3 Difluoromethyl 1 methyl 1H pyrazole 4 carboxylic acid 1 Bromomethyl 1 trifluoromethyl cyclopentane 3H Spiro 2 benzofuran 1 4 piperidine 2 4 Diaminopyrimidine 5 carbaldehyde 4 5 Dimethylquinolin 2 ol 6 Methoxy oxindole 5 Bromo 2 fluoro 3 pyridineboronic acid 3 Methyl 4 isoxazolecarboxylic acid 3 Bromo 2 fluorobenzoic acid 1 Isopropyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl piperazine 2 Amino 5 chloro 3 nitropyridine 5 Formylthiophene 2 boronic acid 8 Bromoquinoline 4 carboxylic acid 1H imidazol 1 ylmethanol 2 2 amino 5 bromobenzoyl pyridine 2 Bromo 4 fluoro 1 3 thiazole 7 Chloroquinazoline 3 formyl 4 hydroxybenzonitrile 1 4 Dihydro 4 oxoquinoline 3 carboxylic acid 6 Bromopurine 4 Isopropylphenylboronic acid 2 Bromoacetamide 2 Chloro 4 methylbenzoic acid 3 Bromo 4 fluorobenzoic acid 3 Fluoro 2 iodoaniline 5 Carboxyindole 2 carboxylic acid 4 Bromothiophenol 3 5 Difluoro 2 nitrophenol 3 Hydroxypropionic acid 2 Chloro n 2 6 diisopropylphenyl quinolin 8 amine

2S 2 N tert Butoxycarbonyl amino 3 hydroxy 3 methylbutanoic acid 2 Fluoro 4 trifluoromethyl benzaldehyde 3 Bromo 5 chloro 1H indole 1 1 Bis diphenylphosphino ferrocene dichloropalladium II 1 2 Hydroxyethyl 1H pyrrole 2 5 dione 3 bromo 2 chloro 6 fluorotoluene 4 Chloro 2 3 difluoronitrobenzene 4 Chlorodifluoromethoxy aniline 4 chlorobenzofuran 5 Cyanothiophene 2 boronic acid pinacol ester 4 isothiocyanato 1 2 dimethylbenzene 1H imidazol 2 3H one 2 Fluoro 5 methoxybenzonitrile 2 hydroxymethyl phenylboronic acid 5 Amino 2 chlorobenzotrifluoride 2 bromo 5 fluoro 4 methylbenzoic acid 4 Fluoro 3 methoxyphenol 1R endo anti 3 bromo 2 oxobornane 8 sulphonic acid 2 4 Difluoro 3 5 dimethoxybenzoic acid 8 Fluoro 4 chromanone 3 4 Dihydroxybenzonitrile 4 Chloro 2 fluorobenzonitrile 1 2H Phthalazinone 4 Bromo N N 2 6 tetramethylaniline 2 3 Dimethyl 4 Nitropyridine N Oxide 2 4 Dimethyl 6 tert butyl phenol 4 Chloro 2 6 dibromoaniline 1 3 Bis 4 bromophenyl propanone 5 Amino 2 4 6 Triiodo Isophthaloyl Chloride 1 Bromo 2 2 dimethylpropane

3 3 4 difluorophenoxy propanoic acid 4 Hydroxy 3 methoxyphenylboronic acid 3 4 5 Trimethoxybenzoic acid 4 Methoxybenzyl Chloride 4 Fluoro 3 5 dimethylaniline 2 Amino 3 bromopyridine 2 3 Di O acetyl 5 deoxy 5 fuluro D cytidine 3 Chlorosulfonyl benzoic acid 2 Fluoro 6 methylbenzoic acid 2 Bromo 5 fluorophenol 3 Difluoromethoxy benzaldehyde 2 Amino 5 chloro 2 fluorobenzophenone 2 4 Pyridinyl benzaldehyde 3 Amino 5 cyanobenzeneboronic acid hydrochloride 4 Fluorothiophenol 1 Vinylimidazole 2 Fluoro 4 methoxybenzaldehyde 3 4 6 tri O benzyl D glucal 5 Methoxy 2 methylindole 5 Aminobenzimidazolinone 3 Fluoro 4 methoxybenzoic acid 2 Methyl 5 pyrimidinecarboxylic acid 7 Ethoxycarbonylindole 2 carboxylic acid ethyl ester 2 Diphenylphosphino pyridine 3 4 Dihydroxybenzaldehyde 2 Amino 4 fluorophenol 1 2 Dihexadecanoyl sn glycero 3 phosphoethanolamine 6 Chlorobenzo d isoxazol 3 ol 2 Chloromethyl 4 6 dimethoxypyrimidine 4 Bromo 9H carbazole

3 Bromopyridine 3 Boc Aminoazetidine hydrochloride 1 3 Sulphonatopropyl pyridinium 2 2 4 Trimethyl 1 4 2 oxazasilinane 4 2 Ethoxy 2 oxoethoxy benzeneboronic acid 9 Fluorenylmethyl chloroformate 4 Amino 3 iodobenzotrifluoride 2 trifluoromethyl biphenyl 4 carboxylic acid 1 Bromo 3 fluoro 4 Trifluoromethoxy benzene 2 Furylacetic acid 2 Chloroadenine 4 Bromo 3 chlorobenzonitrile 1 Tert butyl 3 methyl 4 oxopiperidine 1 3 dicarboxylate 3 Fluoro 4 hydroxy 5 methoxybenzaldehyde 2 4 Dihydroxybenzonitrile 4 4 Carboxy phenyl piperidine 1 carboxylic acid tert butyl ester 4 4 Di tert butyl 2 2 bipyridine 2 Bromo thiazole 5 carboxylic acid ethyl ester 5 Fluoro 2 hydroxyacetophenone 3 Trifluoromethoxy nitrobenzene 3 Cyclopentylpropanoyl chloride 3 Fluorothiophenol 3 Acetylpyridine 4 4 Methylpiperazino benzoic acid 2 Iodo 4 methylaniline 4 Fluoro 2 methylbenzaldehyde 3 5 Dichlorosalicylic acid 2 4 Bromophenyl 4 6 diphenyl 1 3 5 triazine 5 Bromo 2 hydroxy 3 nitropyridine 4 5 Difluoro 2 nitrobenzoic acid