2 Trifluoromethyl benzaldehyde 2 Fluoro 5 methoxyaniline 2 Chloro 5 fluoro 3 nitropyridine 1S 2S 3R 5S Pinanediol 2 Nitro 3 methylbenzoic acid 2 Chloro 4 methylpyridine 3 carbonitrile 4 Pentynoic acid 4 Hydroxymethyl phenylboronic acid 9 3 Bromophenyl 10 2 naphthyl anthracene 3 Bromo 2 fluoroanisole 2 6 Difluorobenzotrifluoride 2 Chloro 6 cyanopyridine 4 5 Difluorophthalic acid 3 Fluoro 4 methoxyaniline 5 Methyl 1H pyrrolo 2 3 b pyridine 2 2 Diphenylglycine 2 Amino 4 5 difluorobenzoic acid 5 Bromo 2 chlorophenol 1 N Boc pyrrolidin 2 ylboronic acid 4 2 Aminoethyl tetrahydropyran 1 hydroxymethyl cyclopropaneactetonitrile 3 Formylphenylboronic acid 3 Fluoro 4 trifluoromethoxy aniline 1 Bromo 3 chloro 2 5 difluorobenzene 3 nitro 4 trifluoromethyl aniline 1 Methylcyclopropene 2 4 5 trifluorophenylacetic acid 2 Chloro 5 nitropyridine 4 amine 5 Methyl 3 2H pyridazinone 2 Chloro 5 cyanomethyl pyridine

3 Aminopropylphosphate 6 Chloro 1H pyrrolo 2 3 b pyridin 2 3H one 4 Bromobenzamidine 1 2 4 5 Tetrafluoro 3 nitrobenzene 4 Methoxy 2 trifluoromethyl benzaldehyde 4 Bromo 3 5 dimethylphenol 3 Chloro 2 iodoaniline 3 Nitrophthalic acid 2 Nitro 4 trifluoromethyl aniline 2 4 Dibromo 3 fluoro nitrobenzene 3 chloro 4 fluorocinnamic acid 2 Chloro 4 methylaniline 2 Amino 4 bromopyridine 3 Bromo 4 fluorotoluene 3 Fluoro 2 nitropyridine 3 4 Dimethylphenylaceticacid 4 chloro 3 nitrophenol 2 4 Difluoro 3 trifluoromethyl benzoic acid 5 Cyano 2 fluoro 3 picoline 4 chloro 2 trifluoromethyl phenylboronic acid 5 Fluoro 2 methylbenzoic acid 5 Bromo 2 chloropyrimidine 2 Pyridineethanol 1 Bromo 2 chloro 4 iodobenzene 3 Fluoro 4 methyl 5 hydroxybenzoic acid 2 Methyl 4 trifluoromethyl aniline 4 Bromo 3 methylthiophenecarboxylic acid 4 Bromo Thiazole 4 Bromo 3 fluorotoluene 4 Amino 2 chloropyridine

3 Chloro 2 fluoroaniline 5 Chloro 1H pyrrolo 2 3 b pyridine 2 Chloro 4 trifluoromethyl aniline 5 Bromo 3 methyl 1H indazole 6 Chloromethyl uracil 5 Chloro 3 n methoxy carbonyl methyl sulfamoyl 2 thiophene carboxylic acid methyl ester 3 4 Dihydro 7 methoxy 4 oxoquinazolin 6 yl acetate 3 Cyclopropyl 3 oxopropanenitrile 6 Trifluoromethyl indole 3 Chloro 4 bromotoluene 2R 2 Aminopropanamide hydrochloride 2 Aminodiphenyl 1 Bromonapthalene 2 Amino 2 fluoro 5 bromobenzophenone 3 Hydroxypyrazine 2 carboxylic acid 2 Chloro 6 phenylnicotinonitrile 2 Fluoro 6 nitrobenzonitrile 1 2 Dimethylaminoethyl 1H Tetrazole 5 Thiol 1 Aminocyclopropane 1 carboxylic acid ethyl ester hydrochloride 3 Amino 4 picoline 2 Fluoro 5 hydroxy 3 picoline 1 4 5 8 tetrahydro 2 7 dimethoxy Naphthalene 5 Chloro 3 fluorobenzene 1 2 diol 5 Chloro 2 fluoro 3 hydroxypyridine 2 amino 3 chloro 4 fluoronitrobenzene 5 bromofuran 2 carbonyl chloride 1 Aminomethyl adamantane 3 4 Difluorotoluene 2 6 10 Trimethylundeca 5 9 dienal Cidalor 3 Isobutylglutaric acid

2 6 Difluorobenzyl alcohol 2 Isopropoxy 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Amino 3 fluoropyridine 3 S 1 Carbamoyl 1 1 diphenylmethyl pyrrolidine L tartrate 3R 4R 1 Benzyl N 4 dimethylpiperidin 3 amine dihydrochloride 2 4 Dichloro 7H pyrrolo 2 3 d pyrimidine 2 Ethylbenzaldehyde 1H Pyrazole 2 Amino 3 5 dibromotoluene 2 3 Pyrazinedicarboxylic anhydride 3 Amino 4 iodopyridine 2 Chloro 4 fluorobenzonitrile 1 1 1 Trifluoro 3 chloropropane 3 Fluoro 4 trifluoromethyl benzonitrile 2 Chloropyridine 3 5 Dimethoxyaniline 3 Cyclohexene 1 carboxylic acid 5 Bromo 2 fluoro 3 nitropyridine 5 Bromo 2 chlorobenzoic acid 5 Bromo 1 2 dimethyl 3 nitrobenzene 1 Benzosuberone 3 Bromo 2 fluoropyridine 3 5 Dimethylphenylboronic acid 2 4 Dibromotoluene 5 Amino 4 chloro 2 methylphenol 2 Bromo 3 5 dimethoxy 1 fluorobenzene 3 Chloro N methylaniline 4 Fluoro 4 methylbenzophenone 3 Trifluoromethyl 5 6 7 8 tetrahydro 1 2 4 triazolo 4 3 a pyrazine hydrochloride 5 Methylpyrazin 2 amine