3 Fluoro 2 methoxybenzoic acid 3 methoxy 5 methylsulfonyl aniline 2 Trifluoromethyl pyridine 3 Bromo 6 iodo o xylene 2 4 Bis trifluoromethyl acetophenone 2 5 Dichlorobenzaldehyde 4 Iodo 2 trifluoromethoxy aniline 5 Fluoro 2 trifluoromethyl benzoic acid 4 Difluoromethoxy benzyl bromide 3 4 Methylenedioxybenzyl alcohol 2 6 Difluorobenzoic acid 2 Chloroethyl benzoate 3 4 Difluorophenylacetic acid 3 Nitrophthalic acid 2 Amino 4 chloro 5 iodopyridine 1 Boc 3 hydroxymethyl pyrrolidine 3 Amino 5 chlorobenzotrifluoride 2 6 Difluoro 4 iodoaniline 3 Bromo 2 fluoro 6 picoline 3 bromo 5 fluorobenzaldehyde 1 1 1 trifluoropentan 2 one 4 4 Dihydroxy 3 3 diformylbiphenyl 4 4 difluoro octahydrocyclopenta c pyrrole 2 3 chloro 4 fluorophenyl 4 4 dimethyl 1 2 3 4 tetrahydroquinoline 6 carboxylic acid 3 3 difluorocyclopentane 1 carboxylic acid 6 trifluoromethyl 2 pyridyl methanol 6 boc 4 4 difluoro 2 6 diazabicyclo 3 2 0 heptane 5 Chloro 2 fluorophenylhydrazine HCl 5 Bromothiophene 3 carboxylic acid 5 bromo 1H pyrazolo 3 4 b pyridin 3 amine

3 3 difluoro 2 methylazetidine hydrochloride 3S 4R 3 fluoro 4 methoxypiperidine 4 chloro 6 fluoro 1 7 naphthyridine 3 carbonitrile 5 trimethylsilyl thiophen 2 ylboronic acid 4 bromopyridin 3 ol 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 7 carboxylic acid 2 4 6 trifluoro 3 methoxyphenylboronic acid 3 chloro 4 iodophenol 2 6 dimethoxyphenyl boronic acid 2 Fluoro 4 methoxybenzoic acid 3 Iodobenzotrifluoride 4 Chloro 2 5 difluorobromobenzene 2 6 bis trifluoromethyl aniline 4 Tert butylpyridine 2 hydroxy 9H thioxanthen 9 one 2 Butene 1 4 diol 5 Bromo 2 fluoro m xylene 4 Iodo 1 2 dimethoxybenzene 4 Benzyloxy 3 methoxyacetophenone 2 4 Dichlorobenzaldehyde 4 Iodo 2 nitroaniline 4 Methoxybenzyl alcohol 2 6 Difluorophenylacetic acid 4 Fluoro 3 trifluoromethyl benzoic acid 3 Difluoromethoxy benzyl bromide 2 4 Difluoro 3 5 dimethoxybenzoic acid 3 Chlorophthalic anhydride 2 5 Difluorobenzoic acid 2 3 Difluorochlorobenzene 5 amino 3 bromo 2 fluoropyridine

2 3 Pyrazinedicarboxylic acid 4 Bromo 2 8 bis trifluoromethyl quinoline 3 Amino 4 iodobenzotrifluoride 1 1 1 3 3 Pentafluorobutane 5 methoxy 2 phenyl 1H indole 2 Bromo 5 fluorobenzaldehyde 2 Amino 3 trifluoromethyl benzoic acid 4 chloro 3 5 difluoropyridine hydrochloride 3r 4s rel 4 fluoro 3 piperidinol hydrochloride 5 bromo 4 trifluoromethyl pyrimidine 3 fluoropyrazolo 1 5 a pyridin 5 amine 2 1 2 fluorophenyl methyl 1H pyrazolo 3 4 b pyridin 3 yl pyrimidine 4 5 6 triamine trihydrochloride 4 6 difluoro 1H indazole 3 carboxylic acid 1R 2S 2 amino 1 3 5 bis trifluoromethyl phenyl propan 1 ol 5 chloro 3 trifluoromethyl pyridin 2 amine 4 chloro 5 fluoro 1H pyrrolo 2 3 b pyridine 2 chloro 5 6 7 8 tetrahydroquinoxaline 3 cyano 4 propoxyphenylboronic acid 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl benzaldehyde 2 bromopyrimidine 4 carbonitrile 4 chloro 2 methoxyphenyl boronic acid 2 fluoro 4 iodo 6 methoxypyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 fluoro 1H pyrazolo 3 4 b pyridin 3 amine 4 methoxypyrimidin 2 amine 2 Fluoro 3 chloro phenylhydrazine HCl 3 4 5 Trichlorobenzotrifluoride 4 Chloro 2 6 dibromonitrobenzene 4 Bromo 2 fluoroacetanilide 8 Chloro 6 trifluoromethyl imidazo 1 2 a pyridine 2 carboxylic acid hydrate

5 Bromo 2 chloro m xylene 3 Fluoro 1 2 diethoxybenzene 2 Iodobenzyl alcohol 2 Iodo 5 nitroaniline 2 3 Dichlorobenzaldehyde 5 Amino 2 fluoroacetophenone 3 5 Difluoro 2 methoxybenzyl bromide 4 Fluoro 2 trifluoromethyl benzoic acid 2 4 Difluorophenylacetic acid 2 4 Difluorobenzoic Acid 3 5 Bis trifluoromethyl benzyl alcohol 2 4 Dichloro 5 methoxyaniline 2 Ethoxy 5 nitropyridine 1 Methylpyrrole 2 acetic acid 2 4 Chlorophenyl 2 Oxoacetaldehyde 2 Bromo 3 fluorobenzaldehyde 2 Chloro 1 1 difluoroethane 3 6 dichloro 4 carboxyphthalic anhydride 3 fluoro 3 methoxymethyl pyrrolidine hydrochloride 3 3 difluoropiperidin 4 ol hydrochloride 4 chloro 3 5 difluoropyridine 4 fluoro 3 methoxybenzaldehyde 2 1 2 fluorophenyl methyl 1h pyrazolo 3 4 b pyridin 3 yl pyrimidine 4 5 6 triamine 5 amino 3 3 difluoro 2 3 dihydro 1H indol 2 one 3S 4R 4 fluoropiperidin 3 ol 3 bromo 1 1 difluorocyclopentane 5 fluoro 1H 2H 3H pyrrolo 2 3 b pyridin 2 one 6 chloro 3 iodo 1H pyrazolo 4 3 c pyridine 7 chloro 3 4 dihydro 2H benzo b 1 4 oxazine 2 2 hydroxyethoxy ethyl 2 3 trifluoromethyl phenyl amino benzoate