3 2 2 dimethoxyethyl thio propene 1H BENZIMIDAZOLE 1 BUTANOIC ACID 2 3 DIHYDRO 2 OX 2 2 diphenyl glycine 2 6 pyridyl diethylazodicarboxylate 4 hydroxy 4 methyl 2 pentanone 1 amino tetrahydronaphthalene 4 cyano biphenyl 1 4 butane sultone 1 3 propane sultone 2 amino 5 chloro benzophenone 7 keto Dehydroepiandrosterone 2 4 hydroxybenzaldehyde 5 methyl pyridin 3 yl methanol chloro 4 6 bis oct thiomethyl o cresol 2 cyanoethyl N N diisopropyl chloro phosphoramidite 3 iodo ethyl propionate 6 Bromo androsterone 2 methyl 3 butyn 2 amine 1 2 3 4 tetrahydro 1 naphthylamine 1 4 dichloro 2 butyne 5 methyl phenazine methosulfate 2 3 Dichloroquinoxaline 2 6 Difluorobenzenesulfonyl chloride 1 3 Thiazol 2 ylmethanol 5 Bromonicotinoylchloride 2 Cyano 3 methylpyridine 1 2 Hydroxy 3 sulfopropyl pyridinium betane 2 amino benzothiazole 3 fluoro 4 pyridinecarboxaldehyde 40273 47 0 3 iodopyridin 2 amine 104830 06 0

3 chloro 4 iodopyridine 77332 79 7 2 3 dichloro 5 trifluoromethyl 4 iodopyridine 3 fluoro 4 iodo pyridine 22282 75 3 3 trifluoromethyl 2 iodopyridine 927434 20 6 2 bromo 6 trifluoromethyl pyridine 189278 27 1 3 chloro 4 pyridinecarboxaldehyde 72990 37 5 2 4 dichloro 3 pyridine Carboxaldehyde 134031 24 6 4 trifluoromethyl 2 pyridinecarboxylic acid 588702 62 9 5 trifluoromethyl pyridine 2 carbaldehyde 31224 82 5 2 bromo 3 trifluoromethyl pyridine 175205 82 0 2 bromo 6 pyridine carboxylic acid 21190 87 4 5 bromo 2 pyridinecarboxaldehyde 31181 90 5 4 iodo 2 trifluoromethyl pyridine 590371 73 6 6 chloropyridine 2 carboxaldehyde 54087 03 5 2 3 difluoro 4 iodopyridine 851386 34 0 6 trifluoromethyl 2 pyridinecarboxylic acid 131747 42 7 6 trifluoromethyl 2 pyridinecarboxaldehyde 131747 65 4 5 bromo 2 pyridinecarboxylic acid 30766 11 1 2 methyl 5 nitropyridine 21203 68 9 5 chloro 2 pyridinecarboxylic acid 86873 60 1 2 chloro 4 hydrazinopyridine 700811 29 6 5 amino 2 methylpyridine 3430 14 6 4 trifluoromethyl 2 hydroxypyridine 50650 59 4 5 bromo 3 pyridinecarboxaldehyde 113118 81 3 2 6 dibromo 3 nitropyridine 55304 80 8 5 chloro 2 fluoro 4 iodopyridine N A 5 trifluoromethyl pyridine 2 carboxylic acid methyl ester 124236 37 9 6 chloro 4 methylpyridine 2 carboxylic acid 324028 95 7 2 bromo 3 chloro 5 trifluoromethyl pyridine 75806 84 7 3 chloro 5 trifluoromethyl pyridine 2 carboxylic acid 80194 18 9

2 chloro 3 bromo 5 trifluoromethyl pyridine 71701 92 3 2 chloro 4 iodo 5 trifluoromethyl pyridine 505084 55 9 5 trifluoromethyl 2 pyridinecarboxylic acid 80194 69 0 3 trifluoromethyl 2 pyridinecarboxylic acid 87407 12 3 5 Chloro 3H iMidazo 4 5 b pyridine 2 Chloro 5 nitronicotinaMide 6 Bromo 2 chloroquinoline 4 Phenylimidazole 2 Amino 2 3 dihydro 1H inden 2 yl phosphonic acid hydrochloride 5 1H Pyrrol 1 yl 2 mercaptobenzimidazole 6 Methylpyridine 2 3 dicarboxylic acid 2 4 Methylphenyl pyridine 3 Pyridylacetic acid hydrochloride 2 4 Dichloro 5 nitropyrimidine 4 Hydroxyindole 6 Chloro 2 3 diaminopyridine 2 Acetyl 5 chlorothiophene 2 chloro 3 nitrothiophene 5 Fluorobenzo 2 1 3 thiadiazole 5 Chloro 4 nitrothiophene 2 sulfonyl chloride 2 5 Dibromopyridine 5 Chlorothiophene 2 sulfonyl chloride 3 Carboxy 4 nitrophenyl disulfide 2 3 5 Triphenyltetrazolium chloride 5 BroMo 6 chloro 3 indoxyl acetate 2 2 Bis hydroxymethyl 2 2 2 nitrilotriethanol 3 4 Dihydroxycinnamic acid 3 4 5 Trihydroxystilbene 3 beta D glucopyranoside 3 Hydroxy 4 iodobenzoic acid 3 METHOXY DL TYROSINE

3 Methyl 5 phenyl 1H pyrazol 4 aMine 3 Fluoro 4 hydroxyacetophenone 3 fluoroazetidine hydrochloride 3 Ethoxy 4 ethoxycarbonyl phenylacetic acid 3 chloro 5 Methoxypyridazine 3 CYANO 4 6 DIMETHYL 2 MERCAPTOPYRIDINE 3 broMo 5 chloropyridine 3 broMo 2 chloro 4 Methoxy Pyridine 3 broMo 2 4 dichloro Pyridine 3 broMo 1H pyrrolo 2 3 b pyridine 3 AMinophthaliMide 3 AMinocyclohexanol 3 AMinoisonicotinic acid 3 AMino 5 Methylthiophene 3 AMino 5 phenyl 2H pyrazole 3 aMino 3 pyridin 3 yl propanoic acid 3 AMino 2 Chloro isonicotinic acid ethyl ester 3 AMino 1 adaMantanol 3 2 4 Cyanophenyl aMino Methyl 1 Methyl 1H benziMidazol 5 yl carbonyl pyridin 2 ylaMino propionic acid ethyl ester 3 5 difluorobenzene 1 2 diaMine 3 5 dichloro 4 3 cyclopropylMethoxy 4 difluoroMethoxy benzaMido pyridine 1 oxide 3 4 bis cyclopropylMethoxy N 3 5 dichloropyridin 4 yl benzaMide 3 cyclopropylMethoxy N 3 5 dichloropyridin 4 yl 4 hydroxybenzaMide 3 3 diMethyl 1 1 diphenyl 1H 1 H 4 4 bipyrazole 5 5 diol 3 cyclopropylMethoxy N 3 cyclopropylMethoxy 4 difluoroMethoxy benzoyl N 3 5 dichloropyridin 4 yl 4 difluoroMethoxy benzaMide 2 4 6 8 Tetraoxa 5 phosphanonanedioic acid 5 1R 2 6 9 2R 5 hydroxy 2 11 diMethyl 5 oxido 9 oxo 3 6 8 10 tetraoxa 5 phosphadodec 1 yl 9H purin 6 yl aMino Methyl aMino 9H purin 9 yl 1 Methylethoxy Methyl 1 9 bis 1 Methylethyl ester 2 4 hydroxy 2 oxopyrrolidin 1 yl acetic acid 2 4 6 8 Tetraoxa 5 phosphanonanedioic acid 5 1R 2 6 aMino 9H purin 9 yl 1 Methylethoxy Methyl 1 Methyl 9 1 Methylethyl ester 5 oxide 2 3 Methyl 5 oxo 1 phenyl 4 5 dihydro 1H pyrazol 4 yl propane 2 sulfonic acid 2 2 oxo 2 5 dihydro 1H pyrrol 1 yl acetaMide