4 BROMO METHOXYCARBONYL METHYL PIPERIDINE 1 CARBOXYLIC ACID TERT BUTYL ESTER 6 4 Tert butoxycarbonyl piperazin 1 yl 5 methylpyridin 3 yl boronic acid 3 pyridin 4 yl phenyl boronic acid 4 Pyrid 4 yl phenylboronic acid 2 METHYL PIPERIDINE 1 2 DICARBOXYLIC ACID 1 BENZYL ESTER 1 BENZYLSPIRO INDOLE 3 4 PIPERIDIN 2 1H ONE 2 4 chloro 2 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 1 3 AMINOPROPYL PIPERIDIN 2 YL METHANOL 4 Piperidin 1 ylmethyl phenylboronic acid 6 PIPERIDIN 4 YL 1H INDOLE 2 4 Difluoro 5 bromophenylboronic acid piancol ester 3 Formyl 4 hydroxyphenylboronic acid 2 Fluoro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 2 Chloro 6 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 3 Cyano 5 fluorophenylboronic acid pinacol ester 3 3 DIFLUORO PIPERIDIN 1 YLAMINE 2 Methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 4 2 4 DIMETHYL PHENYL PIPERIDIN 4 OL 1 BOC 4 2 4 DIFLUOROPHENYL 4 HYDROXYPIPERIDINE 4 Hydroxymethyl 3 methoxyphenylboronic acid pinacol ester 2 Bromo 5 methylphenylboronic acid 2 4 PIPERIDINEDICARBOXYLIC ACID 1 3 ACETYLTHIO 1 OXOPROPYL CIS 4 Fluoro 3 methoxycarbonylphenylboronic acid pinacol ester 2 5 PIPERIDINEDICARBOXYLIC ACID 1 3 MERCAPTO 1 OXOPROPYL CIS 3 Hydroxy 5 methylphenylboronic acid pinacol ester 4 Fluoro 3 hydroxyphenylboronic acid pinacol ester 1 PHENETHYL 4 PHENYL 4 PIPERIDINOL 4 N N Diethylaminomethyl phenylboronic acid pinacol ester 4 HYDROXY PIPERIDINE 1 2 DICARBOXYLIC ACID 1 TERT BUTYL ESTER 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl aniline

3 Fluorophenylboronic acid pinacol ester 1S 2R 5R 2 HYDROXYMETHYL 3 AZA BICYCLO 3 1 0 HEXANE 3 CARBOXYLIC ACID TERT BUTYL ESTER 3 Chloro 2 methylthiopyridine 5 boronic acid 1H INDAZOLE 6 FLUORO 3 1 METHYL 4 PIPERIDINYL 2 Amino 5 trifluoromethyl phenylboronic acid pinacol ester 1H INDAZOLE 6 FLUORO 1 2 FLUOROPHENYL 3 1 METHYL 4 PIPERIDINYL 4 Methoxy 3 1 methylethyl phenylboronic acid 4 Hydroxy 3 isopropylphenylboronic acid pinacol ester 1H INDAZOLE 6 CHLORO 3 1 METHYL 4 PIPERIDINYL 2 Methyl 4 methoxymethoxy phenylboronic acid pinacol ester 2 Isoproxy 3 methylpyridine 5 boronic acid pinacol ester 4 4 BIS 4 METHOXYPHENYL PIPERIDINE 3 Methylindazole 6 boronic acid pinacol ester 5 Methyl 1H indazole 4 boronic acid pinacol ester 3 Cyclopropyl 2 6 difluorophenylboronic acid 2 Amino 5 chlorophenyl boronic acid pinacol ester 4 Cyano 3 fluorophenylboronic acid pinacol ester 2 Fluoro 4 methoxycarbonyl phenylboronic acid pinacol ester 2 8 tert butoxycarbonyl 8 aza bicyclo 3 2 1 octan 3 yl acetic acid 1 tert butoxycarbonyl 1 2 3 6 tetrahydropyridine 4 carboxylic acid 4 Ethoxy 2 3 dimethylphenylboronic acid 2 Chloro 5 formylphenylboronic acid pinacol ester 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 dioxolan 2 yl pyridine 4 Biphenyl 4 yl piperidine 4 Bromo 2 5 bifluorophenylboronic acid pinacol ester 2 Chloro 6 hydroxyphenylboronic acid pinacol ester 2 6 Difluoro 3 methylthio phenylboronic acid 1 tert butyl 4 ethyl 3 hydroxy 4 methylpiperidine 1 4 dicarboxylate 2 6 Dimethyl 4 fluorophenylboronic acid 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 2 3 6 tetrahydropyridine

3 bromo 1 methyl 1 2 5 6 tetrahydropyridine 2 5 Difluoro 4 methylsulfanyl phenylboronic acid 2 3 Dimethyl 4 methoxyphenylboronic acid 4 Cyano 3 methylphenylboronic acid pinacol ester 1 benzyl 3 methyl 5 tert butoxycarbonylamino piperidine 1 3 dicarboxylate 4 Bromo 2 methylphenyboronic acid 3 Bromophenylboronic acid N butyldiethanolamine ester 4 Fluoro 1H indazol 6 yl boronic acid 3 bromo 1 propyl 1 2 5 6 tetrahydropyridine 2 8 DIAZASPIRO 5 5 UNDECAN 1 ONE HYDROCHLORIDE 3 Bromo 5 formylphenylboronic acid 4 Bromo 2 isopropylphenylboronic acid 4 Methoxy 2 trifluoromethoxy phenylboronic acid 4 4 bromophenyl piperidine 4 carbonitrile 3 Bromo 4 chlorophenylboronic acid 4 5 Amino 1H pyrazol 3 yl piperidine 1 carboxylic acid tert butyl ester 2 Trifluoromethylpyridine 5 boronic acid pinacol ester 1 TERT BUTOXYCARBONYL 4 PHENYLPIPERIDINE 4 CARBOXYLIC ACID 2 4 Difluoro 3 iodophenylboronic acid 2 Fluoro 4 formyl 6 methoxyphenylboronic acid 6 Isobutoxy 2 methylpyridine 3 boronic acid 3 hydroxy 4 5 6 7 tetrahydro 2H pyrazolo 3 4 c pyridine 5 carboxylic acid hydrochloride 7 Chloro 1H indazole 4 boronic acid 2 Bromo 4 methylphenylboronic acid 1 benzyl 4 3 phenylpropyl 1 2 3 6 tetrahydropyridine 6 Isopropoxynaphthalene 2 boronic acid 1 tert butyl 2 ethyl 3 oxopiperidine 1 2 dicarboxylate 3 5 Dichloro 2 6 difluorophenylboronic acid 3 3 difluoropiperidin 4 ol 6 Isopropoxy 2 methylpyridine 3 boronic acid

1 benzyl 3 1 benzyl 2 oxo piperidin 4 ylidene piperidine 2 4 dione 2 3 Dimethoxypyridine 5 boronic acid 2 Fluoro 3 isopropoxypyridine 5 boronic acid 5 Chloro 2 methylsulfanyl pyridine 3 boronic acid 5 Fluoro 2 morpholin 4 ylmethyl phenyl boronic acid 1 tert butyl 3 methyl 5 oxopiperidine 1 3 dicarboxylate 4 Bromo 2 Chloro 5 trifluoromethyl phenylboronic acid 3 Bromo 5 methylsulfanyl phenylboronic acid 2 Ethoxy 4 methylphenylboronic acid 4 Bromo 2 fluoro 5 trifluoromethyl phenylboronic acid 2 Chloro 3 5 dimethylphenylboronic acid 4 Bromo 5 chloro 2 methylphenylboronic acid 1 HYDROXYMETHYL 3 OXO 2 AZABICYCLO 2 2 2 OCTANE 2 6 Dimethoxybiphenyl 2 ylboronic acid 1 benzyl 3 hydroxymethyl piperidin 4 ol 4 Amino 3 5 dimethylphenylboronic acid pinacol ester 4 Chloro 3 isopropoxyphenylboronic acid 8 benzyl 3 hydroxyimino 8 AZA BICYCLO 3 2 1 OCTANE 2 Fluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid methyl ester 2 Amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 Tert butylcarbonylamino phenylboronic acid pinacol ester 8 benzyl 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octane 2 Phenoxypyridine 5 boronic acid 5 tert butyl 3a ethyl hexahydro 1H pyrrolo 3 2 c pyridine 3a 5 6H dicarboxylate 2 Bromo 4 chlorophenylboronic acid 4 4 bromophenyl piperidine 4 carbonitrile hydrochloride 6 Fluoro 2 methylsulfanyl phenylboronic acid 5 Fluoro 2 morpholinomethyl phenylboronic acid hydrochloride 1 methyl 4 phenylpiperidine 2 Methoxy 4 methylthio pyridine 5 boronic acid pinacol ester