5 METHOXY 2 TRIFLUOROMETHOXY PHENYLBORONIC ACID 1 6 BROMO PYRIDIN 2 YL 2 2 2 TRIFLUORO ETHANOL 2 6 DIFLUORO 4 1 HYDROXY 1 METHYL ETHYL PHENYL ACETALDEHYDE 4 TRIFLUOROMETHYL ISOINDOLINE 3 3 FLUOROPHENYL CYCLOBUTANONE 1 4 CHLORO PYRIMIDIN 2 YL 2 2 2 TRIFLUORO ETHANOL 4 4 CHLORO PYRIMIDIN 2 YLMETHYL 3 FLUOROMETHYL MORPHOLINE 1 7 FLUORO 1 BENZOFURAN 2 YL ETHAN 1 ONE 2 FLUORO PYRIDIN 4 YL ACETIC ACID TERT BUTYL ESTER 3 BROMO 5 FLUORO ISONICOTINIC ACID TERT BUTYL ESTER 2 CHLORO 6 FLUORO 3 FORMYL BENZOIC ACID 3 BROMO 6 5 TRIFLUOROMETHYL 1H PYRAZOL 3 YL PYRIDINE 2 CARBOXYLIC ACID ETHYL ESTER 2 2 4 6 TRIFLUOROPHENYL ACETALDEHYDE 6 PERFLUOROETHYL NICOTINIC ACID 5 CHLOROMETHYL 4 METHYL 2 TRIFLUOROMETHYL THIAZOLE 2 3 FLUORO PHENYL CYCLOPROPANECARBOXYLIC ACID 2 2 CHLOROPHENYL 2 2 DIFLUOROACETIC ACID 2 CHLORO 4 FLUORO 1 3 BENZOXAZOLE 7 FLUORO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 6 FLUORO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 1R 1 2 FLUOROPHENYL PROPYLAMINE 1 BROMOMETHYL 4 TRIFLUOROMETHYLSULFONYL BENZENE 3 FLUORO 4 HYDROXY PYRROLIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 8 IODO 2 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 6 TRIFLUOROMETHYL FURO 2 3 B PYRIDIN 3 ONE 4 BROMO 5 FLUORO 1 METHYL 1H PYRIDIN 2 ONE 3 2 2 2 TRIFLUORO ETHYL 4 5 6 7 TETRAHYDRO 1H INDAZOLE 6 TRIFLUOROMETHYL 2 3 DIHYDRO FURO 2 3 B PYRIDIN 3 YLAMINE 3 5 3 TRIFLUOROMETHYL PHENYL TETRAHYDRO FURAN 2 YL PROPIONIC ACID 5 TRIFLUOROMETHYL 3 TERT BUTYL OXYCARBONYL AMINO PHENYLBORONIC ACID

3 5 3 5 BIS TRIFLUOROMETHYL PHENYL TETRAHYDROFURAN 2 YL PROPANOIC ACID 1 4 FLUOROPHENYL 2 PHENYLPYRROLIDINE 3 CARBOXYLIC ACID 7 BROMO 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 1 CHLORO 7 TRIFLUOROMETHOXY ISOQUINOLINE 3 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 2 CARBOXYLIC ACID METHYL ESTER 8 BROMO 2 TRIFLUOROMETHYL H IMIDAZO 1 2 A PYRIDINE 4 CHLORO 1 ETHYL 6 TRIFLUOROMETHYL 1H PYRAZOLO 3 4 B PYRIDINE 5 CARBOXYLIC ACID ETHYL ESTER 4 BENZYLOXY 1 2 FLUOROPYRIDIN 4 YL PYRIDIN 2 1H ONE 2 BROMO 6 TRIFLUOROMETHYL ISONICOTINIC ACID METHYL ESTER 2 CHLORO 6 4 3 FLUOROPHENYL 1H IMIDAZOL 2 YL PYRIDINE 3 2 CHLORO 5 FLUORO PHENOXY AZETIDINE 3 TRIFLUOROMETHYL 1 5 6 7 TETRAHYDRO INDAZOL 4 ONE 4 FLUORO 5 METHANESULFONYL 2 3 DIHYDRO 1H INDOLE HCL SALT 3 fluoroazetidin 3 yl methanol 1 tert butyl 4 ethyl 3 fluoropiperidine 1 4 dicarboxylate 4 4 difluoropiperidine 3 carboxylic acid 2 2 DIFLUORO 2 P TOLYLACETIC ACID 2 PENTADECAFLUOROHEPTYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 4 4 bromophenyl 3 fluoropiperidine 4 4 bromophenyl 3 3 difluoropiperidine 3 fluoro tetrahydro 2H pyran 4 amine hydrochloride 2 CHLORO 6 7 DIFLUOROQUINOXALINE 7 BROMO 5 FLUORO 2 METHYL BENZOFURAN 4 YLAMINE 3S 4R 3 fluoro tetrahydro 2H pyran 4 amine hydrochloride 3 4 FLUOROPHENYL CYCLOBUTANONE 2 amino 5 fluoro Benzaldehyde 5 FLUORO 3 PIPERAZIN 1 YLMETHYL 1H INDOLE 6 FLUORO INDAN 1 YLAMINE 2 3 CHLORO PROPENYL 1 4 DIFLUORO BENZENE 2 amino 4 fluoro Benzaldehyde

2 Nitro 1 4 nitrophenoxy 4 trifluoromethyl benzene 2 CHLORO 6 FLUORO 1 3 BENZOXAZOLE 2 CHLORO 7 FLUORO 1 3 BENZOXAZOLE 4 4 FLUORO BENZOYL THIOPHENE 3 CARBOXYLIC ACID 3 3 DIFLUORO PYRROLIDINE 4 CHLORO 6 FLUOROPYRIDO 3 4 D PYRIMIDINE 2 2 difluorohexanoic acid 4 FLUORO PHENYL ACETALDEHYDE 3 4 FLUORO PHENYL 2 2 DIMETHYL CYCLOPROPANECARBOXYLIC ACID 6 FLUORO 3 NITRO PYRIDINE 2 CARBONITRILE 4 TRIFLUOROMETHYL PYRROLIDIN 3 YL METHANOL HYDROCHLORIDE 1 BENZYL 4 TRIFLUOROMETHYL PYRROLIDIN 3 YL METHANOL 9 4 bromobutyl N 2 2 2 trifluoroethyl 9H fluorene 9 carboxamide 4 CHLORO 6 FLUOROPYRIDO 3 2 D PYRIMIDINE 9 4 4 aminopiperidin 1 yl butyl N 2 2 2 trifluoroethyl 9H fluorene 9 carboxamide dihydrochloride 2 2 2 TRIFLUORO 1 4 IODO PHENYL ETHANONE 4 4 DIFLUORO 2 HYDROXYMETHYL PYRROLIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 2 Methyl N 3 trifluoromethyl phenyl propanamide 2 4 TRIFLUOROMETHYL PHENYL CYCLOPROPANECARBALDEHYDE 6 FLUORO 2 3 DIHYDRO BENZO 1 4 DIOXIN 2 YL METHANOL 5 TRIFLUOROMETHYL ISOINDOLINE 2 IODO 4 TRIFLUOROMETHYL PYRIDINE 3 AMINO 6 METHYL 4 TRIFLUOROMETHYL THIENO 2 3 B PYRIDINE 2 CARBOXYLIC ACID METHYL ESTER 1S 4S 2 3 FLUOROPHENYL 2 5 DIAZABICYCLO 2 2 1 HEPTANE HYDROBROMIDE 1 trifluoromethyl cyclobutanecarboxylic acid 1 TRIFLUOROMETHYL CYCLOPENTANE 1 CARBOXYLIC ACID 2 4 FLUOROPHENYL CYCLOPROPANECARBALDEHYDE 7 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIMIDINE 1S 1 4 FLUOROPHENYL PROPYLAMINE 1S 2 2 2 TRIFLUORO 1 5 METHYL 2 FURYL ETHYLAMINE

1 trifluoromethyladamantane 5 CHLORO 3 FLUORO 2 HYDROXY BENZALDEHYDE 1R 2 2 2 TRIFLUORO 1 5 METHYL 2 FURYL ETHYLAMINE 2S 4R methyl 4 fluoropyrrolidine 2 carboxylate hydrochloride 1 5 FLUORO 3 METHYL 1 BENZOFURAN 2 YL ETHAN 1 ONE 4 CHLORO 5 FLUOROQUINAZOLINE HYDROCHLORIDE 1 CHLORO 6 TRIFLUOROMETHOXY ISOQUINOLINE 1 CHLORO 5 TRIFLUOROMETHOXY ISOQUINOLINE 7 TRIFLUOROMETHYL 1 2 3 4 TETRAHYDRO 5 NITROISOQUINOLINE HYDROCHLORIDE 1 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRAZIN 3 YL ETHANONE 4 CHLOROMETHYL 2 2 FLUORO PHENYL 5 METHYL OXAZOLE 2 FLUOROCYCLOHEXANONE 3 CHLORO 6 4 FLUORO PHENYL 1 2 4 TRIAZINE 3 4 FLUOROPHENOXY AZETIDINE 6 FLUORO QUINOLINE 3 CARBOXYLIC ACID ETHYL ESTER 7 TRIFLUOROMETHYL QUINOLINE 3 CARBOXYLIC ACID ETHYL ESTER 3 CHLORO 4 IODO 2 TRIFLUOROMETHYL PYRIDINE 2 BROMO 4 IODO 6 TRIFLUOROMETHYL PYRIDINE 2 BROMO 6 TRIFLUOROMETHYL ISONICOTINIC ACID 6 BROMO 2 TRIFLUOROMETHYL 3 PYRIDINECARBOXYLIC ACID 5 BROMO 3 1 2 6 DICHLORO 3 FLUOROPHENYL ETHOXY PYRIDIN 2 AMINE 2 IODO 4 TRIFLUOROMETHYL NICOTINIC ACID 2 4 FLUORO PHENYL 1 METHYL 5 OXO PYRROLIDINE 3 CARBOXYLIC ACID 1 2 4 BROMO 2 FLUORO PHENYL ETHYL 6 7 DIMETHOXY 1 2 3 4 TETRAHYDRO ISOQUINOLINE 1H INDOLE 7 FLUORO 2 3 DIHYDRO 6 4 FLUORO PHENYL IMIDAZO 2 1 B OXAZOLE 5 BROMO 2 CHLORO 4 TRIFLUOROMETHYL QUINOLINE 7 BROMO 2 CHLORO 4 TRIFLUOROMETHYL QUINOLINE 6 FLUORO 2 3 4 9 TETRAHYDRO 1H CARBAZOL 3 YLAMINE 6 TRIFLUOROMETHYL QUINOLINE 2 CARBOXYLIC ACID