5 Chloro 2 fluoro 4 iodopyridine 5 Chloro 2 fluoro 3 hydroxypyridine 5 Bromo 2 fluoro 3 nitropyridine 2 Fluoro 3 nitro 4 picoline 3 Bromo 2 fluoro 6 picoline 2 Ethoxy 5 nitropyridine 2 chloro 3 nitro 6 picoline 2 Chloro 3 hydroxy 5 picoline 2 Bromo 3 nitro 4 picoline 2 bromo 5 cyano 6 picoline 1R 2R 1 2 Diphenylethylenediamine 4 Carboxybenzylamine 1S 2S 1 2 Diphenyl 1 2 ethanediamine 3 Amino 2 bromo 5 picoline 2 Amino 5 cyano 3 picoline 2 Amino 4 ethoxypyridine 2 Amino 3 nitro 5 bromo 6 picoline 4 Methylbenzylsulfonyl chloride 3 Mercaptobenzoic acid 5 Chlorothiophene 2 sulphonyl chloride 3 Chlorothiophene 2 carboxylic acid 2 4 Dichloro 5 picoline 2 4 Dibromo 3 nitropyridine 3 Fluorothiophenol 4 Fluorothiophenol 4 7 Dimethyl 1H indene 2 3 Difluoro 5 nitropyridine 4 Bromo 2 chloro N N dimethylaniline 2 Ethoxy 4 nitroaniline 2 Iodobenzaldehyde dimethyl acetal

5 Bromo 2 fluoro 3 pyridineboronic acid 5 Chloro 2 iodoanisole 2 Chloro 5 iodoanisole 4 Chloro N N dimethylaniline 2 Bromo 4 chloro 6 methylaniline 4 Fluoro 3 iodobenzaldehyde 2 fluoro N N Dimethylaniline 4 chloro 2 trifluoromethyl phenylboronic acid 4 propoxycarbonyl phenylboronic acid 5 Methyl 2 thiophene carboxaldehyde 4 Fluoro 3 carboxyphenylboronic acid 3 chloro 4 carboxyphenylboronic acid 2 ethoxy 3 pyridineboronic acid 3 chloro 4 methylphenylboronic acid 2 hydroxymethyl phenylboronic acid 3 Cyano 4 fluorobenzenesulfonyl chloride 2 chloro 4 fluorophenylboronic acid 2 chloro 3 bromo 4 pyridineboronic acid 2 Methoxy 3 pyridineboronic acid 2 Fluoro 5 trifluoromethyl phenylboronic acid 2 fluoro 5 hydroxymethyl phenylboronic acid 4 Hydroxy 3 trifluoromethyl benzonitrile 4 Trifluoromethoxy benzonitrile 2 Chloro 3 5 dinitrobenzotrifluoride 2 Fluoro 3 nitrobenzyl alcohol 2 4 Difluoro 3 hydroxybenzoic acid 2 fluoro 3 hydroxy benzoic acid 2 Bromo 3 5 difluorobenzoic acid 2 3 Difluoro 4 bromobenzoic acid 4 Chloro 2 fluorophenylboronic acid

3 Fluoro 4 trifluoromethyl benzonitrile 4 Fluoro 3 Nitrobenzonitrile 2 Fluoro 6 nitrobenzonitrile 2 Fluoro 3 methoxybenzonitrile 2 Fluoro 5 iodobenzonitrile 4 5 Dimethoxy 2 nitrobenzonitrile 2 3 Difluoro 6 methoxybenzonitrile 4 Chloro 2 trifluoromethyl benzonitrile 2 Chloro 3 methylbenzonitrile 2 Chloro 4 hydroxybenzonitrile 2 Amino 4 5 dichlorobenzoic acid 4 Methoxy 3 trifluoromethyl benzyl bromide 2 Methoxybenzyl chloride 3 Trifluoromethoxy nitrobenzene 2 Trifluoromethoxy nitrobenzene 5 Cyano 2 fluorobenzoic acid 4 Cyano 2 6 difluorobenzoic acid 4 Trifluoromethoxy benzoic acid 2 Amino 5 bromobenzonitrile 2 4 5 Trifluoro 3 ethoxy benzoic acid 3 4 5 6 Tetrafluorophthalonitrile 3 5 difluoro 4 methylbenzonitrile 4 5 Difluoroindole 2 Methyl 3 4 6 trifluorobenzoic acid 3 bromo 2 chloro 6 fluorotoluene 2 Methyl 4 trifluoromethyl aniline 2 Amino 3 5 dibromotoluene 1 2 4 5 Tetrabromobenzene 2 6 Difluoro 4 iodoaniline 2 4 Dichloro 5 methoxyaniline

3 5 dichloro 4 fluoronitrobenzene 1 2 Diamino 3 methyl 4 fluorobenzene 3 Amino 5 cyanobenzeneboronic acid hydrochloride 5 chloro 2 nitro 4 trifluoromethoxy aniline 2 6 Dichlorophenylacetic acid 2 4 6 trifluoroacetophenone 4 methoxy 2 nitrobenzoic acid 3 Trifluoromethyl phenylacetonitrile 4 Carboxy 2 6 difluorobenzaldehyde 2 Bromo 6 nitrobenzaldehyde 3 Fluorophenylacetonitrile 4 Fluoro 2 trifluoromethyl phenol 3 Fluorocatechol 2 Bromo 5 methylanisole 3 Bromo 2 fluoroanisole 2 Fluoro 3 methylphenol 2 3 Dimethylanisole 1 2 Difluoro 3 methoxy 4 nitrobenzene 2 4 Pyridinyl benzaldehyde 3 chloro 4 fluorocinnamic acid 3 Hydroxy 2 pyridinemethanol hydrochloride 2 Pyridineboronic acid 4 Bromothiophenol 4 Bromo Thiazole 2 3 Dihydroxynaphthalene 6 sulfonic acid sodium salt 2 Iodophenol 4 4 dichlorobenzil 1 Ethyl 4 iodobenzene 3 3 Pyridyl acrylic acid 4 Ethylphenol