2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 7 CHLORO 3 PHENYL PYRAZOLO 1 5 A PYRIMIDINE 5 7 DICHLORO 2 METHYLPYRAZOLO 1 5 A PYRIMIDINE 2 HYDROXYMETHYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 6 ACETYL 7 METHYLPYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE 2 7 DIMETHYL 3 PHENYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 6 METHYLPYRAZOLO 1 5 A PYRIMIDIN 7 OL 3 THIOPHEN 2 YL 6 3 4 5 TRIMETHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 3 3 THIOPHEN 2 YL PYRAZOLO 1 5 A PYRIMIDIN 6 YL PROPAN 1 OL 2 3 METHOXY PHENYL 6 4 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 2 2 METHOXY PHENYL 6 4 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 3 2 2 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDIN 6 YL PROPAN 1 OL 7 HYDROXY 5 METHYLPYRAZOLO 1 5 A PYRIMIDINE 3 CARBONITRILE 6 4 METHOXY PHENYL 2 PHENYL PYRAZOLO 1 5 A PYRIMIDINE 2 3 BROMO PHENYL 6 4 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 3 PHENYL 6 3 4 5 TRIMETHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDINE 4 6 4 METHOXY PHENYL PYRAZOLO 1 5 A PYRIMIDIN 2 YL PHENYL DIMETHYL AMINE 5 7 DIMETHYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXYLIC ACID 3 3 CHLOROPHENYL 2 7 DIMETHYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 2 2 METHYLPYRAZOLO 1 5 A PYRIMIDIN 6 YL ACETIC ACID 3 METHYLPYRAZOLO 1 5 A PYRIMIDINE 5 7 DIOL 3 4 METHOXYPHENYL 2 7 DIMETHYL PYRAZOLO 1 5 A PYRIMIDINE 6 CARBOXYLIC ACID 2 METHYL PYRAZOLO 1 5 A PYRIMIDINE 3 CARBOXYLIC ACID 2 methylmorpholin 3 one 6 methylmorpholin 3 one 5 6 DIHYDRO 4 METHOXY 2H PYRAN 5 S 5 methyl 2 phenylthio dihydrofuran 2 3H one 7 methoxy 7 oxoheptanoic acid 1 2 4 dimethylphenyl 3 phenyl 1H pyrazole 5 4H one 1 3 tert butyl 5 iodo 4 methoxyphenyl pyrimidine 2 4 1H 3H dione

2 3 4 dimethoxyphenyl 3 hydroxy 8 methyl 4H chromen 4 one 2 3 4 dimethoxyphenyl 3 hydroxy 7 methoxyquinolin 4 1H one 3 3 4 dimethoxyphenyl 1 2 hydroxy 3 methylphenyl prop 2 en 1 one 4 4 methoxyquinolin 2 yl benzene 1 2 diol 2 3 4 dihydroxyphenyl 6 ethyl 3 hydroxy 4H chromen 4 one 4 4 1E 1 E 2 2 1 phenyl 1H pyrazole 3 5 diyl bis ethene 2 1 diyl diphenol 2 3 4 dimethoxyphenyl 3 hydroxyquinolin 4 2H one 1 2 4 dimethylphenyl 3 3 methoxyphenyl 1H pyrazol 5 4H one 2S 4R 1 benzyl 2 Methyl 4 hydroxypyrrolidine 1 2 dicarboxylate 3 Ethynyl 5 trifluoromethyl pyridine 2 2 2 Trifluoro 1 3 methoxypyridin 4 yl ethanone 4 1 Methylpiperidin 4 yl oxy aniline 3 TRIFLUOROMETHOXY PIPERIDINE 3 Fluoro 2 iodoaniline 2R 4S 1 benzyl 2 Methyl 4 hydroxypyrrolidine 1 2 dicarboxylate 4 ethoxycarbonyl methyl cyclohex 1 enyl trifluoromethanesulfonate 3 3 difluoro 1 methylpiperidin 4 ol hydrochloride 1 benzyl 3 3 difluoropiperidine 4 4 diol 2 1 tert butoxycarbonyl piperidin 4 yl 2 methylpropanoic acid 2 4 6 fluoroquinolin 4 yl cyclohexyl acetic acid 2 trifluoromethyl 4 methylsulfonyl phenyl methanol 5 5 5 trifluoro 4 4 dihydroxypentanoic acid 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 3 carboxamide 3 3 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 4 carboxamide 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl piperidine 2 carboxamide 2 3 Aminophenyl 2 methylpropanenitrile 5 Bromo 2 methylpyridin 3 ol 5 5 difluoro N S 3 1S 3R 5R 3 3 isopropyl 5 methyl 4H 1 2 4 triazol 4 yl 8 aza bicyclo 3 2 1 octan 8 yl 1 phenylpropyl 1 methylpiperidine 2 carboxamide 2 Chloromethyl nicotinonitrile 4 Morpholin 4 yl benzene 1 carboximidamide hydrochloride

2 3 Fluoro 5 methoxyphenyl acetonitrile 4 Bromo 1 bromomethyl 2 chlorobenzene 3 2H 1 2 3 Trizazol 2 yl aniline 4 Bromobutan 1 amine hydrobromide 3 Amino 6 bromopyrazine 2 carbaldehyde 4 Hydroxy 4 trifluoromethyl cyclohexanecarboxylic acid 4 tert Butyl cyclohex 1 ene 1 2 Bromo 5 chlorophenyl ethanone 4 6 Dichloro 2 methylthio 5 nitropyrimidine 5 Bromo 2 cyano 4 methylpyridine 3 3 Nitrophenoxy azetidine hydrochloride 4 Chloro 8 fluoro 2 trifluoromethyl quinazoline 1H Pyrrol 2 yl methanamine hydrochloride 1 1 Diphenyl 4 piperidin 1 yl butan 1 ol hydrochloride 3 Amino 4 nitrobenzonitrile 4 Dimethylamino benzamide 4R 5R 3 tert Butyl 4 methyl 2 2 5 trimethyloxazolidine 3 4 dicarboxylate 6 7 Dihydro 5H cyclopenta b pyridin 4 amine 4 4 Ethylpiperazin 1 ylmethyl benzoic acid 5 Pyrimidinecarboxylic acid 4 6 dichloro ethyl ester 2 Bromomethyl 4 chloro benzoic acid methyl ester 2 Chloro 7 nitroquinoxaline 5 Bromo 2 3 dimethoxypyrazine 3 Bromo 5 prop 1 en 2 yl pyridine 3 Bromo 5 trifluoromethyl phenol 4 Oxopiperidine 3 carbonitrile hydrochloride 3 4 Dihydropyrrolo 1 2 a pyrazin 1 2H one 3 Amino 3 methylbutyric acid hydrochloride 6 Bromospiro chroman 2 4 piperidin 4 one 1 Phenoxycarbonyl pyrrolidine 2 carboxylic acid

3 Aminocyclopentanol hydrochloride 4 Amino 3 fluorobenzoic acid allyl ester 6 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl indolin 2 one 3 Ethoxypyridazine 2 Amino 4 bromo 3 nitropyridine 4 4 Dimethylpyrrolidine 3 carboxylic acid hydrochloride 5 Fluoro 2 pyrimidineacetic acid 2 Hydroxycyclopent 2 en 1 one 4 Cyano 3 fluorobiphenyl 4 carboxylic acid 4 Methyl 1H indazol 5 yl boronic acid 3 Amino 3 4 chlorophenyl 1 propanol 1 Cyclobutyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 Phenyl 1 p tolylsulphonyl piperidine 4 carbonitrile 3 4 Dibromo 5 fluoropyridine 2 Bromo 4 trifluoromethyl thiazole 5 Bromoquinoline 2 carboxylic acid 4 Pyrimidinol 5 fluoro 2 methyl 7CI 8CI 5 Methyl 2H isoquinoline 1 one 8 bromoquinoline 5 carboxylic acid 1 Boc 4 5 methyl 1 3 4 oxadiazol 2 yl piperidine 4 Bromo 1H pyrrole 2 carbaldehyde 6 Chloronicotinimidamide hydrochloride 3 Fluoro 5 hydroxybenzoic acid 4 Ethynylphenylacetonitrile 4 Diphenylmethoxypiperidine hydrochloride 2 Chloro 5 iodopyrimidin 4 amine 3 Bromo 4 trifluoromethyl benzoic acid 3 Bromo 2 methyl phenol 4 Bromopyrimidin 2 yl cyclopentylamine 3 fluoro 2 nitrobenzonitrile