1 N BOC 4 4 CHLOROPHENYL PIPERIDINE 4 2 4 DICHLOROPHENYL 4 PIPERIDINOL 5 BROMOSPIRO INDOLINE 3 4 PIPERIDINE 4 2 4 DIFLUOROPHENYL PIPERIDINE HYDROCHLORIDE 1 2 3 CHLORO 2 FLUORO PHENYL ETHYL 6 7 DIMETHOXY 1 2 3 4 TETRAHYDRO ISOQUINOLINE 3 FLUORO PIPERIDIN 1 YLAMINE 1 2 MORPHOLINOETHYL 4 PHENYL 4 PIPERIDINECARBOXALDEHYDE DIHYDROCHLOR IDE 1 BOC 4 2 FLUOROPHENYL 4 PIPERIDINECARBOXYLIC ACID 1 BOC 4 2 FLUOROPHENYL 4 PIPERIDINECARBOXYLIC ACID METHYL ESTER 1 2 BIS 4 FLUOROPHENYL METHOXY ETHYL 4 PHENYL 4 PIPERIDINOL HYDROCH LORIDE 1 N BOC 4 4 METHYLCARBAMOYLPHENYL PIPERIDINE 4 3 5 DICHLORO PHENYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 1 BUTYL 4 FORMYL 1 METHYL 4 PHENYLPIPERIDINIUM IODIDE 4 AMINO 4 4 BROMO PHENYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 2 2 6 6 tetramethylpiperidin 1 ol 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octane 4 methylbenzenesulfonate 4 SPIRO 1 3 4 DIHYDRO NAPHTHALENE PIPERIDINE HCL 1 benzyl 3 5 dimethyl piperidine 1 3 5 tricarboxylate 1 N Boc 1 7 diaza spiro 4 5 decan 6 one 1 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 10 10 DIFLUORO 2 7 DIAZA SPIRO 4 5 DECAN 1 ONE HYDROCHLORIDE 4 bromo 1 propyl 1 2 3 6 tetrahydropyridine 8 Boc 2 8 DIAZA SPIRO 5 5 UNDECAN 1 ONE 7 Boc 2 7 DIAZA SPIRO 5 5 UNDECAN 1 ONE 1 tert butylpiperidin 4 one 8 Boc 2 8 DIAZA SPIRO 5 4 DECAN 1 ONE 2S 1 tert butoxycarbonyl 4 hydroxypiperidine 2 carboxylic acid 1 tert butoxycarbonyl 2 methoxycarbonyl piperidine 4 carboxylic acid 4 5 6 7 tetrahydro 1H pyrazolo 3 4 c pyridin 3 ol hydrochloride 1 2 bis 1 benzylpiperidin 4 ylidene hydrazine

4 bromomethyl piperidine hydrochloride 1 HYDROXYMETHYL 2 AZABICYCLO 2 2 2 OCTANE 1 tert butoxycarbonyl octahydro 1H pyrrolo 3 2 c pyridine 3a carboxylic acid 2 N methyl 1 HYDROXYMETHYL 2 AZABICYCLO 2 2 2 OCTANE 7 N BENZYL 1 OXO 2 7 DIAZA SPIRO 4 5 DECAN 10 ONE ETHYLENE KETAL 1 tert butyl 3 3 dimethyl 4 oxopiperidine 1 3 3 tricarboxylate 3 OXO 2 AZABICYCLO 2 2 2 OCTANE 1 CARBOXYLIC ACID METHYL ESTER 1 benzyl 4 hydroxypiperidin 3 yl methyl acetate 1 1 dibenzyl 1 1 2 2 5 5 6 6 octahydro 3 3 bipyridine 1 tert butyl 4 ethyl 4 methyl 3 oxopiperidine 1 4 dicarboxylate 3 oxa 9 aza bicyclo 3 3 1 nonan 7 one hydrochloride 6 BROMO 2 CHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 2 6 DICHLORO 3 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL PYRIDINE 4 bromo 1 propyl 1 2 3 6 tetrahydropyridine hydrochloride 3 FLUOROPYRIDINE 4 BORONIC ACID HYDRATE 3 BROMO 2 METHOXYPYRIDINE 4 BORONIC ACID 3 5 DIMETHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 2 3 DIMETHOXYPYRIDINE 4 BORONIC ACID 2 ETHOXYPYRIDINE 4 BORONIC ACID 3 CHLORO 2 METHOXYPYRIDINE 4 BORONIC ACID PINACOL ESTER 3 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID 3 PICOLINE 4 BORONIC ACID HCL 3 BROMO 2 FLUOROPYRIDINE 4 BORONIC ACID PINACOL ESTER 5 pentylpicolinic acid 3 BROMO 5 METHOXY 4 PYRIDINYL BORONIC ACID 2 3 FLUOROPHENYL PYRIDINE 4 BORONIC ACID PINACOL ESTER 2 FLUORO 5 METHYLPYRIDINE 4 BORONIC ACID PINACOL ESTER 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 2 6 PYRIDINEDICARBOXYLIC ACID 2 6 DIMETHYL ESTER 5 BROMO 2 ETHOXYPYRIDINE 4 BORONIC ACID 2 ETHOXYCARBONYL PYRIDIN 4 YL BORONIC ACID

2 CHLORO 3 CYANOPYRIDINE 4 BORONIC ACID 2 PICOLINE 4 BORONIC ACID HCL 3 CYANOPYRIDINE 4 BORONIC ACID 2 AMINO 4 PYRIDYL BORONIC ACID 3 CYANOPYRIDINE 4 BORONIC ACID PINACOL ESTER 3 CHLORO 4 5 5 DIMETHYL 1 3 2 DIOXABORINAN 2 YL PYRIDINE 2 PYRIDINECARBOXAMIDE N 2 CHLORO 4 PYRIDINYL 6 METHYL 4 4 4 5 5 TETRAMETHYL 1 3 2 DIOXABOROLAN 2 YL 3 CHLORO 2 MORPHOLINOPYRIDINE 4 BORONIC ACID 3 CHLORO 2 4 MORPHOLINO PYRIDINE 4 BORONIC ACID PINACOL ESTER 5 6 7 8 tetrahydroimidazo 1 2 a pyrazine 2 carboxylic acid 1 ETHYL 4 TERT BUTYLOXYCARBONYL PIPERAZIN 2 ONE 2 METHYL 3 OXOPIPERAZINE HYDROCHLORIDE 4 4 Difluoro L prolinamide hydrochloride 1 benzyl 3 methylpyrrolidin 3 ol 3 ACETAMIDOPYRROLIDINE 1 tert butyl 2 methyl 2 ethyl 4 oxopyrrolidine 1 2 dicarboxylate 1S tert butyl 6 oxo 5 oxa 2 aza bicyclo 2 2 1 heptane 2 carboxylate 3 methylpyrrolidin 3 ol hydrochloride 7 3 TRIFLUOROMETHYL PHENYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXAMIDE 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDIN 2 AMINE 5 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 OL 6 2 CARBOXYBIPHENYL 4 YL METHYL 7 HYDROXY 5 PROPYLPYRAZOLO 1 5 A PYRIMIDINE 5 7 BIS TRIFLUOROMETHYL 2 METHYLTHIO PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXAMIDE 1 2 4 CHLOROPHENYL 7 METHYLPYRAZOLO 1 5 A PYRIMIDIN 6 YL ETHAN 1 ONE 2 TERT BUTYL 7 CHLORO 5 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 5 7 BIS TRIFLUOROMETHYL 3 CYANOPYRAZOLO 1 5 A PYRIMIDINE 5 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 AMINE 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 2 3 DIAMINE 6 4 METHOXY PHENYL 3 PHENYL PYRAZOLO 1 5 A PYRIMIDINE 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE

2 4 BROMOPHENYL 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 6 BROMO PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 7 AMINO 2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 5 1 METHYL CYCLOPROPYL 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 5 METHYL 3 PHENYL PYRAZOLO 1 5 A PYRIMIDIN 7 YL HYDRAZINE 5 ISOPROPYL 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 6 BROMO 3 CHLOROPYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 6 TERT BUTYLSULFONYL 2 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 AMINE 6 NITROPYRAZOLO 1 5 A PYRIMIDINE 7 CHLORO 5 6 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 6 METHYLPYRAZOLO 1 5 A PYRIMIDINE 5 METHYLPYRAZOLO 1 5 A PYRIMIDINE 2 TERT BUTYL 7 CHLORO 3 IODO 5 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 TERT BUTYL 7 HYDRAZINO 5 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 2 METHYL 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 2 METHOXYMETHYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 7 HYDROXY 2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 5 HYDROXY 2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 7 METHOXY 2 5 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 2 5 7 TRIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 7 PYRIDIN 3 YL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE 2 PHENYL PYRAZOLO 1 5 A PYRIMIDIN 5 OL 4 2 PHENYL 5 7 BIS TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDIN 3 YL PHENOL 7 FURAN 2 YL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE 6 METHYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXYLIC ACID 3 3 4 DIETHOXY PHENYL 6 4 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 5 METHYL 2 PHENYL PYRAZOLO 1 5 A PYRIMIDIN 7 OL 7 AMINOPYRAZOLO 1 5 A PYRIMIDINE 6 CARBONITRILE 1 2 3 5 6 7 HEXAHYDRO 4 8A 9 TRIAZA CYCLOPENTA A S INDACEN 8 YLAMINE 6 4 METHOXY PHENYL 3 THIOPHEN 2 YL PYRAZOLO 1 5 A PYRIMIDINE