1 2 Difluoro 4 methylsulfonyl benzene 2 trifluoromethyl pyridin 3 ol 7 bromo 6 fluorobenzo b thiophene 3 methylcarbamoyl phenylboronic acid 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 1 3 trifluoromethyl phenyl ethanone oxime 2 3 6 Trifluoroacetophenone 5 Fluoro 2 nitrophenol 2 4 Difluoronitrobenzene 3 Chloro 4 fluorobenzotrifluoride 3 5 Dibromo 2 methylpyridine 4 Methoxy 2 2 2 trifluoroacetophenone 3 Amino 4 methylphenol 2 Bromo 6 fluorobenzamide 3 3 chlorophenyl 3 oxopropanenitrile 3 Chloro 4 fluorobenzonitrile 5 Amino 2 bromobenzoic acid 1 BROMO 2 3 6 TRIFLUOROBENZENE 3 4 5 Trifluoropyridine 2 Iodo 3 methylbenzoic acid 1 Boc 2 methoxycarbonylmethylpiperazine 4 Cyanophenylboronic acid 4 Chloro 2 fluorobenzonitrile 2 Methoxy 3 pyridineboronic acid 2 methyl 4 heptafluoroisopropylaniline 3 Oxazolidinesulfonyl fluoride 2 oxo 1 3 trifluoromethyl cyclobutyl ethan 1 ol 6 fluoro 5 methoxypyridine 3 carbaldehyde 5 fluoropyrimidin 2 yl methanol 4R 5R 5 3 5 bis trifluoromethyl phenyl 4 methyl 1 3 oxazolidin 2 one

5 fluoropyrimidine 4 carboxylic acid 5 fluoro 3 methyl 1H pyrrolo 2 3 b pyridine 1S 5S 3 methyl 3 6 diazabicyclo 3 2 0 heptane bis trifluoroacetic acid 3 difluoromethoxy azetidine 5 4 4 5 5 tetraMethyl 1 3 2 dioxaborolan 2 yl picolinaMide 6 bromo 5 chloroisoquinoline 4 isopropoxyphenol 2 methoxy 4 6 dimethylphenylboronic acid 2 boronobenzoic acid 2 fluoro 6 methoxybenzaldehyde 4 chloroquinolin 2 amine 7 chlorothieno 3 2 b pyridine 4 bromo 2 trifluoromethyl benzyl alcohol 2 6 Dibromochlorobenzene 3 fluoro 4 iodophenol 6 bromo 7 fluorobenzo b thiophene 2 5 difluoro 4 methoxyphenylboronic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 3 Difluoromethoxy nitrobenzene 2 Trifluoromethyl phenylboronic acid 4 Fluoro 2 nitroanisole 2 3 5 Trifluoroacetophenone 2 Amino 3 fluorophenol 4 Methoxy 3 methylacetophenone 3 Chloro 2 fluorobenzonitrile 3 2 chlorophenyl 3 oxopropanenitrile 4 Bromo N methoxy N methylbenzamide 4 Amino 3 bromobenzoic acid 5 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 BROMO 2 3 DIFLUOROBENZENE

2 Nitrophenylboronic acid 1 Bromo 3 chloro 2 5 difluorobenzene 2 Bromo 6 chloropyridine 2 Fluoro 5 trifluoromethyl phenylboronic acid 2 Chloro 4 fluorobenzonitrile 4 Chlorophenylboronic acid 2 chloro 5 trifluoromethyl pyridin 4 yl boronic acid 1 2 2 trifluorocyclobutyl methanol 5 fluoropyrimidine 2 carbaldehyde 4 fluoro 2 methyl 1H pyrrolo 2 3 b pyridin 5 ol 6 trifluoromethyl pyridazine 3 carboxylic acid 5 3 5 difluorophenyl methyl 1H indazol 3 amine 1R 5R 3 methyl 3 6 diazabicyclo 3 2 0 heptane bis trifluoroacetic acid 5 bromo 3 phenyl 1H indazole 2 4 chlorophenyl thiazole 5 carboxylic acid 5 bromo 2 isopropoxypyrimidine 2 amino 6 methylpyridin 3 ol 6 bromo 3 methylbenzo b thiophene 3 chloro 2 6 difluorophenylboronic acid 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 bromothieno 3 2 b pyridine 2 amino 6 bromoquinazolin 4 ol 1 Bromo 2 isopropyl benzene 2 nitro 4 trifluoromethyl benzyl alcohol 2 Nitro 4 trifluoromethyl acetophenone 3 Fluoro 2 nitrophenol 3 Trifluoromethyl phenoxyacetic acid 2 6 Difluoro 4 iodonitrobenzene 3 5 Bis trifluoromethyl benzamide 4 Amino 3 5 dimethylphenol

4 Methoxyacetophenone 3 4 bromophenyl 3 oxopropanenitrile 3 Amino 5 bromobenzoic acid 3 5 Bis trifluoromethyl benzenesulfonyl chloride 2 Chloro 6 fluorobenzonitrile 3 4 DIFLUORO 2 METHYLANILINE 3 Boc aminomethyl pyridine 4 boronic acid 2 Amino 5 chloropyrimidine 5 Bromo 2 3 dihydro 1 benzofuran 2 Fluoro 5 hydroxymethyl phenylboronic acid 4 Trifluoromethyl phenylboronic acid 2 2 difluoro 1 methylcyclobutyl methanol 2 bromo 5 fluoro 3 methoxypyridine 4 4 methylpiperazin 1 yl 2 2 2 2 trifluoro N oxan 4 yl acetamido benzoic acid 1 5 fluoropyrimidin 2 yl ethan 1 amine hydrochloride 3 2 2 2 trifluoroethyl 5H 6H 7H 8H 1 2 4 triazolo 4 3 a pyrazine 3 methyl 3 6 diazabicyclo 3 1 1 heptane bis trifluoroacetic acid 3 methyl 3 6 diazabicyclo 3 2 0 heptane bis trifluoroacetic acid 4 5 ForMylthiophen 2 yl 2 Methylphenol 7 bromobenzofuran 5 ol 1 chloro 4 methylisoquinoline 2 4 6 trimethoxyphenylboronic acid 2 3 diaminobenzamide 1 2 bromo 3 fluorophenyl propan 1 one 1 3 isopropylphenyl ethanone 2 amino 7 bromoquinazolin 4 ol 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 amine 4 ethylbiphenyl 4 ylboronic acid 4 chlorobenzo b thiophene 2 nitro 4 trifluoromethyl benzyl bromide