5 Bromo 2 fluoroanisole 3 4 difluoro 2 methoxyphenylboronic acid 1 tert Butyl 3 methyl 1H pyrazole 5 carboxylic acid 2 imidazo 1 2 a pyridin 2 ylacetic acid 4 diethylamino methyl aniline 2 4 methoxyphenyl 6 oxo 1H pyrimidine 5 carboxylic acid 2 4 hydroxyphenyl benzo b thiophen 6 ol 3 amino 2 chloroisonicotinic acid 2 2 Dimethyltetrahydropyran 4 one 6 1H benzo d 1 2 3 triazol 5 yl methyl 1H benzo d 1 2 3 triazole 4 1 3 2 dioxaborinan 2 yl benzoic acid 1 6 chloro 1H pyrrolo 3 2 c pyridin 3 yl ethanone 4 Methyl 1H pyrrolo 2 3 b pyridine 2 iodophenylboronic acid 4 BroMo 2 Methyl 1H indole 6 carboxylic acid Methyl ester 7 chlorobenzo b thiophene 2 carboxylic acid 4 methylamino methyl phenylboronic acid 6 Chloroquinoline 8 Carboxylic Acid 3 chloro 6 methoxypyridin 2 amine 3 5 dimethoxypyridin 4 amine 1 prop 2 ynyl piperazine 3 amino 5 bromo 2 hydroxybenzonitrile 3 bromo 2H indazol 6 amine 2 5 dichlorothiophene 3 carbaldehyde 2 6 dibromo 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 6 8 difluoro 2 methylquinolin 4 yl 3 4 dimethylamino phenyl urea 3 4 chlorophenyl piperazin 2 one 2 4 bromophenyl triphenylene 4 methylsulfonyl piperidine 4 Methoxy 3 nitrobenzotrifluoride

4 methyl 3 phenylpiperazin 2 one 1 prop 2 ynyl pyrrolidine 6 Phenylnicotinaldehyde 3 trifluoromethyl 1H pyrazolo 3 4 b pyridine 6 bromobenzo d oxazol 2 amine 7 mercapto 4 methyl 2H chromen 2 one 2 6 bromopyridin 2 yl propan 2 ol 4 5 4 Pentyloxyphenyl isoxazol 3 yl benzoic acid 1 2 chloroethyl 4 methylpiperazine dihydrochloride 2 7 Chloro 1 8 naphthyridin 2 yl 3 2 1 4 dioxa 8 azaspiro 4 5 decan 8 yl 2 oxoethyl 3H isoindol 1 one 7 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H indole 1 4 Amino 3 5 dibromophenyl 2 bromoethanone 6 Chloro 4 hydroxyquinoline 3 carboxylic acid 1 2 3 4 tetrahydroisoquinolin 7 amine 7 4 chlorobutoxy 3 4 dihydroquinolin 2 1H one 2 trifluoromethyl pyridin 4 yl methanamine 5 bromo 2 1H pyrazol 3 yl pyridine 2 chloro 6 trifluoromethoxy pyridine 3 carboxylic acid 6 methoxy 1H quinolin 2 one 1 Phenyl 2 pyridin 2 ylethanone 4 bromo 2 3 dimethoxybenzaldehyde 3 3 difluoroazetidine hydrochloride 6 chloro 2 trifluoromethyl 1H quinolin 4 one 4 bromo 2 fluoro 3 methoxybenzoic acid 5 6 dimethylpyrazin 2 ol 4 Fluoro 1 iodo 2 methylbenzene 3 bromopyrazine 2 carbonitrile 1 fluoro 4 4 fluorophenyl phenylphosphoryl benzene 2 bromonaphthalen 1 ol 2 formyl 5 methylphenylboronic acid

5 Cyano 3 pyridinylboronic acid 1 phenylcyclohexane 1 carbonitrile 5 ethoxy 1H benzo d imidazole 2 3H thione 5 methoxycarbonylthiophene 2 carboxylic acid 2 3 DIPHENYLACRYLONITRILE 4 fluoronaphthalen 1 amine 7 methoxybenzo b thiophene 2 carboxylic acid 3 AMINO 6 IODOPYRAZINE 2 CARBOXYLIC ACID 2 methoxy 6 methylbenzaldehyde 1 isopropyl 1H pyrazol 4 amine 2 cyclohexyl N 1 isopropylpiperidin 4 yl 6 methoxy 7 3 pyrrolidin 1 yl propoxy quinazolin 4 amine 4 methylsulfonyl 3 nitrobenzoic acid 6 Bromo 4 chloroquinoline 4 amino 2 4 4 dimethyl 2 oxoimidazolidin 1 yl N 3 trifluoromethyl phenyl pyrimidine 5 carboxamide 1 4 4 3 4 dichloro 2 fluorophenyl amino 7 methoxyquinazolin 6 yl oxy piperidin 1 yl prop 2 en 1 one 2 4 6 7 dimethoxyquinazolin 4 yl oxy phenyl N 1 isopropyl 1H pyrazol 4 yl acetamide 2 Iodo 6 methoxybenzoic acid 5 ETHYLIDENE 2 NORBORNENE 3 6 7 dimethoxyquinazolin 4 yl amino phenol 2 bromo 4 6 7 dimethoxyquinazolin 4 yl amino phenol 1 2 Dimyristoyl sn glycero 3 phosphocholine 1 2 Epoxypentane 1 2 4 bromophenoxy ethyl pyrrolidine 1 tert butyl 3 p tolyl 1H pyrazolo 3 4 d pyrimidin 4 amine 2 3 4 tri O acetyl D fucopyranosyl bromide 6 4 3 methylsulfonyl benzyl amino 5 trifluoromethyl pyrimidin 2 yl amino 3 4 dihydroquinolin 2 1H one 4 CHLOROBENZOYLACETONITRILE 3 3 fluoro 4 morpholin 4 ylphenyl 2 oxo 1 3 oxazolidin 5 yl methyl methanesulfonate 3 3 5 Difluorophenyl propionic acid 5 AZABENZIMIDAZOLE

1 cyclopentyl N 4 6 dimethyl 2 oxo 1 2 dihydropyridin 3 yl methyl 6 4 morpholinomethyl phenyl 1H indazole 4 carboxamide 4 Hydroxy 6 methylquinoline 3 carboxylic acid 4 cyanophenyl 4 methylbenzoate 2 4 5 ethylpyrimidin 4 yl piperazin 1 yl methyl 5 trifluoromethyl 1H benzo d imidazole 4 2 6 difluoro 4 3 1 piperidin 4 yl 1H pyrazol 4 yl quinoxalin 5 yl benzyl morpholine 1 4 3 amino 1H indazol 4 yl phenyl 3 2 fluoro 5 methylphenyl urea 6 1H indazol 6 yl N 4 morpholinophenyl imidazo 1 2 a pyrazin 8 amine 3 methylsulfonylbenzonitrile 4 6 7 dimethoxyquinazolin 4 yl amino phenol 2 2 3 hydroxyphenyl amino pyrimidin 4 yl amino benzamide 2 IODO 3 METHYLBENZOIC ACID 4 4 aminomethyl 1 1 biphenyl 3 yl oxy pyrimidine 2 carbonitrile 2 amino 4 2 4 dichloro 5 2 pyrrolidin 1 yl ethoxy phenyl N ethylthieno 2 3 d pyrimidine 6 carboxamide 3 Methyl 6 1 methylhydrazinyl pyridazine 2 3 cyanophenyl acetic acid 5 4 2 3 dimethyl 2H indazol 6 yl methyl amino pyrimidin 2 yl amino 2 methylbenzenesulfonamide 3 6 dibromo 2 fluorophenyl boronic acid 6 2 3 dichlorophenyl N4 methylpyrimidine 2 4 diamine 2 chloro 1 3 oxazole 2 4 4 chlorobenzoyl phenoxy 2 methylpropanoate 2 hydroxyethyl trimethyl azanium 5 chloromethyl 2 methylpyridine 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 6 Chloro 5 methoxypyridin 3 amine 7 8 dihydroxy 6 methoxychromen 2 one 1H pyrrolo 2 3 b pyridin 5 ol 1 BOC 4 chloropiperidine 2 3 bromo 5 tert butyl 4 hydroxybenzylidene malononitrile 2 5 dioxopyrrolidin 1 yl 6 2 5 dioxo 2 5 dihydro 1H pyrrol 1 yl hexanoate 6 fluoro 1H pyrrolo 2 3 b pyridine 1 ethylpiperidin 3 yl 2 2 diphenylacetate