4 FLUORO 3 ISOPROPYL BENZYLAMINE 3 AMINO 1 3 CHLORO 4 FLUORO BENZYL PYRROLIDIN 2 ONE 4 BROMO 1 2 FLUOROPHENYL 3 METHYL 1H PYRAZOL 5 AMINE 1 benzyl 3 ethyl 4 4 difluoropiperidine 1 3 dicarboxylate 4 fluoropiperidin 3 yl methanamine 3 fluoropiperidin 4 yl methanamine 7 4 FLUORO PHENYL 5 METHYL 4 OXO 4 5 DIHYDRO THIENO 3 4 C PYRIDINE 6 CARBOXYLIC ACID 6 TRIFLUOROMETHYL PYRIDIN 2 YL METHANOL 2 CHLORO 4 2 4 DIFLUORO PHENYL 6 7 DIHYDRO 5H 1 PYRINDINE 3 fluoro tetrahydro 2H pyran 4 ol 2 CHLORO 6 FLUORO N HYDROXY BENZAMIDINE 1 BENZYL 4 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 3 BROMO 5 FLUORO 2 HYDROXYBENZALDEHYDE 4 4 difluorocyclohexyl methanol 5 4 FLUORO PHENYL 7 METHYL 8 OXO 7 8 DIHYDRO 1 7 NAPHTHYRIDINE 6 CARBALDEHYDE 9 4 4 aminopiperidin 1 yl butyl N 2 2 2 trifluoroethyl 9H fluorene 9 carboxamide 8 AMINO 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 1 PHENYLMETHYL 4 TRIFLUOROMETHYL TRANS 3 PYRROLIDINECARBOXYLIC ACID 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDIN 3 YL METHANOL 2S 4R 1 tert butyl 2 methyl 4 fluoropyrrolidine 1 2 dicarboxylate 1R 1 4 FLUOROPHENYL PROPYLAMINE 5 FLUORO 3 3 DIMETHYL 2 3 DIHYDRO 1H INDOLE 6 CHLORO 3 TRIFLUOROMETHYL 1 2 4 TRIAZOLO 3 4 A PHTHALAZINE 3 3 BROMO 4 FLUORO PHENYL 2 2 DIMETHYL CYCLOPROPANECARBOXYLIC ACID 5 FLUORO 3 METHYL BENZOFURAN 3 FLUOROSALICYLALDEHYDE 2 CHLORO 6 FLUORO 1 METHYL 1H BENZOIMIDAZOLE 2 TERT BUTYL 4 FLUOROPHENOL 4 5 6 7 TETRAHYDRO 3 TRIFLUOROMETHYL 1H INDAZOLE

4 1 1 2 2 2 PENTAFLUOROETHYL BENZOIC ACID 2 CHLORO 5 FLUORO 1 METHYL 1H BENZO D IMIDAZOLE 4 4 CHLORO BENZENESULFONYL 4 2 5 DIFLUORO PHENYL CYCLOHEXYLAMINE 2S 4S N TERT BUTOXYCARBONYL 4 TRIFLUOROMETHYLPROLINE 4 METHYL 2 4 TRIFLUOROMETHYL PHENYL PYRIDINE 2 2 difluoropropane 1 3 diol 2 BROMO 1 2 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDIN 3 YL ETHANONE 2 4 CHLOROPHENYL 2 2 DIFLUOROACETIC ACID 3 AMINO 1 4 FLUOROBENZYL PYRROLIDIN 2 ONE 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 B PYRIDAZINE 3 SULFONIC ACID AMIDE 5 TRIFLUOROMETHYL THIENO 3 2 B PYRIDINE 4 4 difluoropyrrolidine 2 carboxylic acid 3 TRIFLUOROMETHYL 1H INDAZOLE 4 BROMO 1 4 FLUORO PHENYL 1H IMIDAZOLE 2S 4S methyl 4 fluoropyrrolidine 2 carboxylate hydrochloride 5 CHLORO 3 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDIN 7 YL CARBAMIC ACID TERT BUTYL ESTER 2 AMINO 4 4 4 TRIFLUORO BUTYRIC ACID ETHYL ESTER 4 CHLOROMETHYL 2 4 FLUORO PHENYL 5 METHYL OXAZOLE 3 fluoro tetrahydropyran 4 one 2 4 FLUORO PHENYL 5 HYDROXY BENZOFURAN 3 CARBOXYLIC ACID ETHYL ESTER 3 3 DIFLUOROCYCLOBUTYL METHANOL 3 4 FLUORO PHENYL 2 PYRIDIN 4 YL ACRYLONITRILE 3 CHLORO 2 TRIFLUOROMETHYL 4 PYRIDINECARBOXYLIC ACID 6 4 FLUORO PHENYL IMIDAZO2 1 BTHIAZOLE 6 CHLORO 5 FLUORO 3 METHYL BENZO B THIOPHENE 2 BROMO 4 TRIFLUOROMETHYL NICOTINIC ACID 2 BROMO 6 TRIFLUOROMETHYL 3 TRIMETHYLSILANYL PYRIDINE 2 BROMO 3 IODO 6 TRIFLUOROMETHYL PYRIDINE 5 CHLORO 6 TRIFLUOROMETHYL PYRIDINE 2 CARBOXYLIC ACID 5 CHLORO 6 TRIFLUOROMETHYL NICOTINIC ACID

3 CHLORO 5 IODO 2 TRIFLUOROMETHYL PYRIDINE 2 BROMOMETHYL 6 TRIFLUOROMETHYL PYRIDINE 6 7 DIMETHOXY 1 2 4 TRIFLUOROMETHYL PHENYL ETHYL 1 2 3 4 TETRAHYDRO ISOQUINOLINE 3 3 TRIFLUOROMETHYL PHENOXY AZETIDINE 5 FLUORO 3 3 DIMETHYL 1 3 DIHYDRO INDOL 2 ONE 1 BROMOMETHYL 3 TRIFLUOROMETHYLSULFONYL BENZENE 3 AMINO 4 FLUORO 6 MORPHOLIN 4 YL BENZO B THIOPHENE 2 CARBOXYLIC ACID AMIDE 3 CHLORO 5 FLUORO 2 HYDROXYBENZALDEHYDE 2 3 FLUORO 4 METHYL PHENYL 1 1 DIMETHYL ETHYLAMINE 4 FLUORO 3 ISOPROPYLBENZOIC ACID 2 DIETHYLAMINO 5 2 2 2 TRIFLUORO ETHYL PYRIMIDIN 4 OL 1 4 FLUORO BENZYL 4 HYDROXY 1H PYRROLO 2 3 C PYRIDINE 5 CARBOXYLIC ACID METHYL ESTER 2 THIAZOLAMINE 4 5 FLUORO 1H PYRROLO 2 3 B PYRIDIN 3 YL 2 AMINO 6 FLUORO NICOTINAMIDE 3 FLUORO 2 HYDROXY 6 METHYL BENZALDEHYDE 2 BROMO 4 TRIFLUOROMETHYL BIPHENYL 4 YL ACETIC ACID METHYL ESTER 8 METHYL 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 2 1 AMINO 2 2 2 TRIFLUORO ETHYL 3 4 DIFLUORO PHENYLAMINE 4 S 1 AMINO 2 2 2 TRIFLUORO ETHYL BENZOIC ACID ETHYL ESTER 1 4 AMINOMETHYL PHENYL 2 2 2 TRIFLUORO ETHYL CARBAMIC ACID TERT BUTYL ESTER 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 2 1 F PYRIDAZINE 3 CARBOXYLIC ACID 2 2 2 TRIFLUORO 1 2 4 6 TRICHLORO PHENYL ETHANONE 5 FLUORO 4 3 ISOPROPYL 2 METHYL 3H IMIDAZOL 4 YL PYRIMIDIN 2 YLAMINE 3 3 TRIFLUOROMETHYL PHENYL PIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 9 ETHOXYCARBONYLMETHYL 6 FLUORO 2 3 4 9 TETRAHYDRO 1H CARBAZOLE 3 CARBOXYLIC ACID 2 AMINO 4 2 TRIFLUOROMETHYL PHENYL THIOPHENE 3 CARBOXYLIC ACID ETHYL ESTER 3 TRIFLUOROMETHYL 6 7 DIHYDRO 5H PYRROLO 3 4 B PYRIDINE 5 IODO 3 TRIFLUOROMETHYL PYRIDIN 2 YLAMINE 2 2 2 2 TRIFLUORO ETHOXY 6 7 DIHYDRO 5H PYRROLO 3 4 D PYRIMIDINE 3 2 FLUOROPHENOXY AZETIDINE

2 TERT BUTYL 4 4 FLUORO PHENYL 5 6 7 8 TETRAHYDRO PYRIDO 4 3 D PYRIMIDINE 2 FLUOROPHENACYLAMINE HYDROCHLORIDE 4 4 difluorocyclohexanecarboxamide 3 FLUOROPHENACYLAMINE HYDROCHLORIDE 3 BROMO 2 METHYL 7 TRIFLUOROMETHYL 4 5 6 7 TETRAHYDROPYRAZOLO 1 5 A PYRIMIDINE 2 TRIFLUOROMETHYL QUINOLINE 6 CARBOXYLIC ACID 6 TRIFLUOROMETHYL PYRIDINE 2 4 DIOL 3 NITRO 6 TRIFLUOROMETHYL PYRIDINE 2 4 DIOL 3 4 FLUORO 2 METHYL PHENOXY AZETIDINE 2 2 2 2 TRIFLUORO 1 1 DIMETHYL ETHYL QUINOLINE 6 CARBOXYLIC ACID 4 METHYL 7 TRIFLUOROMETHYL QUINOLINE 3 CARBOXYLIC ACID ETHYL ESTER 7 FLUORO 5 TRIFLUOROMETHYL ISOQUINOLIN 3 YLAMINE 5 FLUORO 8 METHYL ISOQUINOLIN 3 YLAMINE 1 1 1 trifluoro 4 iodobutane 3 3 3 Trifluoropropylamine 2 2 bis trifluoromethyl oxirane 4 Bromo 3 3 4 4 tetrafluorobutan 1 ol 4 4 4 trifluoro 1 4 methoxyphenyl butane 1 3 dione 6 FLUORO 7 TRIFLUOROMETHYL QUINOLINE 3 CARBOXYLIC ACID 4 BROMO 6 CHLORO 7 TRIFLUOROMETHYL QUINOLINE 3 CARBOXYLIC ACID ETHYL ESTER 6 CHLORO 7 TRIFLUOROMETHYL QUINOLINE 3 CARBOXYLIC ACID 4 CHLORO 6 METHOXY 2 TRIFLUOROMETHYL QUINOLINE 3 CARBONITRILE 3 4 FLUORO BENZYL FURO 3 4 B PYRIDINE 5 7 DIONE 1 tert butyl 4 methyl 3 fluoropiperidine 1 4 dicarboxylate 4 4 difluoropiperidin 3 amine hydrochloride dihydrochloride 4 4 4 Trifluorobutyronitrile 3 Indoleglyoxylic acid 1 Benzyl 3 indolylaldehyde 1 Boc 4 carboxyindole 4 methoxy 1 Methylindole