2 1H Benzo d 1 2 3 triazol 1 yl 1 1 3 3 tetramethyluronium tetrafluoroborate 2 Chloro N N dimethylethanamine 1 Hydroxycyclohexyl phenyl methanone 7 Chloro 1 cyclopropyl 6 fluoro 4 oxo 1 4 dihydro 1 8 naphthyridine 3 carboxylic acid 2 4 Benzylpiperazin 1 yl benzaldehyde 2 Trifluoromethyl biphenyl 3 carboxylic acid 2 Acetylphenanthrene 4 Trifluoromethyl biphenyl 3 carbaldehyde 2 Trifluoromethyl biphenyl 4 carbaldehyde 4 Pyridin 3 yl benzoic acid 1 Benzylpiperidine 2 carboxylic acid 4 Piperidin 1 yl benzaldehyde 4 Pyrimidin 5 yl benzaldehyde 4 Bromo 6 7 dimethoxyquinoline 2 Methyl 1 4 nitrobenzyl 1H imidazole 2 Benzofuranylglyoxal hydrate 1 Bromomethyl 2 3 dimethylbenzene 3 Aminobenzeneboronic acid hemisulfate salt 2 Isopropyl 5 methyl 4 nitrosophenol 1 5 Bromopyrimidin 2 yl piperidine 4 carboxylic acid 4 Piperidinopiperidine 7 Hydroxy 4 trifluoromethyl coumarin 2 Hydroxy 4 trifluoromethyl quinoline 2 Amino 5 bromo 4 hydroxy 6 phenylpyrimidine 3 Bromomethyl phenyl methanol 3 Methoxy 4 methyl aniline 1 3 Chloro 2 hydroxyphenyl ethan 1 one 2 Bromophenylacetonitrile 1 bromo 2 fluoro 4 methoxybenzene 5 Fluorosalicylic acid

2 Amino 5 fluorobenzotrifluoride 3 4 Difluorophenyl hydrazine hydrochloride 2 Methoxythiazole 3 5 Dichloropyridin 4 ol 2 Chloro 5 methylthiazole 2 Bromo 5 methyl 1 3 4 thiadiazole 6 Fluoro 3 4 piperidinyl 1 2 benzisoxazole 5 Bromo 4 trifluoromethyl thiazol 2 amine 4 Bromo 3 fluoropyridine hydrochloride 3 Methoxy 4 methylbenzaldehyde 2 Methyl 3 Nitroaniline 2 Hydroxyisonicotinic acid 4 Methyl indole 2 Chlorobenzothiazole 6 carbonitrile 4 2 Bromoacetyl benzoic acid 4 Methoxy N methyl 2 nitrobenzenamine 4 Isopropylphenylboronic acid 2 Amino 2 4 bromophenyl acetic acid 4 Hydroxy 3 trifluoromethyl benzoic acid 2 Chloro 6 trifluoromethoxy benzo d thiazole 4 5 6 7 Tetrahydrothieno 3 2 c pyridine hydrochloride 3 5 Dibromo 2 6 dimethylpyridine 4 Methoxy 2 nitrobenzenesulfonyl chloride 4 Methoxythiophene 3 carboxylic acid 3 Aminohomopiperidine 4 Chloro 2 fluoro 6 iodoaniline 5 Bromo oxazole 1 Quinolin 2 yl methyl piperidin 4 one 4 Trifluoromethoxy pyridin 2 amine 4 Morpholin 4 yl phenylamine

5 Bromopyrimidin 2 ol 4 Chloro 6 hydrazinopyrimidine 2 2 2 2 Trifluoroethoxy pyridine 5 carbonitrile 5 6 7 8 tetrahydro 1 8 naphthyridine 2 carbaldehyde 6 tert Butylnicotinonitrile 8 Ethyl quinoline 2 Phenyloxazole 5 carbaldehyde 4 Methoxy 2 methylpyrimidine 8 Chloro 10 11 dihydro 4 aza 5H dibenzo a d cycloheptan 5 one 5 Nitro 3 isothiazolecarboxylic acid 1 3 Acetyloxy 5 bromo 1H indol 1 yl ethanone 2 Trifluoromethyl 5 6 7 8 tetrahydroimidazo 1 2 a pyrazine 5 Benzyloxy 2 chloromethyl pyridine 5 Chloro 1H indazole 3 carbonitrile 5 Bromo 6 chloropyridine 3 sulfonamide 3 Pyrazolidinone 4 Hydroxy 7 methoxy 2H quinolin 2 one 6 7 Dimethyl 1H indole 2 3 dione 4 Benzothiazolol 5 Chloro 1H Pyrrolo 2 3 C Pyridin 2 3H one 4 Phenylindolin 2 one 1 Phenyl 1H benzoimidazole 1 3 4 Oxadiazole 2 carboxylic acid 5 methyl ethyl ester 2 Bromo 3 hydroxy 5 picoline 5 Bromo 4 chloro 2 methylpyridine 3 Chloro 2 Methylquinoline 3 Bromo 5 bromomethyl 1 2 4 oxadiazole 4 6 Pyrimidinedicarbonitrile 1 6 Bromo 1H indol 3 yl ethanone 2 Chlorothieno 2 3 d pyrimidin 4 yl morpholine

2 Chloro 5 6 7 8 tetrahydro pyrido 3 4 d pyrimidine 2 Chloro 4 morpholin 4 yl thieno 2 3 d pyrimidine 6 carboxaldehyde 5H Pyrrolo 2 3 b pyrazine 7 carboxaldehyde 4 Chloro 5 8 dihydro 6H pyrido 3 4 d pyrimidine 7 carboxylic acid tert butyl ester 5 Butyl 2 mercapto 6 methylpyrimidin 4 ol 4 Chloro 8 cyanoquinoline 3 carboxylic acid ethyl este 3 Iodo pyridin 4 yl carbamic acid tert butyl ester 2 Amino 1H pyrrole 3 carboxylic acid ethyl ester 6 Amino pyrazolo 1 5 a pyrimidine 3 carboxylic acid ethyl ester 3 Pyridinemethanesulfonamide 3 4 Methoxy phenyl 1H indazole 4 methyl 4H 1 2 4 triazol 3 ylamine 5 2 methylphenyl 1H pyrazole 3 amine 5 4 Bromophenyl 1H pyrazol 3 amine 5 3 Chlorophenyl 1H pyrazol 3 amine 3 Amino 5 4 iodophenyl 1H pyrazole 3 Amino 5 3 iodophenyl 1H pyrazole 1H Benzimidazole 6 carbonitrile 7 Aminobenzo d oxazol 2 3H one 3 phenylpyrazin 2 ol 4 Methylisoxazole 3 carboxylic acid 4 6 Pyrimidinedicarboxylic acid 3 Chlorotetrahydrofuran 9 Benzyl 3 9 diaza spiro 5 5 undecane 2 4dione 3 Chloro tetrahydropyran 4 Benzyl 2 chloromethyl morpholine 2 Bromo 6 chloro 4 nitropyridine 1 Boc 3 methylene pyrrolidine 1 Benzhydryl 3 chloroazetidine 7 Azabicyclo 4 2 0 octan 8 one