2S 5R 2 carbamoyl 7 oxo 1 6 diazabicyclo 3 2 1 octan 6 yl sulfate 4 2S 5R 6 benzyloxy 7 oxo 1 6 diazabicyclo 3 2 1 octan 2 yl carbonyl amino piperidine 1 carboxylic acid benzyl ester 4 Trifluoromethyl benzene 1 sulfonyl chloride 4 1H pyrazol 1 yl benzonitrile 5 6 dihydro 4H pyrrolo 3 2 1 ij quinoline 1 carboxylic acid 1 2 3 4 tetrahydroquinoline 8 chloro 2 phenyl 3 1S 1 9 tetrahydro 2H pyran 2 yl 9H purin 6 yl amino ethyl isoquinolin 1 2H one 1H Imidazole 5 acetic acid hydrochloride 1tetrazole 2 benzylamino ethanol 4 chlorotetrahydro 2H pyran 1 2 2 difluorobenzo d 1 3 dioxol 5 yl cyclopropanecarboxylic acid 3 fluoro 4 nitroaniline 1 bromo 2 chloroethane 1R 2S 3S 5S methyl 3 4 fluorophenyl 8 azabicyclo 3 2 1 octane 2 carboxylate 3aS 5R 6S 6aS 6 hydroxy 2 2 dimethyltetrahydrofuro 2 3 d 1 3 dioxol 5 yl morpholino methanone 1 chloro 2 4 ethoxybenzyl 4 iodobenzene 2 6 Dimethylpiperazine 1H ​Pyrido 3 ​4 4 ​5 ​pyrrolo 1 ​2 ​3 ​de ​quinoxaline ​8 7H ​ ​carboxylic acid 2 ​3 ​6b ​9 ​10 ​10a ​hexahydro ​3 ​methyl ​ ethyl ester 6bR ​10aS ​ 1 ​Butanone 4 ​chloro ​1 ​ 4 ​fluorophenyl ​ 1H ​Pyrido 3 ​4 4 ​5 ​pyrrolo 1 ​2 ​3 ​de ​quinoxaline 2 ​3 ​6b ​7 ​8 ​9 ​10 ​10a ​octahydro ​3 ​methyl ​ 6bR ​10aS ​ 1H ​Pyrido 3 ​4 4 ​5 ​pyrrolo 1 ​2 ​3 ​de ​quinoxaline ​8 7H ​ ​carboxylic acid 2 ​3 ​9 ​10 ​tetrahydro ​2 ​oxo ​ ethyl ester 4 nitroso 3 4 dihydroquinoxalin 2 1H one 4 aMino 2 3 difluoro 5 nitrobenzoic acid 5 4 broMo 2 chlorophenylaMino 4 fluoro 1 Methyl N 2 vinyloxy ethoxy 1H benzo d iMidazole 6 carboxaMide 2 3 4 Trifluorobenzoic acid 2 ​4 ​5 ​6 ​Pyrimidinetetramine hydrochloride 1 2 6 ​Oxaspiro 4 5 ​decane ​9 ​acetic acid α ​cyano ​9 ​ 2 ​pyridinyl ​ ​ methyl ester 6 oxaspiro 4 5 decan 9 one 3 5 Bis trifluoromethyl benzonitrile

2 ​Propanesulfinamide N ​ 1 ​ 2 ​fluoro ​5 ​nitrophenyl ​ethylidene ​ ​2 ​methyl ​ S R ​ ​ 6 Aminonicotinaldehyde 3 Pyridinecarboxaldehyde 6 5 fluoro 4 4 fluoro 2 methyl 1 1 methylethyl 1H benzimidazol 6 yl 2 pyrimidinyl amino 1H BenziMidazole 6 2 chloro 5 fluoro 4 pyriMidinyl 4 fluoro 2 Methyl 1 1 Methylethyl 1 6 Bromo 3 pyridinyl methyl 4 ethylpiperazine 4 Bromo 2 6 difluoroaniline 2 benzo b thiophen 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 benzofuran 7 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1H BenziMidazole 4 fluoro 2 Methyl 1 1 Methylethyl 6 4 4 5 5 tetraMethyl 1 3 2 dioxaborolan 2 yl 2 benzo b thiophen 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 5 Dimethyl 4 hydroxybenzaldehyde 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiophene 2 carbaldehyde 1 4 methylthiophenyl 3 3 5 dimethyl 4 hydroxyphenyl prop 2 en 1 one 4 methoxy 7 morpholin 4 yl benzothiazol 2 yl carbamic acid phenyl ester 2 4 dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 2 Methoxy 5 Morpholinophenyl thiourea 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 triisopropylsilyl 1H pyrrole 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyrimidin 2 amine 5’ 6’ 7’ 8’ tetrahydrospiro cyclohexane 1 2’ 1’h quinazolin 4’ 3’h one 2 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 9 Amino 2 bromoacridine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 6 dichloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 cyclopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 methoxy 2 methylphenylboronic acid 1 methyl 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 4 Aminophenylboronic acid pinacol ester 4 isopropylthio phenylboronic acid

2 2 2 diethylaminoethylamino ethyl 4 methyl 1H pyrrole 3 carboxylicacid ethyl ester 3 dimethylcarbamoyl phenylboronic acid 3 methoxymethyl phenylboronic acid 2 4 boronophenyl acetic acid 2 Chloro 4 6 di morpholin 4 yl 1 3 5 triazine 2 2 diethylaminoethylcarbamoyl methyl 4 methyl 1H pyrrole 3 carboxylic acid ethyl ester 4 piperidin 1 yl phenylboronic acid hydrochloride 4 bromo 2 6 difluorophenylboronic acid 2 carboxymethyl 4 methyl 1H pyrrole 3 carboxylic acid ethyl ester 2 ethylthio phenylboronic acid 3 4 dichlorobenzoyl chloride 4 pyrrolidin 1 yl phenylboronic acid 4 chloro 2 6 difluorophenylboronic acid 3 4 5 trichlorophenylboronic acid 4 cyanobenzoyl chloride 3 3 methoxy 3 oxoprop 1 enyl phenylboronic acid 2 chloro 4 trifluoromethyl phenylboronic acid 4 cyano N 4 cyanophenyl benzamide 2 3 difluoro 6 methoxyphenylboronic acid 3 amino 4 fluorophenylboronic acid 4 methoxy 3 methylphenylboronic acid 4 2 tert butyldimethylsilyloxy ethoxy methyl phenyl methanol 3 aminomethyl phenylboronic acid hydrochloride 2 tert butyl 4 chloro 5 hydroxypyridazin 3 2H one 4 benzyloxycarbonylamino phenylboronic acid 3 benzyloxycarbonyl phenylboronic acid 2 tert butyl 4 chloro 5 4 2 hydroxyethoxymethyl benzyloxy 2H pyridazin 3 one 3 isopropoxycarbonyl phenylboronic acid 2 6 difluoro 4 formylphenylboronic acid 2S 3R 3 2 methylpropan 2 yl oxy 2 2 methylpropan 2 yl oxycarbonylamino butanoic acid

3 tert butoxycarbonyl phenylboronic acid 2 morpholinomethyl phenylboronic acid 4S 5S 5 methyl 2 oxo 1 3 oxazinane 4 carboxylic acid 2 dimethylamino phenylboronic acid 4 benzyloxy phenylboronic acid 4 aminophenylboronic acid 4 1H imidazol 1 yl phenylboronic acid 2 ethynylphenylboronic acid 4 trimethylsilyl ethynyl phenylboronic acid 3 amino 5 trifluoromethyl phenylboronic acid 1 chloromethyl 4 trifluoromethyl benzene 2S 3S 3 2S 1 4 aminobutylamino 4 methyl 1 oxopentan 4 formyl 3 methoxyphenylboronic acid 2 methylbenzo d oxazol 6 ylboronic acid 4 fluoro 2 formylphenylboronic acid 2S 6 dimethylamino 2 2 methylpropan 2 yl oxycarbonylamino hexanoic acid 2 tert butoxycarbonylamino 5 fluorophenylboronic acid 3 cyano 4 methoxyphenylboronic acid 2 methoxy 5 nitrophenylboronic acid 4 borono 2 nitrobenzoic acid 5 2 2 dibromoethenyl 2 methoxyphenol 3 benzyloxy 4 methoxyphenylboronic acid 4 chloro 2 cyanophenylboronic acid 4 2 2R 3R 3 2 4 difluorophenyl 3 hydroxy 4 1 2 4 triazol 1 yl b utan 2 yl 1 3 thiazol 4 yl benzonitrile 3 acetyl 4 fluorophenylboronic acid 3 chloro 5 cyanophenylboronic acid 3 chloro 5 methylphenylboronic acid 2 cyano 6 fluorophenylboronic acid 3 cyano 5 fluorophenylboronic acid 1 3 5 Trichloro 1 3 5 triazinane 2 4 6 trione