3 AMINO 5 FLUORO 3 4 DIHYDRO 1H QUINOLIN 2 ONE 2 Fluoro 6 trifluoromethyl phenylboronic acid pinacol ester 1 ETHYL PIPERIDINE 2 CARBOXYLIC ACID 2 4 Bromonaphthalen 1 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 Bromo 2 6 difluorophenyl 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 Iso propoxyphenylboronic acid pinacol ester 4 2 TRIFLUOROMETHYL PHENYL 4 PIPERIDINOL 4 3 CHLOROPHENYL PIPERIDIN 4 OL 2 6 Dimethyl 4 cyanophenylboronic acid pinacol ester 3 Formyl 4 methoxyphenylboronic acid pinacol ester 3 3 PIPERIDINE PROPIONIC ACID HYDROCHLORIDE 2 3 5 Dichloro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 3 METHYLPHENYL PIPERIDIN 4 OL 2 5 Bromo 2 fluoro 4 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Chloro 4 propoxyphenylboronic acid pinacol ester 3 AMINO 6 FLUORO 3 4 DIHYDRO 1H QUINOLIN 2 ONE 3 Chloro 4 methylthio phenylboronic acid pinacol ester 3 AMINO 7 TRIFLUOROMETHYL 3 4 DIHYDRO 1H QUINOLIN 2 ONE 2 Fluoro 5 methoxyphenylboronic acid pinacol ester 3 TRIFLUOROMETHYL 1 4 5 7 TETRAHYDRO PYRAZOLO 3 4 C PYRIDINE 6 CARBOXYLIC ACID TERT BUTYL ESTER 2 5 Dimethoxyphenylboronic acid pinacol ester 4 TRIFLUOROMETHYL 1 4 6 7 TETRAHYDRO IMIDAZO 4 5 C PYRIDINE 5 CARBOXYLIC ACID TERT BUTYL ESTER 5 Fluoro 2 methylthio phenylboronic acid pinacol ester 3 5 Difluoro 4 methylphenylboronic acid 1H INDAZOLE 5 CHLORO 1 METHYL 3 4 PIPERIDINYL 1 ISOPROPYLPIPERIDIN 4 YL ACETIC ACID 4 Methyl 3 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 Bromo 3 hydroxyphenylboronic acid 6 7 DIMETHOXY 1 2 2 3 4 TRIFLUORO PHENYL ETHYL 1 2 3 4 TETRAHYDRO ISOQUINOLINE 1 2 2 6 DIFLUORO PHENYL ETHYL 6 7 DIMETHOXY 1 2 3 4 TETRAHYDRO ISOQUINOLINE

2 Methyl 6 methylthio 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 Fluoro 2 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 7 DIMETHOXY 1 2 2 TRIFLUOROMETHOXY PHENYL ETHYL 1 2 3 4 TETRAHYDRO ISOQUINOLINE 5 Chloro 2 ethoxyphenylboronic acid pinacol ester 2 Chloro 6 isopropylpyridine 3 boronic acid pinacol ester 2 PIPERIDIN 4 YL BENZOIC ACID 2 Benzyloxy 5 methylphenylboronic acid pinacol ester 2 Chloro 6 fluoro 3 methylphenylboronic acid pinacol ester 4 Fluoro 3 trifluoromethyl phenylboronic acid pinacol ester 2 Chloro 5 fluoropyridine 4 boronic acid pinacol ester 2 PIPERIDINECARBOXYLIC ACID 1 2 AMINO 5 IMINO NITROAMINO METHYL AMINO 1 OXOPENTYL 4 METHYL ETHYL ESTER 2R 1 S 2ALPHAR 4BETA 3 4 Dichloro 5 methylphenylboronic acid 4 AMINOPHENYL 1 PHENETHYLPIPERIDINE 3 4 Dichloro 5 methylphenylphenylboronic acid pinacol ester 4 2 FLUOROPHENYL 4 PIPERIDINECARBOXYLIC ACID ETHYL ESTER 2 Fluoro 6 methylsulfanyl benzoic acid 4 3 TRIFLUOROMETHYL PHENYL 4 PIPERIDINECARBOXYLIC ACID ETHYL ESTER HYDROCHLORIDE 1 METHYL 3 4 DIHYDRO 2H SPIRO ISOQUINOLINE 1 4 PIPERIDINE 5 Chloro 2 fluoropyridine 4 boronic acid pinacol ester 5 Chloro 2 ethoxypyridine 3 boronic acid 3 Chloro 2 methylphenyboronic acid pinacol ester 5 Ethoxy 2 methylphenylboronic acid pinacol ester 2 Bromo 4 5 difluorophenylboronic acid pinacol ester 4 2 METHOXYPHENYL PIPERIDIN 4 OL 4 2 CHLORO PHENYL PIPERIDINE HYDROCHLORIDE 2 5 Difluoro 4 methylsulfanyl phenylboronic acid pinacol ester 4 Methoxy 2 trifluoromethoxy phenylboronic acid pinacol ester 2 4 Difluoro 5 formylphenylboronic acid 1 BENZYL 4 PHENYLPIPERIDIN 4 YL METHANAMINE 3 Bromo 4 methoxyphenylboronic acid

1 FORMYL PIPERIDINE 4 CARBOXYLIC ACID 4 Methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 1 BOC 4 3 CARBOXY PHENYL PIPERIDINE 3 Hydroxy 4 methoxyphenylboronic acid 2 Methoxy 5 trifluoromethoxyphenylboronic acid pinacol ester 2S 5R 5 Hydroxypipecolic acid HCl 4 Cyclopentylphenylboronic acid pinacol ester 4 2 BROMOPHENYL PIPERIDINE 1 BOC 4 4 CHLOROPHENYL 4 PIPERIDINECARBOXYLIC ACID METHYL ESTER 2 3 Chloro 4 phenoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 HYDROXY PIPERIDINE 1 2 DICARBOXYLIC ACID 1 BENZYL ESTER 2 METHYL ESTER 5 n Octylthiophene 2 boronic acid pinacol ester 5 n Octylthiophene 2 boronic acid 5 Ethylthiophene 2 boronic acid pinacol ester 5 n Propylthiophene 2 boronic acid pinacol este 1 BOC 4 CYANO 4 3 BROMOPHENYL PIPERIDINE 2 8 DIAZA SPIRO 4 5 DECANE 2 3 8 TRICARBOXYLIC ACID 8 TERT BUTYL ESTER 2 9H FLUOREN 9 YLMETHYL ESTER 4 Trifluoromethoxy phenylboronic acid pinacol ester 4 4 METHYLPHENYL 4 PHENYLPIPERIDINE HYDROCHLORIDE 2 5 Dimethyl 4 formylphenylboronic acid pinacol ester 2 5 butylthiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 TRIFLUOROMETHYL 4 5 6 7 TETRAHYDRO 1H PYRAZOLO 4 3 B PYRIDINE 3 Chloro 2 fluorobenzeneboronic acid pinacol ester 4 4 BROMOPHENYL 4 4 CHLOROPHENYL PIPERIDINE 1 2 AMINOETHYL PIPERIDIN 2 YL METHANOL 2 Methoxy 4 methoxymethoxyphenylboronic acid 2 3 Ethoxy 5 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 6 METHYL 2 PIPERIDINEACETIC ACID 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 3 4 trahydroquinoline 3 Fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol

4 2 NITROPHENYL PIPERIDINE 2 2 2 trifluoro 1 piperidin 4 yl ethanone 4 Hydroxy 2 methoxyphenylboronic acid 2 Benzyloxy 4 trifluoromethyl phenylboronic acid 4 2 FLUORO PHENYL PIPERIDIN 4 OL 1 BOC 4 1 3 BENZODIOXOL 5 YL 4 HYDROXYPIPERIDINE 4 Phenylaminocarbonyl benzeneboronic acid pinacol ester 1 BOC 4 2 TRIFLUOROMETHYL PHENYL 4 HYDROXYPIPERIDINE 4 Cyclopropyl 3 mehtoxyphenylboronic acid 1 BOC 4 3 METHOXYPHENYL 4 HYDROXYPIPERIDINE 4 Isopropoxy 3 methoxyphenylboronic acid 2 Bromo 4 methoxyphenylboronic acid 3 Cyano 4 methoxyphenylboronic acid pinacol ester 4 5 6 7 Tetrahydro 1H Pyrazolo 3 4 c pyridine 1H INDAZOLE 7 CARBONITRILE 5 BROMO 3 1 ETHYLSULFONYL 4 PIPERIDINYL 4 Benzyloxy 2 isopropylphenylboronic acid 4 Phenoxy 2 methoxyphenylboronic acid pinacol ester 4 Phenoxy 2 trifluoromethyl phenylboronic acid 1H INDAZOLE 7 CARBOXAMIDE 5 BROMO 3 4 PIPERIDINYL 1 METHYL 4 PIPERIDINEACETIC ACID 5 Ethoxy 2 methylphenylboronic acid 1 BOC BETA OXO 3 PIPERIDINEPROPANOIC ACID ETHYL ESTER 3 Bromo 2 methoxyphenylboronic acid 2 Fluoro 4 methylphenylboronic acid pinacol ester 5 1 METHYL PIPERIDIN 4 YL 1H INDAZOLE 2 Benzyloxy 5 chloropyridine 3 boronic acid 6 1 METHYL PIPERIDIN 4 YL 1H INDAZOLE 2 Fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 AZABICYCLO 2 2 1 HEPTANE 3 CARBOXYLIC ACID 3 hydroxymethyl 5 methoxyphenyl boronic acid