2 Butylthiophene 1 7 Iodo 3 4 dihydro H quinolin 1 yl ethanone 7 Iodo 1 2 3 4 tetrahydroquinoline 4 Fluoro 1 naphthaldehyde 5 Hexylthiophene 2 carboxaldehyde 5 Bromo 2 hexylthiophene 5 Methoxymethyl thiophene 2 carbaldehyde 1 4 Methylphenyl sulfonyl 1H indole 1 Bromo 3 fluoro 5 piperidinobenzene 1 4 Dioxaspiro 4 5 decan 8 yl benzoate 2 4 Bromobenzyl malonic acid 1 3 4 Dichloro benzyl piperidine 4 Bromo 2 fluorobenzoyl piperidine 5 Methoxy 1H pyrazolo 3 4 b pyridine 5 Bromo 2 4 BOC piperazin 1 yl 3 methylpyridine 4 3 Bromo pyridin 4 ylmethyl morpholine 4 Bromo 7 iodo 1H indazole 4 Fluoro 7 methylthio 1H indazole 5 5 Bromo 2 methylphenyl 1H tetrazole 5 2 Aminophenyl 1H tetrazole 5 3 Bromo 5 fluorophenyl 2H tetrazole 5 3 Fluorophenyl 1H tetrazole 4 2 Bromo 5 hydroxybenzyl morpholine 4 2 6 Difluoro 3 bromobenzyl morpholine 5 Bromo 2 methoxymethyl pyridine 4 2 fluoro 3 methoxybenzyl morpholine 4 Fluoro 6 methylthio 1H indazole 4 2 6 Dichloropyridine 3 yl methyl mopholine 1 4 Bromo 3 chlorophenyl methyl pyrrolidine 7 Chloro 6 fluoro 1H indazole

1 4 Bromo 2 6 difluorobenzyl pyrrolidine 4 4 Bromo 2 fluorobenzyl morpholine 4 Chloro 5 methyl 1H indazole 4 2 Chloro 6 fluoro 3 methylbenzyl morpholine 1 4 Bromo 3 chlorobenzyl piperidine 1 2 6 Dibromobenzyl pyrrolidine 1 2 Bromo 5 methylphenyl methyl pyrrolidine 1 2 bromo 5 trifluoromethyl phenyl methyl piperidine 4 5 Bromo 2 methoxybenzyl morpholine 4 Bromo 2 chlorophenyl methyl morpholine hydrochloride 2 5 Dibromo 3 pyrrolidinocarbonyl pyridine 2 Bromo 6 propan 2 yloxy naphthalene 4 5 Bromopyridin 3 yl methyl morpholine 3 Bromo 5 pyrrolidin 1 yl methyl pyridine 4 2 Bromo 5 methylphenyl methyl morpholine 2 Bromo 5 methylthio thiophene 4 4 Bromobenzyl morpholine 1 2 Bromo 5 methoxyphenyl methyl piperidine 1 1 Ethoxyethyl 1H pyrazole 4 2 Bromo 4 fluoro 6 methylbenzyl morpholine 4 4 Bromo 3 methoxybenzyl morpholine 4 2 Bromo 5 trifluoromethyl phenyl methyl morpholine 5 Bromo 3 methyl 2 methylthio pyridine 2 Bromo 5 piperidin 1 ylmethyl pyridine 4 6 Bromopyridine 3 yl methyl mopholine 3 4 Dibromo 2 5 bis methylthio thiophene 2 Methylthio thiophene 3 carboxaldehyde 2 Methylthio thiophene 4 carboxaldehyde 1 4 Bis tert butoxycarbonyl piperazine 3 Morpholinomethyl benzaldehyde

1 3 Bromo 4 methoxy benzyl piperidine 1 3 Bromo 4 methoxyphenyl methyl 4 methylpiperazine 1 5 Bromo 2 methoxy benzyl pyrrolidine 7 Chloroindazole 5 Bromo 2 phenylmethyl 2H indazole 1 3 Bromobenzyl piperidine 1 2 Bromobenzyl piperidine 3 Bromoquinoline 2 carbaldehyde 4 3 Bromo 4 fluorobenzyl morpholine 1 4 Bromo 2 6 difluorophenyl carbonyl pyrrolidine 4 6 Difluoro 1H indazole 6 Chloro 5 fluoro 1H indazole 4 Trifluoromethyl 1H indazole 4 Bromo 7 ethoxy 1H indazole 3 Bromo 2 iodoquinoline 2 Phenyl 1 3 2 dioxaborinane 1 4 Bromo 3 fluorophenyl carbonyl pyrrolidine 4 Chloro 7 methoxy 1H indazole 4 Bromo 7 methoxy 1H indazole 1 Boc 4 fluoro 1H indazole 1 Butyl 1H pyrazole 6 Bromo 5 fluoro 1H indazole 1 Propyl 1H pyrazole 4 Bromo 1 1 ethoxy ethyl 1H pyrazole 5 Bromobenzo 1 3 dioxole 4 boronic acid 6 Bromo 1 chloro 2 methoxynaphthalene 2 3 Dihydro 1 benzofuran 5 ol 3 Methylthio thiophene 5 Bromo 1 tert butoxycarbonylindole 4 Methylthiophene 2 carboxaldehyde

5 Bromo 1 phenylmethyl 1H indazole 4 4 Bromo 2 6 difluorobenzyl morpholine 6 Chloro 1 3 dihydro 2 1 benzoxaborol 1 ol 4 5 Bromo pyridin 2 yl morpholine 2 2 Bromophenyl 6 butyl 1 3 6 2 dioxazaborolane 2 Chloro 1 tetrahydro 2H pyran 2 yl 1H imidazole 2 3 Bromo 5 chlorophenyl 1 3 dioxolane 5 Methoxy 6 methylpicolinaldehyde 5 Bromo 2 fluoroisonicotinic acid 3 Bromo 4 chloropyridine 5 methanol 2 3 4 Trichloropyridine 2 Chloro 6 methoxynicotinaldehyde 4 5 6 Trichloronicotinic acid 2 Fluoropyridine 3 carboxaldehyde oxime 5 Bromo 2 ethoxypyridin 3 yl methanol 5 Chloro 2 ethoxynicotinic acid 5 Chloro 2 isopropoxy pyridine 3 carbaldehyde 2 4 Methoxyphenyl pyridine 2 Bromo 5 chloronicotinaldehyde 2 Ethoxy 3 pyridinemethanol 5 Chloro 2 methoxypyridine 3 methanol 2 Isopropoxypyridin 3 yl methanol 2 Chloro 5 fluoro pyridin 4 ol 2 Chloro 5 methoxy 3 pyridinecarboxylic acid 2 6 dimethoxy 3 trimethylsilyl pyridine 3 5 Dibromo 2 6 dimethoxypyridine 1 5 Bromo 2 6 dimethoxy 3 pyridinyl ethanone 2 Chloro 3 fluoro 4 methylthio pyridine 5 Isopropoxypyridin 3 yl methanol 2 Chloro 6 trifluoromethyl pyridin 4 yl methanol