1 benzyl 3 3 difluoropiperidine 4 4 diol 3 3 difluoro 1 methylpiperidin 4 ol hydrochloride 4 ethoxycarbonyl methyl cyclohex 1 enyl trifluoromethanesulfonate 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 3 carboxamide 5 5 5 trifluoro 4 4 dihydroxypentanoic acid 3 3 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 4 carboxamide 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl piperidine 2 carboxamide 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 2 carboxamide 5 Bromo 2 methylpyridin 3 ol 2 3 Aminophenyl 2 methylpropanenitrile 4 Morpholin 4 yl benzene 1 carboximidamide hydrochloride 2 Chloromethyl nicotinonitrile 2 3 Fluoro 5 methoxyphenyl acetonitrile 4 Bromo 1 bromomethyl 2 chlorobenzene 3 2H 1 2 3 Trizazol 2 yl aniline 4 Aminobicyclo 2 2 2 octane 1 carboxylic acid methyl ester 3 Amino 6 bromopyrazine 2 carbaldehyde 4 Bromobutan 1 amine hydrobromide 4 Hydroxy 4 trifluoromethyl cyclohexanecarboxylic acid 4 tert Butyl cyclohex 1 ene 1 2 Bromo 5 chlorophenyl ethanone 3 3 Nitrophenoxy azetidine hydrochloride 5 Bromo 2 cyano 4 methylpyridine 4 6 Dichloro 2 methylthio 5 nitropyrimidine 4 Chloro 8 fluoro 2 trifluoromethyl quinazoline 5 Pyrimidinecarboxylic acid 4 6 dichloro ethyl ester 4 4 Ethylpiperazin 1 ylmethyl benzoic acid 4R 5R 3 tert Butyl 4 methyl 2 2 5 trimethyloxazolidine 3 4 dicarboxylate 6 7 Dihydro 5H cyclopenta b pyridin 4 amine 4 Dimethylamino benzamide

3 Amino 4 nitrobenzonitrile 1 1 Diphenyl 4 piperidin 1 yl butan 1 ol hydrochloride 1H Pyrrol 2 yl methanamine hydrochloride 2 Bromomethyl 4 chloro benzoic acid methyl ester 4 Oxopiperidine 3 carbonitrile hydrochloride 3 Bromo 5 prop 1 en 2 yl pyridine 3 Bromo 5 trifluoromethyl phenol 5 Bromo 2 3 dimethoxypyrazine 2 Chloro 7 nitroquinoxaline 7 Benzenesulfonyl 4 chloro 6 methyl 7H pyrrolo 2 3 d pyrimidine 3 4 Dihydropyrrolo 1 2 a pyrazin 1 2H one 6 Bromospiro chroman 2 4 piperidin 4 one 1 Phenoxycarbonyl pyrrolidine 2 carboxylic acid 3 Amino 3 methylbutyric acid hydrochloride 3 Aminocyclopentanol hydrochloride 4 Amino 3 fluorobenzoic acid allyl ester 6 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl indolin 2 one 2 Amino 4 bromo 3 nitropyridine 3 Ethoxypyridazine 4 4 Dimethylpyrrolidine 3 carboxylic acid hydrochloride 3 Amino 3 4 chlorophenyl 1 propanol 1 4 Dioxa 8 azaspiro 4 5 decane hydrochloride 2 Hydroxycyclopent 2 en 1 one 4 Cyano 3 fluorobiphenyl 4 carboxylic acid 4 Methyl 1H indazol 5 yl boronic acid 5 Fluoro 2 pyrimidineacetic acid 1 Cyclobutyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 Phenyl 1 p tolylsulphonyl piperidine 4 carbonitrile 4 Pyrimidinol 5 fluoro 2 methyl 7CI 8CI 5 Methyl 2H isoquinoline 1 one

1 Boc 4 5 methyl 1 3 4 oxadiazol 2 yl piperidine 5 Bromoquinoline 2 carboxylic acid 8 bromoquinoline 5 carboxylic acid 2 Bromo 4 trifluoromethyl thiazole 3 4 Dibromo 5 fluoropyridine 4 Diphenylmethoxypiperidine hydrochloride 4 Ethynylphenylacetonitrile 3 Fluoro 5 hydroxybenzoic acid 6 Chloronicotinimidamide hydrochloride 5 Bromo 2 nitroaniline 3 Chloroisoquinoline 4 carbaldehyde 1 Benzenesulfonyl 1H pyrrolo 2 3 b pyridine 2 carboxylic acid 1 H Spiro piperidine 4 2 quinazolin 4 3 H one 1 5 Bromo 2 nitrophenyl ethanone 5 Bromo 1H pyrrolo 2 3 b pyridine 3 carbaldehyde 5 Benzyloxy pyridin 2 amine 5 Fluorospiro cyclopropane 1 3 indoline 4 4 Chlorophenoxy phenyl methanamine hydrochloride 2 Bromo 5 methylthiazole 4 carboxylic acid 1H Pyrazolo 4 3 b pyridine 3 carboxylic acid 5 Bromo 2 4 chlorophenyl pentanoic acid 7 Bromo 2 chlorothieno 3 2 d pyrimidine 3 chloro 5 methylpyridin 4 amine 2 Bromoimidazo 2 1 b 1 3 4 thiadiazole 1 Bromo 2 methoxy 4 trifluoromethyl benzene 3 Bromo 2 methyl phenol 4 Bromopyrimidin 2 yl cyclopentylamine 3 fluoro 2 nitrobenzonitrile 2 Chloro 5 iodopyrimidin 4 amine 3 Bromo 4 trifluoromethyl benzoic acid

4 Bromo 1H pyrrole 2 carbaldehyde 6 Chloro 3 methylpyrimidin 4 3H one 4 Hydroxycyclohexanecarbonitrile 6 Chloro N N dimethylpyrimidin 4 amine 1 6 Chloropyrimidin 4 yl 4 piperidinol 2 Morpholin 3 yl acetic acid hydrochloride 5 Bromo 3 fluoro 4 methylbenzaldehyde 2 7 Dichlorothiazolo 5 4 c pyridine 5 Bromo 3 methoxypyridin 2 amine 2 Amino 5 methoxybenzamide 6 Bromo 2 chloronicotinaldehyde 3 4 Fluorophenoxy pyrrolidine hydrochloride 3 Bromo 2 chlorobenzonitrile 3 Bromo 4 6 dichloro 1H pyrazolo 3 4 d pyrimidine 3 Chloro 2 fluoroanisole 6 Methyl 2 4 pyrimidinediamine 7 Nitro 3 4 dihydro 2H 1 4 benzooxazine 3 2 Isopropyl 1H Imidazol 1 YL Methyl Phenyl Amine Dihydrochloride 2 Bromo 6 morpholinopyridine 2 Isopropoxyaniline 11 A Hydroxy canrenone methyl ester 6 Bromo 2 methyloxazolo 4 5 b pyridine 2 Amino N methylethanesulfonamide hydrochloride 4 Iodo 1H pyrazole 5 carboxylic acid 4 Ethyl 2 methyl 1 3 thiazole 5 carboxylic acid 2 Chloro 4 ethynylpyridine 3 Boc 3 8 diazabicyclo 3 2 1 octane 4 Oxocyclohexanecarbonitrile 1 Phenylpiperidin 4 yl methanol 4 4 Benzylpiperazin 1 ylmethyl phenylamine