5 Fluoro 4 methylpyridin 3 yl boronic acid 5 Hydroxy 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 3 Ffluoro N N dimethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 3 Cyano 2 methylphenylboronic acid 3 Fluoro 5 pyrrolidino phenylboronic acid pinacol ester 4 Methyl 3 phenylbenzenboronic acid 2 Dimethylamino 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl cyclohex 3 enol 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl aniline 2 Hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzenemethanol 2 6 difluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzenemethanol 3 Amino 4 methylphenylboronic acid pinacol ester 4 Cyano 2 methylphenylboronic acid pinacol ester 4 Tert butylaminomethyl phenylboronic acid pinacol ester 5 Bromo 2 methylphenylboronic acid pinacol ester 2 Fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl methanol 4 Dimethylamino 5 formylphenylboronic acid pinacol ester 3 Methoxy 4 methoxymethoxy phenylboronic acid 3 Chloro 5 cyanophenylboronic acid pinacol ester 7 Methyl 1H indazole 4 boronic acid pinacol ester 3 Chloro 2 fluoropyridne 5 boronic acid pinacol ester 3 4 Boc 1 piperazinylmethyl benzeneboronic acid pinacol ester 2 Hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 2 Chloro 6 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 2 Methoxyethoxy pyridine 5 boronic acid 3 Chloro 4 N N dimethylamino phenylboronic acid pinacol ester 2 Ethyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 4 Amino 3 trifluoromethoxy phenylboronic acid pinacol ester 4 Bromo 3 methoxyphenylboronic acid 4 Trifluoromethoxy 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline

3 Bromo 5 chloro 2 6 difluorophenylboronic acid pinaco ester 2 Amino 5 isopropylphenylboronic acid pinacol ester 2 3 4 Trifluoro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl aniline 3 N N Dimethylamino phenylboronic acid pinacol ester 5 Bromo 3 chloro 2 fluorophenylboronic acid 4 Chlorophenylboronic acid pinacol ester 4 Hydroxy 3 isopropylphenylboronic acid 2 Fluoro biphenyl 5 ylboronic acid 3 5 Dimethyl 2 methoxyphenylboronic acid 3 1H Tetrazol 5 yl phenyl boronic acid 5 Chloro 2 isopropoxypyridine 4 boronic acid 3 Bromo 5 chloro 2 6 difluorophenylboronic acid 2 6 Difluoro 4 methylthio phenylboronic acid 4 Methylbiphenyl 3 ylboronic acid 1 Methylindazole 5 boronic acid pinacol ester 2 6 Difluoro 3 methylthio phenylboronic acid pinacol ester 4 Pyridin 2 yl phenylboronic acid 4 Methoxy 2 methoxymethyl phenylboronic acid 2 5 Difluorophenylboronic acid pinacol ester 4 Formyl 2 trifluoromethyl phenylboronic acid pinacol ester 2 3 Dimethyl 4 methoxymethoxy phenylboronic acid 2 Chloro 4 trifluoromethyl phenylboronic acid pinacol ester 2 5 Difluoro 4 ethoxyphenylboronic acid 3 Ethoxy 2 6 difluorophenylboronic acid 2 6 Difluoro 3 propoxyphenylboronic acid 2 4 Bromo 2 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Chloro 6 trifluoromethyl phenylboronic acid pinacol ester 2 Methoxy 4 methylthio pyridine 3 boronic acid 4 Methoxy 3 methylthio phenylboronic acid 2 Choro 3 5 difluorophenylboronic acid

3 5 Difluoro 4 methylthio phenylboronic acid 2 Fluoro 3 methoxypyridine 4 boronic acid 5 Bromo 3 chloro 2 ethoxyphenylboronic acid 5 Chloro 2 methythio phenylboronic acid 2 Methyl 6 methylthio 3 pyridylboronic acid 4 Methyl 2 methylthio 5 pyridylboronic acid 2 Fluoro 5 methylsulfanyl pyridin 3 yl boronic acid 4 N O Dimethylhydroxylaminocarbonyl 2 chlorophenylboronic acid 5 Chloro 3 meththio phenylboronic acid 20Chloro 4 1 piperidinylcarbonyl phenylboronic acid 2 Chloro 4 1 pyrrolidinylcarbonyl phenylboronic acid 2 Chloro 4 methylcarbamoyl phenylboronic acid 4 Bromo 2 chloro 6 methylphenylboronic acid 2 Fluoro 3 methylsulfanyl phenylboronic acid 4 Methyl 2 methylthio phenylboronic acid 2 Isopropoxy 4 methylphenylboronic acid 4 Methoxy 2 pyrrolidin 1 ylmethyl phenylboronic acid 2 2 Methoxyethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 Chloro 1H indazole 4 boronic acid pinacol ester 3 Methyl 2 methylthio pyridine 5 boronic acid 4 N N Diisopropylaminocarbonyl phenylboronic acid 3 Chloro 2 fluoropyridne 5 boronic acid 5 Methothio thiophene 2 boronic acid 3 Morpholinomethyl phenylboronic acid pinacol ester 4 Fluoro 3 methylthio phenylboronic acid 2 Dimethylamino 4 methylpyridine 5 boronic acid 5 Ethoxymethyl pyridine 3 boronic acid 3 Bromo 6 Chloro 2 fluorophenylboronic acid pinacol ester 2 Fluoro 5 isopropoxypyridine 3 boronic acid 2 Isopropoxypyridine 4 boronic acid

3 Piperidin 1 ylmethyl phenylboronic acid pinacol ester 2 4 ethoxy 3 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 7 Methyl 1H indazole 4 boronic acid 7 Methoxy 1H indazole 4 boronic acid pinacol ester 3 Hydroxymethyl 2 methylphenylboronic acid pinacol ester 4 Cyano 2 6 dimethylphenylboronic acid 4 Bromo 3 5 dimethylphenylboronic acid 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzyl pyrrolidine 4 Methylthio 3 trifluoromethyl phenylboronic acid pinacol ester 3 CHLORO 2 CYANOPHENYLBORONIC ACID NEOPENTYL GLYCOL ESTER 4 4 methylpiperazin 1 yl methyl phenylboronic acid 3 4 Difluoro 5 formylphenylboronic acid 3 Pyrrolidin 1 ylmethyl phenylboronic acid 3 Chloro 2 morpholinomethyl phenylboronic acid 2 Fluoro 6 methoxy 4 methylphenylboronic acid 4 Piperidin 1 ylmethyl phenylboronic acid hydrochloride 4 Fluoro 3 methoxy 5 methylphenylboronic acid 3 Carboxy 4 chloro 2 fluorophenylboronic acid 4 Carboxy 2 chloro 3 methylphenylboronic acid 3 Benzyloxy 5 trifluoromethylphenylboronic acid 2 6 Dimethyl 4 isopropoxyphenylboronic acid 3 5 Dichloro 4 hydroxyphenylboronic acid pinacol ester 3 Fluoro 5 methoxycarbonylpohenylboronic acid pinacol ester 4 Methoxycarbonyl 2 methylphenylboronic acid 2 Methyl 4 methoxycarbonylphenylboronic acid pinacol ester 6 Propoxynaphthalen 2 yl boronic acid 2 Bromo 6 fluorobenzoic acid methyl ester 3 5 Difluoro 4 propan 2 yloxy benzoic acid 6 2 Methylpropoxy 2 naphthaleneboronic acid 3 5 Difluoro 4 isopropoxyphenylboronic acid