2 Methoxy 4 methylthio pyridine 5 boronic acid 4 Isopropoxy 3 trifluoromethyl phenylboronic acid 4 Fluoro 3 methanesulfonyl phenylboronic acid 2 Methylthio thiophene 4 boronic acid 2 Methylthio thiophene 3 boronic acid 3 Methoxy 2 methylphenylboronic acid 2 CHLORO 3 METHYL 5 PHENYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 3 Bromo 5 carboxythiophene 2 boronic acid 2 CHLORO 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 4 N Boc piperazino pyridine 5 boronic acid 3 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 3 Bromo 2 formylthiophene 5 boronic acid 2 Benzyloxy 4 methylpyridine 5 boronic acid 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 PYRIDINAMINE 2 Phenoxypyridine 4 boronic acid 2 CHLORO 5 METHOXYPYRIDINE 4 BORONIC ACID 2 Isopropoxy 4 methylpyridine 5 boronic acid pinacol ester 2 Isopropoxy 4 methylpyridine 5 boronic acid 2 CARBOXYPYRIDINE 4 BORONIC ACID 4 Benzyloxy 2 chlorophenylboronic acid 6 Ethoxy 2 fluoro 3 methylphenylboronic acid 5 BROMO 2 TRIFLUOROMETHYL PYRIDIN 4 YLBORONIC ACID 2 CHLORO 3 FLUORO 5 PICOLINE 4 BORONIC ACID 5 Methyl 1H indazole 4 boronic acid 2 TRIFLUOROMETHYL PYRIDINE 4 BORONIC ACID 2 4 Difluoro 3 hydroxymethyl phenylboronic acid 4 Piperazin 1 ylmethyl phenylboronic acid 4 2 methylpropyl amino methyl phenylboronic acid 2 CHLORO 3 FLUOROPYRIDINE 4 BORONIC ACID

4 BORONO 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIETHYL ESTE 6 Fluoro 2 hydroxy 3 methylphenylboronic acid pinacol ester 2 N BOC AMINO 6 ETHOXYCARBONYL 4 PYRIDINE BORONIC ACID PINACOL ESTER 5 Methoxy 4 methylpyridine 3 boronic acid 3 N N Dimethylaminomethyl phenylboronic acid pinacol ester 2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 Fluoro 4 5 dimethoxyphenylboronic acid 5 BROMO 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 PYRIDINECARBONITRILE 5 Diethylamino methyl 2 fluorophenylboronic acid 2 6 DIMETHYL PYRIDINE 4 BORONIC ACID 2 4 Difluoro 3 isopropoxyphenylboronic acid 4 Isobutoxyphenylboronic acid 5 hexylpicolinic acid 2 Fluoro 4 morpholinomethyl phenylboronic acid pinacol ester 2 TERT BUTYLDIMETHYLSILYLOXY METHYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 2 HYDROXY PYRIDINE 4 BORONIC ACID 5 Hydroxymethylthiophene 2 boronic acid pinacol ester 2 CYANOPYRIDIN 4 YL BORONIC ACID 4 Bromo 3 fluorophenylboronic acid pinacol ester 1 3 DIHYDRO 1 HYDROXY 1 2 OXABOROLO 4 3 C PYRIDINE 2 Fluoro 4 morpholinomethyl phenylboronic acid 3 4 Dichloropyridine 5 boronic acid pinacol ester 3 Fluoro 4 piperidin 1 ylmethyl phenylboronic acid 2 PYRIDINECARBOXAMIDE 6 METHYL N 4 METHYL 2 THIAZOLYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 Fluoro 4 methoxycarbonylphenylboronic acid pinacol ester 3 FLUORO 2 4 MORPHOLINO PYRIDINE 4 BORONIC ACID PINACOL ESTER 4 Methoxy 2 6 dimethylphenylphenylboronic acid pinacol ester 2 Chloro 5 trifluoromethyl phenylboronic acid pinacol ester 6 Azaindole 4 boronic acid 1 ISOPROPYLPIPERAZINE

1 Boc 4 3 NITRO PYRIDIN 2 YL PIPERAZINE 2 3 Difluoro 6 chlorophenylboronic acid 3 Bromo 2 fluoro 6 methoxyphenylboronic acid 1 BENZYL 4 3 NITROPYRIDIN 2 YL PIPERAZINE 4 Hydroxy 3 methoxyphenylboronic acid pinacol ester 1 BOC 4 BUTYLPIPERAZINE 2 Fluoro 3 piperidin 1 ylmethyl phenylboronic acid 1 PROPYLPIPERAZINE 4 Bromo 3 trifluoromethyl phenylboronic acid pinacol ester 1 BOC 4 ISOPROPYLPIPERAZINE 4 BENZYL 3 OXOPIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 4 Trifluoromethylphenylboronic acid pinacol ester 2 CARBOXYMETHYL 3 OXO PIPERAZINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 3 Fluoro 5 pyrrolidinophenylboronic acid 5 Chloro 2 propoxy 4 pyridinyl boronic acid 5 Bromo 6 methylpyridine 2 carboxylic acid methyl ester 4 benzylpiperazin 1 amine 3 Carboxy 5 trifluoromethyl phenylboronic acid 2 4 tert butoxycarbonyl 2 methylpiperazin 1 yl acetic acid 5 Methyl 2 methylthio phenylboronic acid 3 benzyl 7 tert butyl 9 oxo 3 7 diaza bicyclo 3 3 1 nonane 3 7 dicarboxylate 6 Isobutoxy 5 methylpyridine 3 boronic acid 3 Cyano 5 methylphenylboronic acid pinacol ester 6 Chloro 5 methoxypyridine 3 boronic acid 1 1 9H fluoren 9 yl methoxy carbonyl pyrrolidine 2 carbonyl pyrrolidine 2 carboxylic acid 1 benzyl 3 methylpyrrolidin 3 amine 2 Fluoro 3 hydroxymethyl phenylboronic acid 5 Hydroxy 2 methylphenylboronic acid pinacol ester 4 Methoxycarbonyl 3 trifluoromethyl phenylboronic acid pinacol ester 3 Fluoro 2 methoxy 4 methylphenyl phenylboronic acid

3 N O Dimethylhydroxylaminocarbonyl 5 fluorophenylboronic acid 1 1 ADAMANTYLCARBONYL PYRROLIDINE 2 CARBOXYLIC ACID 6 Bromo 2 methoxypyridin 3 ylboronic acid 5 Bromo 2 fluoro 3 formylphenylboronic acid pinacol ester 1 benzylpyrrolidine 3 carbonitrile oxalate 6 Ethoxy 2 methylpyridine 3 boronic acid 1 tert butyl 2 methyl 2 3 chloropropyl pyrrolidine 1 2 dicarboxylate 2 Formyl 5 isopropylphenylboronic acid 3 Fluoro 4 methylcarbamoyl phenylboronic acid 2 5 Difluoro 4 formylphenylphenylboronic acid 1 Tetrahydro pyran 2 yl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 2 Fluoro 6 iodophenylboronic acid pinacol ester 4 4 Methylpiperazino methylphenylboronic acid pinacol ester 2 Chloro 5 methoxymethylphenylboronic acid pinacol ester 5 hydroxymethyl 1 methylpyrrolidin 2 one 3 Fluoro 4 morpholinylmethyl phenylboronic acid 3 Morpholinomethyl phenylboronic acid 1 tert butyl 3 ethyl 3 methyl 4 oxopyrrolidine 1 3 dicarboxylate 4 Bromo 2 hydroxyphenylboronic acid 5 Tert butylcarbmoyl 2 fluorophenylboronic acid 3 benzyl 6 oxa 3 aza bicyclo 3 1 0 hexane 3 pyridin 4 yl 1H pyrazol 5 amine 2 Fluoro 5 pyrolidine 1 carbonyl phenylboronic acid 5 Carbamoyl 2 fluorophenyboronic acid 2 Fluoro 5 propylcarbamoyl phenylboronic acid 5 Dimethylcarbamoyl 2 fluorobenzeneboronic acid 4 Methoxymethyl 2 6 dimethylphenylboronic acid 2 Fluoro 5 methoxypyridine 3 boronic acid 4 4 5 5 Tetramethyl 2 3 trifluoromethyl benzyl 1 3 2 dioxaborolane 2 5 Difluoro 4 benzyloxyphenylboronic acid