2 Fluoro 6 nitrobenzyl bromide 2 Bromo 3 fluoroanisole 3 Fluoro 2 iodonitrobenzene 2 Chloro 1 2 5 difluorophenyl ethanone 1 4 Trifluoromethyl benzyl piperazine 3 5 Bis trifluoromethyl thiophenol 2 amino 5 Bromo 3 methoxypyrazine 4 Cyano 3 fluoroacetophenone 4 Hydroxy 3 methoxybenzaldehyde 2 6 Dimethylacetanilide 2 Bromo 4 chlorobenzyl cyanide 2 4 Dimethylbenzyl chloride 2 Trifluoromethyl phenylacetic acid 3 4 5 Trimethoxybenzoic acid 4 fluoro 3 nitrotoluene 2 Methyl 1 octylindole 9 Bromoanthracene 5 Bromo 2 chlorobenzonitrile 2 Methoxy 5 picoline 1 Acetoxy 4 fluorobenzene 4 Bromo 3 trifluoromethyl benzonitrile 3 5 dimethoxyisonicotinic acid 2 bromo N N dimethylpyrimidin 5 amine 4 chloro 7 8 dimethoxyquinazoline 4 chloro 2 3 dimethylpyridine 4 cyano 3 methoxyphenylboronic acid 1 2 methylbenzo d oxazol 6 yl 3 1 5 naphthyridin 4 yl urea 2 iodonicotinonitrile 1 3 iodothiophen 2 yl ethanone 2 4 fluorophenyl 3 oxo 2 3 dihydropyridazine 4 carboxylic acid

4 Amino 6 chloro 2 methoxypyrimidine 2R pyrrolidine 2 carbonitrile trifluoroacetate 2 bromo 5 fluoro 4 iodopyridine 3s 4r rel 4 boc amino 3 fluoropiperidine 2 7 ethoxy 4 3 fluorophenyl 1 oxo 1 2 dihydrophthalazin 2 yl N methyl N 2 methyl 1 3 benzoxazol 6 yl acetamide 4 4 trifluoromethyl phenyl phenyl methanamine 6 bromo 4 fluoro 1H pyrrolo 2 3 b pyridine 6 bromo 5 fluoro 3 methyl 1H indazole 5 chloro 3 methylbenzo b thiophene 5 bromoisoquinolin 1 amine 3 chloro 4 methoxyphenylboronic acid 3 5 Dichlorotoluene 2 Fluoro 5 nitronbenzyl alcohol 5 Bromo 2 3 difluorophenol 2 Fluoro 5 iodonitrobenzene 4 4 Trifluoromethoxy phenoxy piperidine 4 Chloro 2 2 2 trifluoroacetophenone 1 Acetyl 4 piperidinecarboxylic acid 3 Cyanoacetophenone 2 Nitro 1 3 5 tri tert butylbenzene 3 Hydroxy 4 methoxybenzaldehyde 4 Bromobenzyl cyanide 2 6 Difluorobenzyl chloride 2 Trifluoromethyl benzoic acid 4 Trifluoromethoxy phenylacetic acid 4 Fluoro 2 nitrotoluene 1 3 5 Triazine 1 3 5 tributylhexahydro 2 Fluoro 6 iodoanisole 2 Methoxy 5 nitro 4 picoline 4 Bromo 2 trifluoromethyl benzonitrile

2 4 5 Triiodoimidazole 4 Trifluoromethyl biphenyl 4 carbaldehyde 1 4 fluorophenyl methyl cyclopropane 1 carboxylic acid 5 5 difluorooxan 3 amine 4 fluoro 1H pyrrolo 2 3 b pyridine 6 carbonitrile 4 fluoro 2 methyl 1H pyrrolo 2 3 b pyridine 6 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl indolin 2 one 2 iodonicotinic acid 2 anthracen 9 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 trifluoromethyl phenoxy nicotinic acid 2S pyrrolidine 2 carbonitrile trifluoroacetate 1 2 bromophenyl 3 2 hydroxy 4 nitrophenyl urea 2 bromo 5 methoxypyridine 3 6 dichloropyridin 2 amine 5 methoxy 2 trifluoromethyl phenylboronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinamide 6 chloro 3 methylbenzo b thiophene 2 6 dibromo 4 iodophenol 7 8 dimethoxyquinazolin 4 3H one 3 bromopyrazine 2 carboxylic acid 4 bromoquinolin 2 amine 3 Chloro 2 nitrotoluene 2 Fluoro 4 nitrobenzyl alcohol 2 Ethyl iodobenzene 4 Chloroacetophenone 4 Bromo 2 6 difluoroanisole 2 Hydroxy 5 methoxybenzaldehyde 3 Chloro 5 trifluoromethoxy 2 2 2 trifluoroacetophenone 1 bromo 2 methoxymethyl benzene 4 Iodo 1 Tert butylbenzene

1 Acetylpiperazine 2 Aminobenzaldehyde 5 Fluoro 2 nitrotoluene 3 Trifluoromethoxy phenylacetic acid 2 4 6 Triisopropylbenzoic acid 2 4 Difluorobenzyl chloride 3 Bromobenzyl cyanide 2 Chloro 4 trifluoromethyl acetanilide 1 4 Dimethoxy 2 fluorobenzene 2 Amino 4 5 difluorobenzoic acid 5 Fluoro 2 methoxy 6 picoline 4 Chloro 2 5 Difluorobenzonitrile 2S 3R 4S 5S 6R 4 amino 2 1S 2S 3R 4S 6R 4 6 diamino 3 2R 3R 6S 3 amino 6 aminomethyl 3 6 dihydro 2H pyran 2 yl oxy 2 hydroxycyclohexyl oxy 6 hydroxymethyl tetrahydro 2H pyran 3 5 diol 1 2 Dibromohexafluoropropane 3 3 difluoro 3 pyridin 4 yl propanoic acid 3s 4r rel 1 boc 3 fluoro 4 hydroxymethyl piperidine 2 2 4 fluorobenzylthio 4 oxo 4 5 6 7 tetrahydro 1H cyclopenta d pyrimidin 1 yl acetic acid 1 5 4 3 trifluoromethyl phenyl piperazin 1 yl sulfonyl 2 3 dihydro 1H indol 1 yl ethan 1 one 4 fluorooxan 3 amine 6 trifluoromethyl 1H pyrrolo 2 3 b pyridine 3 carboxylic acid 5 chloromethyl 2 trifluoromethyl pyrimidine 5 3 fluorocyclobutyl 1H pyrazol 3 amine 2 dibenzofuranamine 1 hydroxy N methyl 2 naphthamide 7 bromo 5 nitro 1H indazole 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 2 chloro N 2 N cyanosulfamoyl 1 1 biphenyl 4 yl methyl N 4 methylbenzyl benzamide 5 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl isoxazole 2 iodo 4 methoxybenzonitrile