1S 2R 5R 3 AZA BICYCLO 3 1 0 HEXANE 2 3 DICARBOXYLIC ACID 3 TERT BUTYL ESTER 6 Bromo 2 fluoro 3 methoxybenzaldehyde 3 Bromo 2 chloro 6 fluorobenzoic acid 1 BENZYL 4 4 DIPHENYLPIPERIDINE 6 Bromo 2 fluoro 3 propoxybenzaldehyde 1 BOC 4 2 FLUOROPHENYL 4 HYDROXYPIPERIDINE 4 Benzyloxy 3 fluorobenzaldehyde 4 4 BIS 4 CHLOROPHENYL PIPERIDINE 5 FLUORO 1 2 3 4 TETRAHYDRO ISOQUINOLINE 3 Bromo 6 chloro 2 fluorobenzoic acid 6 Bromo 3 chloro 2 fluorobenzaldehyde 3 5 Dibromo 1 fluoro 4 isopropoxybenzene 2 4 PHENYLPIPERIDIN 1 YL ETHANAMINE 3 Chloro 2 iodobenzotrifluoride 2 3 DIHYDROSPIRO INDENE 1 4 PIPERIDINE 5 Benzyloxy 2 bromobenzotrifluoride 1 5 METHYL FURAN 2 CARBONYL PIPERIDINE 2 CARBOXYLIC ACID 5 Bromo 2 trifluoromethoxy benzoic acid 2R 4R 1 TERT BUTOXYCARBONYL 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID 3 Bromo 2 trifluoromethoxy benzoic acid 2S 4S N BOC 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID BENZYLAMINE SALT 2R 4R BOC 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID BENZYLAMINE SALT 3 5 Dibromo 2 iodopyridine 2 Chloro 6 iodopyridine 2 TRIFLUOROMETHYL 1 2 3 4 TETRAHYDRO QUINOLINE 2 Bromo 5 chloro isonicotinic acid 1 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine 5 Bromo pyridine 2 carboxylic acid t butyl ester 6 Bromo 7 methylimidazo 1 2 a pyridine hydrochloride 4 BENZYL PIPERIDINONE 3 FLUORO

2 PIPERIDINONE 3 FLUORO 2 Ethoxypyridine 3 carbaldehyde 2 Bromo 5 formyl 3 methylpyridine 5 Carboxy 2 chloro 3 methylpyridine 2 METHYL N 4 METHYL 3 4 PIPERIDINYL PHENYL PROPANAMIDE 5 Bromo 3 methyl 2 pyridinecarbaldehyde 1S 2R 5R 2 HYDROXYMETHYL 5 ETHYNYLQUINUCLIDINE 2 Fluoro 4 iodo 5 methyl 3 pyridinecarboxaldehyde 1 AZABICYCLO 2 2 2 OCTANE 2 CARBOXYLIC ACID 3 Fluoro 4 trimethylsilyl pyridine 5 Formyl 2 methoxy 4 picoline 4 CYANO 4 PHENYLPIPERIDINE HYDROCHLORIDE 2 Chloro 5 methylpyridine 3 carbaldehyde 4 Chloro 5 fluoropyridine 3 carboxylic Acid 4 PIPERIDIN 4 YL ANILINE HYDROCHLORIDE 2 6 Dibromo 3 fluoropyridine 3 Bromo 2 bromomethyl 6 fluoropyridine 1 BENZYL 4 CYANO 4 PHENYLPIPERIDINE HYDROCHLORIDE 5 Bromo N N diethyl 3 pyridinecarboxamide 2 PIPERIDIN 4 YL 6 TRIFLUOROMETHYL 1H BENZOIMIDAZOLE 2 6 Dichloro 3 hydroxypyridine 2 4 PHENYLPIPERIDIN 1 YL ETHANOL 5 Bromopyridin 3 yl morpholin 4 yl methanone 4 4 METHYLPHENYL PIPERIDIN 4 OL 5 Bromo N methylpyridine 2 carboxamide 7 METHYL 2 INDOLINONE 3 SPIRO 4 N ETHYLPIPERIDINE 5 Bromo N isopropylpyridine 2 carboxamide 2 INDOLINONE 3 SPIRO 4 N ETHYLPIPERIDINE 2 5 Dichloro 4 hydroxypyridine 1 BOC 4 CYANO 4 3 FLUOROPHENYL PIPERIDINE

3 Fluoro 2 methylphenylboronic acid pinacol ester 7 OXO 3 TRIFLUOROMETHYL 5 6 7 8 TETRAHYDRO 1 6 NAPHTHYRIDINE 8 CARBOXYLIC ACID TERT BUTYL ESTER 1 2 Chloro 3 fluoropyridin 4 yl ethanone 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl benzaldehyde 2 5 Dibromophenylboronic acid pinacol ester 2 6 DIOXO PIPERIDIN 4 YL ACETIC ACID 4 O TOLYL PIPERIDINE 2 4 Methoxy 3 methylthio phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 6 Difluoro 4 isopropoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 BOC 4 3 TRIFLUOROMETHYL PHENYL 4 HYDROXYPIPERIDINE 1 BOC 4 CYANO 4 3 TRIFLUOROMETHYLPHENYL PIPERIDINE 2 4 benzyloxy 3 ethylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Ethyl 4 methoxyphenylboronic acid 2 Methyl 4 trifluoromethyl phenylboronic acid pinacol ester 1 BOC 4 CYANO 4 2 TRIFLUOROMETHYLPHENYL PIPERIDINE 2 3 DIHYDRO 2 OXOSPIRO PIPERIDINE 4 4 1H QUINAZOLINE 3 Aminocarbonylphenylboronic acid pinacol ester 3 Bromo 5 isopropylphenylboronic acid pinacol ester 4 Methoxy 3 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 1 TERT BUTOXYCARBONYL 4 4 CHLOROPHENYL PIPERIDINE 4 CARBOXYLIC ACID 9 Phenyl 9H carbazol 3 yl 3 boronic acid pinacol ester 4 4 DIPHENYLPIPERIDINE HYDROCHLORIDE 3 Trifluoromethyl 5 fluorophenylboronic acid pinacol ester 5 Acetylthiophene 3 boronic acid pinacol ester 1 TERT BUTOXYCARBONYL 4 4 FLUOROPHENYL PIPERIDINE 4 CARBOXYLIC ACID 2 1 TERT BUTOXYCARBONYL 4 PHENYLPIPERIDIN 4 YL ACETIC ACID 4 Fluoro 2 trifluoromethyl phenylboronic acid pinacol ester 1 3 4 AMINOPHENOXY 2 HYDROXYPROPYL 4 PHENYL 4 PIPERIDINYL ETHANONE 4 Methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 2 3 Dichlorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane

3 5 Dibromophenylboronic acid pinacol ester 1 4 METHOXYPHENOXY 3 4 2 METHOXYPHENYL PIPERIDINO PROPAN 2 OL 2 2 4 Dichloro 3 fluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2S 4R FMOC 4 HYDROXYPIPERIDINE 2 CARBOXYLIC ACID 2 4 Bromo 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 Dichloro 4 methylphenylboronic acid 1 BENZYL PIPERIDINE 2 CARBOXYLIC ACID HYDROCHLORIDE 2 4 Bromo 2 5 dimethylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 BOC 4 CYANO 4 3 4 DIMETHOXYPHENYL PIPERIDINE 2 Chloro 3 fluorophenylboronic acid pinacol ester 3 Hydroxymethyl 4 methoxyphenylboronic acid pinacol ester 1 BOC 4 CYANO 4 3 CYCLOBUTYLOXY 4 METHOXYPHENYL PIPERIDINE 1 BOC 4 CYANO 4 3 4 CHLOROPHENYL PIPERIDINE 3 Chloro 2 4 difluorophenylboronic acid pinacol ester 4 Methoxy 3 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 AMINO 4 3 BROMO PHENYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 4 Chloro 2 methylphenylboronic acid pinacol ester 4 4 ethylphenyl piperidine 4 Carboxy 2 nitrophenylboronic acid pinacol ester 3 AMINO 5 FLUORO 3 4 DIHYDRO 1H QUINOLIN 2 ONE 2 5 Bromo 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Ethylphenylboronic acid pinacol ester 1 PIPERIDINEACETAMIDE N 3 METHYLPHENYL AMINO CARBONYL 4 PHENYL 1 ETHYL PIPERIDINE 2 CARBOXYLIC ACID 2 4 Bromonaphthalen 1 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Fluoro 6 trifluoromethyl phenylboronic acid pinacol ester 2 4 Bromo 2 6 difluorophenyl 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Chloro 4 methylthio phenylboronic acid pinacol ester 2 6 Dimethyl 4 cyanophenylboronic acid pinacol ester 3 Formyl 4 methoxyphenylboronic acid pinacol ester