2 hydroxy 4 trifluoromethyl phenyl boronic acid 4 Maleimidomethyl cyclohexanecarboxylic acid 2 hydroxy 5 trifluoromethyl phenyl boronic acid 2 5 methoxynaphthalen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 3 Chlorophenyl 1 2 3 4 tetrahydro 6 methyl 2 oxo 5 pyrimidinecarboxylic acid 4 2 Chlorophenyl 1 4 5 6 tetrahydro 2 methyl 6 oxo 3 pyridinecarboxylic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoindolin 1 one 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl indoline 1 Boc piperidine 4 carboxylic acid ethyl ester 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indole 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 6 Chlorobenzo d isoxazol 3 ol 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 2 3 dimethyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyrimidine 2 Chloro 4 methoxyphenylacetonitrile 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 3 Amino 5 hydroxypyrazole 7 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 7 methylimidazo 1 2 a pyridin 6 yl boronic acid 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 5 Amino 1 2 4 thiadiazole 7 Ethyl 10 hydroxycamptothecin 1H indazol 5 yl boronic acid

1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 1H indazol 4 yl boronic acid 2 4 6 Trichloropyridine 5 Methyl 3 2H pyridazinone 1H indazol 7 yl boronic acid 3 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Nitrobenzyl chloroformate 1 methyl 1H indazol 7 yl boronic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 3 tert butylbenzenesulfonyl chloride 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methanol 4 Phenoxybenzoic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl methanol 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl ethanone 4 Ethoxybenzoyl chloride 3 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 Fluoronaphthalene 1 4 Cyclohexanedicarboxylic acid 3 ethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 Chlorobenzaldehyde 4 4 5 5 tetramethyl 2 3 methylbenzofuran 6 yl 1 3 2 dioxaborolane 2 iodo 4 methoxyaniline 7 methylbenzofuran 5 yl boronic acid 2 benzo b thiophen 3 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Bromo 4 butanolide 2 7 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Methyl 4 methylthio phenol 3 hydroxymethyl thiophen 2 yl boronic acid 3 bromothiophen 2 yl boronic acid 6 Fluoronicotinic acid methyl ester

6 Bromopyridine 2 carboxylic acid ethyl ester 3 methylthiophen 2 yl boronic acid 2 Chloro 6 iodoaniline 4 bromo 5 methylthiophen 2 yl boronic acid 3 chloro 2 iodoaniline 2 5 chlorothiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 4 Methylpiperazino benzoic acid 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 3 Aminopropylphosphate 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 Bromo 3 methoxypropanol 1 Chloro 3 isothiocyanato 2 methylbenzene 1 4 chlorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl morpholine 2 Chloro 5 fluoro 4 methylpyridine 5 Amino 4 chloro 2 methylphenol 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 Bromo 3 fluoro 2 methoxypyridine 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 4 fluorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 Benzyloxyphenol 1 3 chlorophenyl 1H pyrazol 4 yl boronic acid 1 4 fluorophenyl 1H pyrazol 4 yl boronic acid 2 4 Diaminopyrimidine 5 carbaldehyde 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl propan 2 ol 2 trifluoromethyl biphenyl 4 carboxylic acid 5 4 trifluoromethylphenyl 1H pyrazole 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 carbonitrile

4 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 6 Methyl 5 nitropyridin 2 ol 3 Amino 2 6 dichloropyridine 3 5 Dichloro 2 Bromopyridine 6 chloro 2 fluoropyridin 3 yl boronic acid 1 hydroxymethyl cyclopropaneacetonitrile 3 Amino 2 Hydroxyacetophenone 2 ethoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 Bromo 2 methylbenzaldehyde 2 isopropoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 bromobenzaldehyde 5 fluoro 2 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Mercapto Thiadiazole 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 ol 3 Bromothiophene 2 carboxylic acid 3 chloro 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 nitro 4 trifluoromethyl aniline 2 3 difluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Bromo 2 3 difluorobenzaldehyde 2 chloro 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Trifluoromethoxy benzylsulphonyl chloride 1 1 Dimethoxy acetone 2 5 Dimercapto 1 3 4 thiadiazole 2 3 dichloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Methyl 2 propanesulfinamide 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 methoxy 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 Nitroindole 2 carboxylic acid 5 Chloro 2 hydroxy 3 picoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile