1 1 ADAMANTYLMETHYL PIPERAZIN 4 IUM CHLORIDE 1 ISOPROPYLADAMANTANE 1 CHLOROMETHYL ADAMANTANE 1 PHENYLADAMANTANE 1 2 CHLOROETHYL TRICYCLO 3 3 1 13 7 DECANE 4 hydroxy 1 hydroxymethyladmantane 4 AMINO 1 ADAMANTANECARBOXYLIC ACID 2 ADAMANTYL 4 BROMO 1 2 2 2 TRIFLUOROETHOXY BENZENE 1 adamantaneethylsulfonamide 4 HYDROXY 4 METHOXY 3 ADAMANTANE 1 CARBOXYLIC METHYL ESTER 7 methylenebicyclo 3 3 1 nonan 3 one oxime 1 hydroxymethyl 4 oxoadamantane 3 methoxy 1 hydroxymethyladamantane 1 Hydroxymethyladamantan 4 one Ethylene Ketal 1 hydroxymethyl 3 methyl 2 oxadamantane 3 BROMO 2 5 DIMETHYL 4 4 TRIFLUOROMETHYL BENZYL THIOPHENE 4 FLUORO 3 FORMYLBENZAMIDE 2 fluoro 6 trifluoromethylbenzyl chloride 7 hydroxymethyl 2 4 dimethylbicyclo 3 3 1 nonan 3 one 3 AMINO 6 FLUORO 1 2 3 4 TETRAHYDRO CARBAZOL 9 YL ACETIC ACID ETHYL ESTER 4 FLUORO 3 5 DIMETHYL 1H PYRROLE 2 CARBOXYLIC ACID ETHYL ESTER 2 4 METHANESULFONYL PHENYL 5 TRIFLUOROMETHYL 2H PYRAZOL 3 OL 8 CHLORO 2 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 4 FLUORO 7H PYRROLO 2 3 D PYRIMIDINE 6 CARBOXYLIC ACID 5 5 difluoro 2 2 dimethyl 1 3 dioxane 4 6 dione 4 CHLORO 5 FLUORO 2 METHOXYMETHYL PYRIMIDINE 3 BROMO 6 TRIFLUOROMETHYL THIENO 2 3 B PYRIDINE 2 CARBOXYLIC ACID ETHYL ESTER 6 FLUORO 3 IODO PYRAZOLO 1 5 A PYRIMIDINE 7 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 C PYRIMIDIN 5 OL 2 3 DIHYDROSPIRO 6 TRIFLUOROMETHYLBENZOFURAN 2 3 PYRROLIDINE

2 BROMO 5 FLUORO 4 IODOPYRIDINE 2 CHLORO 5 TRIFLUOROMETHYL PYRIDIN 4 YLAMINE 5 CHLOROMETHYL 3 1 2 FLUORO PHENYL CYCLOPROPYL 1 2 4 OXADIAZOLE 5 BROMO 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 3 FLUOROPHENOXY AZETIDINE 6 CHLORO 2 FLUORO NICOTINIC ACID METHYL ESTER 3 4 BROMO PHENYL 3 FLUORO OXETANE 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 B PYRIDAZINE 3 3 TRIFLUOROMETHYL PHENYL CYCLOBUTANONE 3 4 TRIFLUOROMETHYL PHENYL CYCLOBUTANONE 3 2 6 DIFLUORO PHENYL CYCLOBUTANONE 6 CHLORO 2 FLUORO 3 METHANESULFONYL PYRIDINE 6 CHLORO 2 FLUOROPYRIDINE 3 CARBOXALDEHYDE 4 CHLORO 2 FLUOROMETHYL PYRIMIDINE 1 6 CHLORO 2 METHYL PYRIDIN 3 YL 2 2 2 TRIFLUORO ETHANOL 1 TRIFLUOROMETHYL CYCLOPROPANAMINE 2 TERT BUTOXYCARBONYLAMINO 4 4 4 TRIFLUORO 3 TRIFLUOROMETHYL BUTYRIC ACID 5 FLUORO 2 METHOXYMETHYL PYRIMIDIN 4 OL 4 CHLORO 7 TRIFLUOROMETHOXY QUINAZOLINE 8 FLUORO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID 1 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDIN 3 YL ETHANONE 1 3 Dichlorotetrafluorobenzene 1 3 dichloro 2 4 5 6 tetrafluoro Benzene 1 CHLORO 6 TRIFLUOROMETHYL ISOQUINOLINE 1 CARBOXYMETHYL 3 TRIFLUOROMETHYL 1 4 5 7 TETRAHYDRO PYRAZOLO 3 4 C PYRIDINE 6 CARBOXYLIC ACID TERT BUTYL ESTER 8 FLUORO 7 IODO 2 METHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 5 CHLORO 7 TRIFLUOROMETHYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXYLIC ACID METHYL ESTER 8 TRIFLUOROMETHYL H PYRROLO 1 2 A QUINOXALINE 7 FLUORO PYRROLO 1 2 A QUINOXALINE 4 METHYL 2 TRIFLUOROMETHYL THIAZOL 5 YL METHANOL 6 BROMO 5 4 FLUORO BENZENESULFONYL 1 3 DIHYDRO INDOL 2 ONE

4 FLUORO 2 3 DIHYDRO 1H INDOLE 4 FLUORO 5 HYDROXY AZEPANE 1 CARBOXYLIC ACID TERT BUTYL ESTER 8 8 DIMETHYL 3 TRIFLUOROMETHYL 5 6 7 8 TETRAHYDRO 1 6 NAPHTHYRIDINE 4 METHYL 1 5 TRIFLUOROMETHYL PYRIDIN 2 YL PYRROLIDINE 3 CARBOXYLIC ACID 2 2 difluoro 1 3 propanediol 1 3 cyclic sulfate 5 BROMO 2 TRIFLUOROMETHYL ISONICOTINIC ACID METHYL ESTER 5 7 DICHLORO 2 TRIFLUOROMETHYLPYRAZOLO 1 5 A PYRIMIDINE 5 7 DICHLORO 3 TRIFLUOROMETHYLPYRAZOLO 1 5 A PYRIMIDINE 6 BROMO 2 TRIFLUOROMETHYL NICOTINIC ACID METHYL ESTER 3 4 FLUORO BENZOYL PYRIDINE 2 CARBOXYLIC ACID 2 BROMO 4 TRIFLUOROMETHYL NICOTINIC ACID METHYL ESTER 7 FLUORO 2 3 DIHYDRO BENZOFURAN 4 OL 4 5 DIBROMO 2 TRIFLUOROMETHYL BENZONITRILE 5 3 BENZYLOXYCARBONYLAMINO PYRROLIDIN 1 YL 4 FLUORO 1 METHYL 1H PYRAZOLE 3 CARBOXYLIC ACID ETHYL ESTER 2 BROMO 3 CHLORO 4 FLUORO 6 NITRO PHENOL 4 CYCLOPROPYLMETHOXY 3 TRIFLUOROMETHYL PHENOL 5 FLUORO 6 METHYL PYRIDINE 2 CARBOXYLIC ACID METHYL ESTER 4 FLUORO 3 ISOPROPYL BENZYLAMINE 3 AMINO 1 3 CHLORO 4 FLUORO BENZYL PYRROLIDIN 2 ONE 4 BROMO 1 2 FLUOROPHENYL 3 METHYL 1H PYRAZOL 5 AMINE 4 FLUOROISOINDOLINE 4 METHYL 2 TRIFLUOROMETHYL THIAZOLE 5 CARBOXYLIC ACID 4 fluoropiperidin 3 yl methanamine 1 benzyl 3 ethyl 4 4 difluoropiperidine 1 3 dicarboxylate 3 fluoropiperidin 4 yl methanamine 6 TRIFLUOROMETHYL PYRIDIN 2 YL METHANOL 2 CHLORO 4 2 4 DIFLUORO PHENYL 6 7 DIHYDRO 5H 1 PYRINDINE 3 fluoro tetrahydro 2H pyran 4 ol 8 AMINO 2 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDINE 3 CARBOXYLIC ACID ETHYL ESTER 1 PHENYLMETHYL 4 TRIFLUOROMETHYL TRANS 3 PYRROLIDINECARBOXYLIC ACID

9 4 4 aminopiperidin 1 yl butyl N 2 2 2 trifluoroethyl 9H fluorene 9 carboxamide 2 CHLORO 6 FLUORO N HYDROXY BENZAMIDINE 7 4 FLUORO PHENYL 5 METHYL 4 OXO 4 5 DIHYDRO THIENO 3 4 C PYRIDINE 6 CARBOXYLIC ACID 1 BENZYL 4 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 5 4 FLUORO PHENYL 7 METHYL 8 OXO 7 8 DIHYDRO 1 7 NAPHTHYRIDINE 6 CARBALDEHYDE 3 BROMO 5 FLUORO 2 HYDROXYBENZALDEHYDE 4 4 difluorocyclohexyl methanol 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDIN 3 YL METHANOL 1 BENZYL 3 TRIFLUOROMETHYL PYRROLIDINE 3 CARBOXYLIC ACID 2S 4R 1 tert butyl 2 methyl 4 fluoropyrrolidine 1 2 dicarboxylate 1R 1 4 FLUOROPHENYL PROPYLAMINE 5 FLUORO 3 3 DIMETHYL 2 3 DIHYDRO 1H INDOLE 6 CHLORO 3 TRIFLUOROMETHYL 1 2 4 TRIAZOLO 3 4 A PHTHALAZINE 4 5 6 7 TETRAHYDRO 3 TRIFLUOROMETHYL 1H INDAZOLE 2 CHLORO 6 FLUORO 1 METHYL 1H BENZOIMIDAZOLE 3 FLUOROSALICYLALDEHYDE 3 3 BROMO 4 FLUORO PHENYL 2 2 DIMETHYL CYCLOPROPANECARBOXYLIC ACID 5 FLUORO 3 METHYL BENZOFURAN 4 1 1 2 2 2 PENTAFLUOROETHYL BENZOIC ACID 2 TERT BUTYL 4 FLUOROPHENOL 2 CHLORO 5 FLUORO 1 METHYL 1H BENZO D IMIDAZOLE 2 BROMO 1 2 METHYL 6 TRIFLUOROMETHYL IMIDAZO 1 2 A PYRIDIN 3 YL ETHANONE 2 2 difluoropropane 1 3 diol 4 METHYL 2 4 TRIFLUOROMETHYL PHENYL PYRIDINE 2S 4S N TERT BUTOXYCARBONYL 4 TRIFLUOROMETHYLPROLINE 4 4 CHLORO BENZENESULFONYL 4 2 5 DIFLUORO PHENYL CYCLOHEXYLAMINE 2S 4S methyl 4 fluoropyrrolidine 2 carboxylate hydrochloride 3 TRIFLUOROMETHYL 1H INDAZOLE 6 CHLORO 2 TRIFLUOROMETHYL IMIDAZO 1 2 B PYRIDAZINE 3 SULFONIC ACID AMIDE 5 TRIFLUOROMETHYL THIENO 3 2 B PYRIDINE