acid 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Amino 6 chlorobenzonitrile