1 Amino 1H pyrrole 2 carboxamide 1 2 Bis 2S 5S 2 5 diethylphospholano ethane 5 6 7 8 Tetrahydro 1 6 naphthyridin 3 ol 6 Amino 2 methylquinoline 6 bromo 5 methoxypyridine 2 carboxylic acid 3 Fluoro 4 hydroxyacetophenone 8 Benzyl 2 8 diazaspiro 4 5 decane 2 Chloro 5 Fluoropyrimidin 4 One 1 3 Dibromo 5 iodobenzene 2 methylthio pyrimidin 4 amine 5 amino 3H 1 3 thiazole 2 thione 4 Chloro 6 methylquinoline 2 HYDROXY 3 4 DIMETHOXYBENZOIC ACID 5 Bromo 2 2 methyl 2H tetrazol 5 yl pyridine 3 Bromo 5 Nitrotoluene 5 6 N SUCCINIMIDYLOXYCARBONYL 3 6 O O DIACETYLFLUORESCEIN 3 IODOPROPIONIC ACID 2 Chloro 4 Methoxycarbonyl Benzeneboronic Acid 2 Oxo 3 3 trifluoromethyl phenoxy propyl phosphonic Acid Dimethyl Ester 3 AMINO 5 METHYL 4 PHENYLPYRAZOLE 2 amino 1 3 thiazole 4 carbonitrile 2 6 Dichlorophenylhydrazine hydrochloride 3 methyl 5 nitro 2H pyrazolo 3 4 b pyridine 1 benzylindol 5 amine 2 Bromo 5 iodothiophene 3 hydroxythiophene 2 carboxylic acid 3 5 Dimethyl 4 Isoxazolecarbaldehyde 5 Bromo 1H benzimidazole 6 Methyl 4 azaindole 3 carboxaldehyde 6 Nitro 1H indole 4 carboxylic acid

6 Chloro 2 Methyl 1H indole 4 carboxylic acid Methyl ester 4 Chloro 3 methylisoxazol 5 amine 2 methoxy 5 methyl 3 nitropyridine 2 methoxy 4 propylphenol 1 nitro 4 2 4 nitrophenyl ethyl benzene 5 chloro 6 methoxy 2 3 dihydroinden 1 one 2 Chloromethyl 6 Methylpyridine 3 Amino 5 bromo 4 hydroxybenzoic acid 1 O benzyl 3 O ethyl 4 oxopiperidine 1 3 dicarboxylate 6 7 dihydro 5H cyclopenta b pyridin 7 ol 6 trifluoromethyl pyridine 2 3 diamine 2 6 Dichloro 3 Nitro Benzyl Alcohol 3 2 Methylphenyl propionic acid 6 Bromophthalazin 1 2H One 6 chloro N pentylpyridazin 3 amine 1 3 chloropropyl 4 methylpiperazine dihydrochloride 7 CHLORO 5 METHYLPYRAZOLO 1 5 A PYRIMIDINE 2 methylbenzenecarbothioamide 3 Bromo 5 iodopyridine 1 2 5 bis trifluoromethyl phenyl ethanone 2 3 Difluoro 4 methoxybenzaldehyde 1 1 methylpiperidin 4 yl piperazine 1 chloro 4 fluorophenyl phenylmethyl 4 fluorobenzene 4 5 6 7 Tetrahydrobenzo b thiophene 2 carboxylic acid 3 Benzyloxybenzaldehyde 2 pyrrolidin 1 yl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 bromo 5 methylaniline hydrochloride 2 3 dimethylamino 6 dimethylazaniumylidenexanthen 9 yl 5 isothiocyanatobenzoate 1R 2R Boc Acpc 2 FLUORO 4 NITROBENZONITRILE

2 1 Pyrrolidinyl benzaldehyde 2 3 5 Trichlorothiophene 4 Bromo 6 fluoro 2 3 dihydro 1H inden 1 one 1 Chloro 4 2 chloroethoxy benzene 6 7 dihydropyrido 2 3 d pyridazine 5 8 dione 1H Pyrrolo 2 3 b pyridine 2 carbaldehyde 3 Chloro 2 methoxypyridin 4 yl boronic acid 3 5 Dibromoisonicotinic Acid 7 chloro 1H quinazolin 4 one 2 chloro 4 methyl 1 3 thiazole 5 sulfonamide 5 acetyl 2 methylfuran 3 carbonitrile 7 Bromoquinolin 2 1H one 2 Bromo 4 chlorobenzonitrile 2 Pyridineacetic Acid Methyl Ester 5 isocyanato 2 3 dihydro 1H indene 1R 3R 3 1Z 2 Chloro 3 3 3 trifluoro 1 propen 1 yl 2 2 dimet hylcyclopropanecarboxylic acid 2 pyrazol 1 ylaniline 2 1H imidazol 2 yl pyridine 1 3 5 tris 3 trimethoxysilylpropyl 1 3 5 triazinane 2 4 6 trione 1 benzotriazol 1 yl octan 1 one 2 4 Mesitylenedisulfonyl Dichloride 2 AMINO 5 CHLOROBENZOPHENONE OXIME 2S 6 methoxy 1 2 3 4 tetrahydronaphthalen 2 amine 6 7 Dimethoxy 2 4 nitrophenethyl 1 2 3 4 tetrahydroisoquinoline 2 AMINO 2 4 METHOXYPHENYL ACETIC ACID 3 3 Amino 4 bromophenyl propanoic acid 3 S Methoxycarbonyl 4 t butoxycarbonylmorpholine 3S 3 Methylpyrrolidine 2 3 Methoxybenzyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 6 fluoro 1 2 methylpropan 2 yl oxycarbonyl indol 2 yl boronic acid

2 3 DIHYDRO 1 4 BENZODIOXINE 5 CARBOXAMIDE 2 AMINO N 2 BROMOPHENYL BENZAMIDE 4 9H Carbazol 9 yl phenyl boronic acid 5 fluoro 2 3 dimethyl 1H indole 1 3 bis 2 4 6 trimethylphenyl 4 5 dihydroimidazol 1 ium tetrafluoroborate 5 chlorosulfonyl 2 ethoxybenzoic acid 4 methoxyfuro 2 3 b quinoline 5 7 DIMETHYLPYRAZOLO 1 5 A PYRIMIDINE 2 CARBOXYLIC ACID 1R 2R 2 methylsulfonyloxymethyl cyclohexyl methyl methanesulfonate 4 Hydroxypyrimidine 5 carbonitrile 1 3 benzothiazole 2 6 diamine 1 3 ditert butylimidazol 1 ium tetrafluoroborate 4 chloro 1 3 thiazole 5 carboxylic acid 1 benzenesulfonyl 2 iodopyrrolo 2 3 b pyridine 5 6 Dihydro 4H pyrrolo 1 2 b pyrazole 2 carboxylic acid 5H benzo c 1 benzazepine 6 11 dione 1S 4S 2 Methyl 2 5 diazabicyclo 2 2 1 heptane 4 methylamino cyclohexan 1 one 2 Chloro 5 Methylbenzoic Acid 3 3 Dichloro 1 4 iodophenyl 2 piperidinone 2 Chloro 4 fluoro 1 iodobenzene 4 diethylamino 2 methoxybenzaldehyde 3 3 Cholamidopropyl dimethylammonium 1 propanesulfonate 4 4 2 2 Propanediyl dicyclohexanamine 2 Amino 5 bromo 4 6 dimethylpyridine 4 Nitrophenylhydrazine Hydrochloride 1 2 dihydropyrazolo 3 4 b pyridin 3 one 7 Chloroquinoline 3 carboxylic acid 1 tert Butyloxycarbonyl 4 3 aminopropyl piperazine 2 Acetyl 5 chlorothiophene