4 5 6 7 tetrahydro 1H pyrazolo 4 3 c pyridine 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 triisopropylsilyl 1H pyrrole 6 bromo 2 methyl 1H imidazo 4 5 b pyridine 2 chloropyrimidin 5 ol 4 fluorobenzo b thiophene 2 carboxylic acid 4 Acetamido 3 bromobenzotrifluoride 4 Ethoxybenzenesulfonyl chloride 2 Chloro 3 6 difluorobenzonitrile 3 Bromo 2 fluorobenzoyl chloride 2 Chloro 3 6 difluorobenzaldehyde 5 Bromo 2 nitropyridine 2 Amino 1 3 benzothiazol 2 2 Dibromobutanal 3 Bromo 4 methoxyaniline hydrochloride 1 Bromo 3 fluorobenzene 4 Trifluoromethyl benzophenone 4 Chloro 2 methoxyphenol 4 Fluorophenyl isothiocyanate 3 Fluoro 5 trifluoromethyl benzonitrile 2 Iodobenzenesulphonic acid 4 Bromo 2 methylbenzoic acid 2 3 DIFLUORO 4 METHYLBENZONITRILE 6 Chloro 3 fluoropyridine 2 carboxylic acid 5 11 Dihydro 11 chloroacetyl 6h pyrido 2 3 b 1 4 benzodiazepine 6 one 4 methyl 2 3 5 6 tetrafluoro lbenzyl alcohol 4 Bromomethyl biphenyl 4 Amino 1 Boc piperidine 4 carboxylic acid 5 6 Dichloro 1 ethyl 2 methylbenzimidazole 3 Fluoro 2 nitropyridine 2 Bromo 4 nitrotoluene

3 Amino 5 bromo 2 chloropyridine 2 fluoro 4 methoxy 1 propan 2 yl benzene 3 1 fluoropropyl azetidine 2 5 dihydro 1H Pyrrole 1 sulfonyl fluoride 1 5 chloro 6 fluoro 1H indol 3 yl ethan 1 ol 1R 2 tert butyldimethylsilyl oxy 1 4 chloro 3 fluorophenyl ethan 1 ol 3 fluorooxetan 3 yl methanamine 2 6 Difluoropyridin 4 yl boronic acid 6 fluoropyridazin 3 amine 2R 3S 3 hydroxypyrrolidine 2 carboxylic acid trifluoroacetic acid 2 chloromethyl oxazolo 5 4 b pyridine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 cyanobenzohydrazide 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrole 2 methylpropane 1 2 diamine 6 bromo 1H imidazo 4 5 b pyridine 2 methylbenzo d oxazol 5 ol 2 6 difluoropyridin 3 amine 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 chloro 5 cyanophenylboronic acid 4 fluorobenzofuran 2 carboxylic acid 7 fluorobenzo b thiophene 2 carboxylic acid 4 Butyryl benzonitrie 2 Chloro 4 5 difluorobenzaldehyde 3 4 Difluorobenzenesulfonyl chloride 2 Bromo 6 methylpyridine N oxide 5 Aminobenzimidazole 2 Bromo 3 methylaniline 1 Bromo 2 fluorobenzene 2 Trifluoromethyl benzophenone

2 Chloro 4 methoxyphenol 3 Fluorophenyl isothiocyanate 4 Trifluoromethyl benzyl amine 2 Fluoro 6 trifluoromethyl benzonitrile 3 Bromo 5 methylbenzoic acid 2 Bromo 6 picoline 2 Bromo 5 nitrobenzoic acid 2 4 Dibromopyridine 2 Chlorobenzimidazole 2 Bromo 5 trifluoromethoxy aniline 2 Amino 3 iodo 6 methylpyridine 5 6 Dihydro 6 oxo 11H pyrido 2 3 b 1 4 benzodiazepine 4 Bromo 2 3 5 6 tetrafluorobenzaldehyde 3 4 5 triethoxybenzoic acid 4 Methyl 2 oxopentanoic acid methyl ester 3 1 fluoroethyl azetidine 3 5 difluoro 4 4 4 fluorophenyl piperidin 1 yl aniline 3 fluorooxetan 3 yl methanol 2 4 trifluoromethyl phenyl piperazine dihydrochloride 3 fluoropyrazine 2 carboxylic acid 3 Fluoropyridin 4 yl boronic acid 5 chloro 6 fluoro 1H indole 2‐ tert‐butoxy carbonyl amino ‐3‐ 3 3‐difluorocyclobutyl propanoic acid 2R 3R 4R 5R 5 2 amino 6 chloro 9H purin 9 yl 2 4 chlorobenzoyloxy methyl 4 fluoro 4 methyloxolan 3 yl 4 chlorobenzoate 6 chloroisoquinolin 1 amine 1 tert butoxycarbonyl 2 oxospiro indoline 3 4 piperidine 5 carboxylic acid 4 4 dimethylimidazolidin 2 one 2 chloro 6 trifluoromethyl nicotinonitrile 3 fluoropicolinaldehyde 1H imidazo 4 5 b pyridin 2 amine

2 2 difluoro 1 pyridin 2 yl ethanone 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 2 1H pyrazol 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 chloro 5 formylphenylboronic acid 4 bromobenzofuran 2 carboxylic acid 4 bromobenzo b thiophene 2 carboxylic acid 3 Chloro 2 methylbenzenesulfonyl chloride 3 amino 9 ethylcabazole 3 Trifluoromethyl benzyl amine 2 Ethoxyphenyl isothiocyanate 4 Chloro 3 fluorophenol 1 Bromo 2 6 difluoro 4 iodobenzene 2 Bromomethyl 6 methylpyridine 2 Bromo 4 iodoaniline 4 Bromo 3 trifluoromethyl benzaldehyde 5 Bromo 2 trifluoromethyl benzonitrile 2 Fluoro 5 trifluoromethyl benzonitrile 3 Bromo 2 methylbenzoic acid 2 AMINO 3 BROMOBENZONITRILE 2 3 5 6 tetrafluorobenzene 1 4 dicarboxylic acid 4 methoxy 2 6 dimethyl aniline 5 5‘ Bis 2H tetrazole diammonium salt 6 Bromoisoquinoline 3 Chloro 2 hydroxybenzaldehyde 3 Cyano 4 isopropoxybenzoic acid 2 Amino 6 nitrobenzimidazole 2 4 Dibromo 3 nitropyridine 2 5 Dimethoxybenzaldehyde 2 5 Dibromo 3 picoline 2 chloro 5 fluoropyridine 3 carboxylic acid