3 Cyanobenzoyl chloride 2 3 chloro 5 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 5 Difluoro 3 nitropyridine 2 2 chloro 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Methyl 4 isoxazolecarboxylic acid 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 4 5 5 tetramethyl 2 2 4 6 trichlorophenyl 1 3 2 dioxaborolane 3 Fluoro 4 hydroxy 5 methoxybenzaldehyde 4 chlorobenzoicanhydride 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 chloro 3 nitrophenol 2 3 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 fluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Methoxyisonicotinic acid 4 chlorobenzofuran 5 bromofuran 2 carbonyl chloride 2 3 5 difluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 fluorobenzofuran 7 carboxaldehyde 2 chloro 6 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 2 chloro 5 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 chloro 5 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 5 methyl 1H pyrazole 2 Iodo 4 nitroaniline 2 4 tert butyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 3 Bromo 5 chlorobenzaldehyde 2 chloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 tert butyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 Fluoropyridine 3 carboxylic acid

4 chloro 4 methylbenzophenone 3 5 difluoro 4 methoxycarbonyl phenyl boronic acid 5 4 fluorophenyl 1H pyrazole 4 chloro 4 fluorobenzophenone 3 Chloro 5 nitrobenzotrifluoride 3 cyano 2 4 difluorophenyl boronic acid 4 hydroxy 2 trifluoromethyl phenyl boronic acid 4 1 methoxycarbonyl cyclopropyl phenyl boronic acid 2 3 5 Tribromopyridine 1 4 boronophenyl cyclopropanecarboxylic acid 3 4 dimethylphenyl boronic acid 2 methoxy 3 trifluoromethyl phenyl boronic acid 3 Aminopropylphosphonic acid 2 bromo 5 trifluoromethoxy aniline 4 fluoro 3 methoxyphenyl boronic acid 2 6 difluoro 4 methoxyphenyl boronic acid 1 2 Bis bromomethyl benzene 4 chloro 2 3 difluorophenyl boronic acid 2 fluoro 5 methylphenyl boronic acid 5 chloro 2 methoxyphenyl boronic acid 5 Bromo 3 methylthiophene 2 carboxylic acid 3 Methyl thiophene 2 carboxylic acid methyl ester 5 chloro 2 methoxymethoxy phenyl boronic acid 2 chloro 3 methoxyphenyl boronic acid 2 fluoro 4 methoxyphenyl boronic acid 5 bromo 3 fluoro 2 pyridinone 1 4 Cyclohexanedione monoethyleneacetal 3 chloro 5 fluoro 4 hydroxyphenyl boronic acid 3 chloro 5 fluorophenyl boronic acid 2 fluoro 4 hydroxyphenyl boronic acid

2 chloro 5 hydroxyphenyl boronic acid 2 hydroxy 5 methylphenyl boronic acid 2 hydroxy 4 methylphenyl boronic acid 4 Bromo 2 3 difluoroaniline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzofuran 3 2H one 2 3 Dihydro 1 4 benzodioxine 5 carboxylic acid 2 Amino 6 chlorobenzoic acid 1 chloro 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoquinoline 4 Chloropyridin 2 yl methanol 8 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinolin 4 ol 2 Amino 3 trifluoromethyl pyridine 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 amine 3 Amino 2 6 dibromopyridine 2 3 dihydrobenzofuran 4 yl boronic acid 5 Methoxy 2 3 4 trifluorobenzoic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 amine 4 4 Bipyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazol 2 amine 3 Azabicyclo 3 3 0 octane hydrochloride 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 4 isothiocyanato 1 2 dimethylbenzene 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 5 Aminopyrimidine 2 carbonitrile 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 amine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 4 2 Aminoethyl tetrahydropyran 1H indazol 6 yl boronic acid 3 Chloro 4 phenoxyaniline hydrochloride

4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 7 trifluoromethyl 1H indazole 3 methyl 1H indazol 6 yl boronic acid 2 Bromo 6 chloropyridine 3 methyl 1H indazol 5 yl boronic acid 1 Boc 2 methoxycarbonylmethylpiperazine 3 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 6 fluoro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 4 amino 2 chloro 3 fluorophenol 2 Pyrimidinecarboxylic acid 1 methyl 1H indazol 4 yl boronic acid 5 Chloro 2 iodophenol 3 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 methoxymethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 3 Dichloro 2 methyl 5 nitrobenzene 3 Amino 6 chloropyridazine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinamide 3 Methyl 6 nitro 1H indazole 2 6 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Amino 5 Bromo 3 Hydroxymethyl Pyridine 4 4 5 5 tetramethyl 2 3 methylbenzofuran 5 yl 1 3 2 dioxaborolane 2 Mercapto 5 trifluoromethylpyridine 2 7 chlorobenzofuran 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Hydroxy 3 nitro 5 trifluoromethyl pyridine 6 Benzylaminopurine 4 Chloro 3 nitropyridine 6 fluorobenzo b thiophen 7 yl boronic acid 3 Fluoro 4 methylpyridine 3 acetylthiophen 2 yl boronic acid 2 6 Dichloro 3 nitropyridine