4 Phenylindolin 2 one 1 Phenyl 1H benzoimidazole 1 3 4 Oxadiazole 2 carboxylic acid 5 methyl ethyl ester 2 Chlorothieno 2 3 d pyrimidin 4 yl morpholine 5 Bromo 4 chloro 2 methylpyridine 3 Iodo pyridin 4 yl carbamic acid tert butyl ester 2 Bromo 3 hydroxy 5 picoline 1 6 Bromo 1H indol 3 yl ethanone 4 6 Pyrimidinedicarbonitrile 3 Bromo 5 bromomethyl 1 2 4 oxadiazole 3 Chloro 2 Methylquinoline 4 Chloro 8 cyanoquinoline 3 carboxylic acid ethyl este 5 Butyl 2 mercapto 6 methylpyrimidin 4 ol 4 Chloro 5 8 dihydro 6H pyrido 3 4 d pyrimidine 7 carboxylic acid tert butyl ester 2 Chloro 4 morpholin 4 yl thieno 2 3 d pyrimidine 6 carboxaldehyde 5H Pyrrolo 2 3 b pyrazine 7 carboxaldehyde 2 Amino 1H pyrrole 3 carboxylic acid ethyl ester 6 Amino pyrazolo 1 5 a pyrimidine 3 carboxylic acid ethyl ester 2 Chloro 5 6 7 8 tetrahydro pyrido 3 4 d pyrimidine 5 4 Bromophenyl 1H pyrazol 3 amine 5 2 methylphenyl 1H pyrazole 3 amine 4 methyl 4H 1 2 4 triazol 3 ylamine 3 4 Methoxy phenyl 1H indazole 3 Pyridinemethanesulfonamide 5 3 Chlorophenyl 1H pyrazol 3 amine 1H Benzimidazole 6 carbonitrile 7 Aminobenzo d oxazol 2 3H one 3 Amino 5 3 iodophenyl 1H pyrazole 3 phenylpyrazin 2 ol 3 Amino 5 4 iodophenyl 1H pyrazole

4 Methylisoxazole 3 carboxylic acid 3 Chlorotetrahydrofuran 4 6 Pyrimidinedicarboxylic acid 3 Chloro tetrahydropyran 9 Benzyl 3 9 diaza spiro 5 5 undecane 2 4dione 2 Bromo 6 chloro 4 nitropyridine 4 Benzyl 2 chloromethyl morpholine 1 Boc 3 methylene pyrrolidine 1 Benzhydryl 3 chloroazetidine 6 Bromo 1 2 3 4 tetrahydro 1 1 4 4 tetramethylnaphthalene 7 Azabicyclo 4 2 0 octan 8 one 4 Bromo 2 3 dimethylanisole 2 Methyl 2H 1 4 Benzoxazin 3 4H one 5 Methyl 4 phenyl 3 4 dihydro 2H pyrrole 2 Bromo N tert butoxycarbonyl aniline 1 3 5 tris chloromethyl 2 4 dimethylbenzene 3 Iodomethyl oxetane 6 Chloroisoindolin 1 one 5 Bromo 2 3H benzofuranone 2 4 Dibromofuran 7 Bromo 3 methoxyquinoline 3 Bromo 7 chloroquinoline 1 4 Methoxy benzyl piperidine 2 4 dione 8 Bromochroman 3 one 8 Oxabicyclo 3 2 1 octan 3 one 1R Dimenthyl succinate 4 Boc 3 2 Oxo ethyl morpholine 4 Morpholinocyclohexanone 2 Azabicyclo 2 2 2 octane 2 6 dicarboxylic acid 2 1 1 dimethylethyl 6 methyl ester 1R 4S 6R rel 4 4 Chlorobenzenesulfonyl benzaldehyde

7 Bromo 2 3 dihydro 1 8 naphthyridin 4 1H one 5 Nitroisatoic anhydride 2 Cyclohepten 1 one 8 Methyl 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 6 carbaldehyde 1 4 1 3 Dioxolan 2 yl phenyl ethanone 3 Chromanone 1 Acetamido acetone 1 Boc 3 5 dioxopyrrolidine 1 2H Naphthalenone 3 4 dihydro 7 phenylmethyl 3 Hydroxy 5 methoxybenzaldehyde 9H Fluoren 9 yl methyl 2 oxoethylcarbamate 4 Bromo 3 hydroxybenzaldehyde 5 Bromo 3 methoxybenzaldehyde 7 Methoxy 4 trifluoromethyl coumarin 5 Boc Amino pyridine 3 boronic acid pinacol ester 4 Boronicacid biphenyl 4 carboxylicacid methyl ester 3 Pyrrolylboronic acid 3 tert Butoxycarbonyl amino methyl pyridin 4 yl boronic acid 1 1H indol 3 yl 2 2 phenylvinyl sulfonyl 1 2 dihydroisoquinoline 1H 1 2 4 Triazole 3 5 diamine N3 4 aminosulfonyl phenyl 1 3 5 dimethyl 2 thienyl carboyl 9CI 1 3 Chlorobenzyl 6 4 isopropoxyphenyl 3 pentanoyl amino indole 2 carboxylic acid 3 4 Chlorobenzoylamino 1 3 chlorobenzyl 6 4 isopropoxyphenyl indole 2 carboxylic acid 1H 1 2 4 Triazole 3 5 diamine N3 4 2 dimethylamino ethyl mino sulfonyl phenyl 1 3 5 dimethyl 2 thienyl carbonyl 9CI 3 Cyclohexyl L alanine hydrate 2 4 2 4 Dioxo 5 thiazolidinyl methyl phenoxy acetic acid 2S 3R 2 Methyl 3 morpholinecarboxylic acid 1S 3aR 6aS Hexahydro cyclopenta c pyrrole 1 2 dicarboxylic acid 2 tert butyl ester 4S 1 Boc 4 Methyl L proline 1 Amino cyclopentanecarboxylic acid ethyl ester hydrochloride 1S 3aR 6aS Octahydro cyclopenta c pyrrole 1 carboxylic acid hydrochloride

3 N Boc 3 methylbutane 1 3 diamine HCl 3 Pyridin 4 yl 3 9 diazaspiro 5 5 undecane 6aR tert Butyl 6a trifluoromethyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 6aR tert Butyl 6a phenyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 3aR tert Butyl 3a ethyl hexahydropyrrolo 3 4 c pyrrole 2 3a 1H dicarboxylate 2 Amino 2 2 pyridyl ethanol 4 Bromophenyl piperidin 4 yl methanone 4 4 Acetylpiperazin 1 yl 3 trifluoromethyl aniline 1 2 3 4 Tetrahydroisoquinolin 4 ol 3 Dimethylamino pyrrolidine 3R 4R 4 4 Fluorophenyl 3 piperidinemethanol 2 Methoxy 1 propanamine 1 Cbz 3 aminomethylazetidine 3 8 Diazabicyclo 3 2 1 octane 2S 5S 2 5 Dimethylmorpholine 4 3 nitrophenyl piperidine 1 Amino 3 buten 2 ol 1S 2R 2 Amino cyclohexanol HCl 1S 2R 2 Amino cyclohexanol 1 6 7 dimethoxy 2H benzo d 1 3 dioxolan 5 yl prop 2 ylamine 1S 3R 3 Aminocyclopentanol 1 Cyclopropylethanamine 1S 3S 3 Aminocyclopentanol 1R 3R 3 Aminocyclopentanol 2 piperidin 2 yl ethanamine 8 Oxa 2 azaspiro 4 5 decane 7 Oxa 2 aza spiro 4 5 decane 6 Oxa 2 aza spiro 4 5 decane 1 Oxa 7 azaspiro 4 5 decane 2 Ethenylmorpholine