4 Piperidin 1 ylmethyl phenylboronic acid 2 4 chloro 2 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Formyl 4 hydroxyphenylboronic acid 3 Hydroxy 5 methylphenylboronic acid pinacol ester 4 Fluoro 3 hydroxyphenylboronic acid pinacol ester 4 Fluoro 3 methoxycarbonylphenylboronic acid pinacol ester 2 Bromo 5 methylphenylboronic acid 4 Hydroxymethyl 3 methoxyphenylboronic acid pinacol ester 2 Methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 2 Chloro 6 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 3 Cyano 5 fluorophenylboronic acid pinacol ester 2 Fluoro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl aniline 4 N N Diethylaminomethyl phenylboronic acid pinacol ester 3 Fluorophenylboronic acid pinacol ester 3 Chloro 2 methylthiopyridine 5 boronic acid 2 Amino 5 trifluoromethyl phenylboronic acid pinacol ester 4 Methoxy 3 1 methylethyl phenylboronic acid 4 Hydroxy 3 isopropylphenylboronic acid pinacol ester 2 Methyl 4 methoxymethoxy phenylboronic acid pinacol ester 2 Isoproxy 3 methylpyridine 5 boronic acid pinacol ester 3 Methylindazole 6 boronic acid pinacol ester 2 Chloro 6 hydroxyphenylboronic acid pinacol ester 5 Methyl 1H indazole 4 boronic acid pinacol ester 3 Cyclopropyl 2 6 difluorophenylboronic acid 2 Amino 5 chlorophenyl boronic acid pinacol ester 4 Cyano 3 fluorophenylboronic acid pinacol ester 2 Fluoro 4 methoxycarbonyl phenylboronic acid pinacol ester 4 Ethoxy 2 3 dimethylphenylboronic acid 2 6 Difluoro 3 methylthio phenylboronic acid

4 Bromo 2 methylphenyboronic acid 4 Cyano 3 methylphenylboronic acid pinacol ester 2 6 Dimethyl 4 fluorophenylboronic acid 2 5 Difluoro 4 methylsulfanyl phenylboronic acid 2 3 Dimethyl 4 methoxyphenylboronic acid 2 Chloro 5 formylphenylboronic acid pinacol ester 5 chloro 2 fluoro 3 4 4 5 5 tetramethyl 1 3 dioxolan 2 yl pyridine 4 Bromo 2 5 bifluorophenylboronic acid pinacol ester 4 Fluoro 1H indazol 6 yl boronic acid 3 Bromophenylboronic acid N butyldiethanolamine ester 3 Bromo 5 formylphenylboronic acid 4 Bromo 2 isopropylphenylboronic acid 2 Trifluoromethylpyridine 5 boronic acid pinacol ester 3 Bromo 4 chlorophenylboronic acid 4 Methoxy 2 trifluoromethoxy phenylboronic acid 2 Fluoro 4 formyl 6 methoxyphenylboronic acid 2 4 Difluoro 3 iodophenylboronic acid 6 Isobutoxy 2 methylpyridine 3 boronic acid 7 Chloro 1H indazole 4 boronic acid 2 Bromo 4 methylphenylboronic acid 3 5 Dichloro 2 6 difluorophenylboronic acid 6 Isopropoxynaphthalene 2 boronic acid 6 Isopropoxy 2 methylpyridine 3 boronic acid 2 3 Dimethoxypyridine 5 boronic acid 2 Fluoro 3 isopropoxypyridine 5 boronic acid 5 Chloro 2 methylsulfanyl pyridine 3 boronic acid 5 Fluoro 2 morpholin 4 ylmethyl phenyl boronic acid 4 Bromo 2 Chloro 5 trifluoromethyl phenylboronic acid 3 Bromo 5 methylsulfanyl phenylboronic acid 4 Bromo 2 fluoro 5 trifluoromethyl phenylboronic acid

2 Ethoxy 4 methylphenylboronic acid 2 Chloro 3 5 dimethylphenylboronic acid 4 Bromo 5 chloro 2 methylphenylboronic acid 2 6 Dimethoxybiphenyl 2 ylboronic acid 4 Amino 3 5 dimethylphenylboronic acid pinacol ester 4 Chloro 3 isopropoxyphenylboronic acid 2 Fluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid methyl ester 6 Fluoro 2 methylsulfanyl phenylboronic acid 2 Phenoxypyridine 5 boronic acid 2 Amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 Tert butylcarbonylamino phenylboronic acid pinacol ester 2 Bromo 4 chlorophenylboronic acid 5 Fluoro 2 morpholinomethyl phenylboronic acid hydrochloride 2 Methoxy 4 methylthio pyridine 5 boronic acid pinacol ester 2 Methoxy 4 methylthio pyridine 5 boronic acid 4 Isopropoxy 3 trifluoromethyl phenylboronic acid 4 Fluoro 3 methanesulfonyl phenylboronic acid 2 Methylthio thiophene 4 boronic acid 2 Methylthio thiophene 3 boronic acid 3 Methoxy 2 methylphenylboronic acid 2 4 N Boc piperazino pyridine 5 boronic acid 3 Bromo 5 carboxythiophene 2 boronic acid 3 Bromo 2 formylthiophene 5 boronic acid 2 Benzyloxy 4 methylpyridine 5 boronic acid 2 Phenoxypyridine 4 boronic acid 2 Isopropoxy 4 methylpyridine 5 boronic acid pinacol ester 2 Isopropoxy 4 methylpyridine 5 boronic acid 6 Ethoxy 2 fluoro 3 methylphenylboronic acid 2 4 Difluoro 3 hydroxymethyl phenylboronic acid 5 Methyl 1H indazole 4 boronic acid

4 Benzyloxy 2 chlorophenylboronic acid 4 Piperazin 1 ylmethyl phenylboronic acid 5 Methoxy 4 methylpyridine 3 boronic acid 6 Fluoro 2 hydroxy 3 methylphenylboronic acid pinacol ester 4 2 methylpropyl amino methyl phenylboronic acid 2 4 Difluoro 3 isopropoxyphenylboronic acid 4 Isobutoxyphenylboronic acid 2 Fluoro 4 morpholinomethyl phenylboronic acid pinacol ester 3 N N Dimethylaminomethyl phenylboronic acid pinacol ester 2 Fluoro 4 5 dimethoxyphenylboronic acid 5 Diethylamino methyl 2 fluorophenylboronic acid 5 Hydroxymethylthiophene 2 boronic acid pinacol ester 2 Fluoro 4 morpholinomethyl phenylboronic acid 4 Bromo 3 fluorophenylboronic acid pinacol ester 3 4 Dichloropyridine 5 boronic acid pinacol ester 3 Fluoro 4 piperidin 1 ylmethyl phenylboronic acid 2 Chloro 5 trifluoromethyl phenylboronic acid pinacol ester 3 Fluoro 4 methoxycarbonylphenylboronic acid pinacol ester 4 Methoxy 2 6 dimethylphenylphenylboronic acid pinacol ester 6 Azaindole 4 boronic acid 2 Fluoro 3 piperidin 1 ylmethyl phenylboronic acid 4 Hydroxy 3 methoxyphenylboronic acid pinacol ester 3 Bromo 2 fluoro 6 methoxyphenylboronic acid 5 Methyl 2 methylthio phenylboronic acid 3 Carboxy 5 trifluoromethyl phenylboronic acid 2 3 Difluoro 6 chlorophenylboronic acid 4 Bromo 3 trifluoromethyl phenylboronic acid pinacol ester 4 Trifluoromethylphenylboronic acid pinacol ester 3 Fluoro 5 pyrrolidinophenylboronic acid 5 Chloro 2 propoxy 4 pyridinyl boronic acid