1 Methylindazole 5 boronic acid pinacol ester 3 Bromo 5 chloro 2 6 difluorophenylboronic acid 4 Formyl 2 trifluoromethyl phenylboronic acid pinacol ester 4 Methoxy 2 methoxymethyl phenylboronic acid 2 5 Difluorophenylboronic acid pinacol ester 4 Pyridin 2 yl phenylboronic acid 2 Chloro 6 trifluoromethyl phenylboronic acid pinacol ester 2 3 Dimethyl 4 methoxymethoxy phenylboronic acid 2 Chloro 4 trifluoromethyl phenylboronic acid pinacol ester 2 4 Bromo 2 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 6 Difluoro 3 propoxyphenylboronic acid 2 5 Difluoro 4 ethoxyphenylboronic acid 3 Ethoxy 2 6 difluorophenylboronic acid 2 Methoxy 4 methylthio pyridine 3 boronic acid 2 Choro 3 5 difluorophenylboronic acid 4 Methoxy 3 methylthio phenylboronic acid 3 5 Difluoro 4 methylthio phenylboronic acid 2 Methyl 6 methylthio 3 pyridylboronic acid 5 Chloro 2 methythio phenylboronic acid 5 Bromo 3 chloro 2 ethoxyphenylboronic acid 2 Fluoro 3 methoxypyridine 4 boronic acid 4 Methyl 2 methylthio 5 pyridylboronic acid 5 Chloro 3 meththio phenylboronic acid 2 Fluoro 5 methylsulfanyl pyridin 3 yl boronic acid 20Chloro 4 1 piperidinylcarbonyl phenylboronic acid 4 N O Dimethylhydroxylaminocarbonyl 2 chlorophenylboronic acid 2 Chloro 4 1 pyrrolidinylcarbonyl phenylboronic acid 2 Chloro 4 methylcarbamoyl phenylboronic acid 6 Chloro 1H indazole 4 boronic acid pinacol ester 4 Methoxy 2 pyrrolidin 1 ylmethyl phenylboronic acid

2 2 Methoxyethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Bromo 2 chloro 6 methylphenylboronic acid 2 Isopropoxy 4 methylphenylboronic acid 4 Methyl 2 methylthio phenylboronic acid 2 Fluoro 3 methylsulfanyl phenylboronic acid 3 Methyl 2 methylthio pyridine 5 boronic acid 3 Chloro 2 fluoropyridne 5 boronic acid 4 N N Diisopropylaminocarbonyl phenylboronic acid 3 Bromo 6 Chloro 2 fluorophenylboronic acid pinacol ester 2 Fluoro 5 isopropoxypyridine 3 boronic acid 5 Ethoxymethyl pyridine 3 boronic acid 2 Dimethylamino 4 methylpyridine 5 boronic acid 4 Fluoro 3 methylthio phenylboronic acid 3 Morpholinomethyl phenylboronic acid pinacol ester 5 Methothio thiophene 2 boronic acid 2 Isopropoxypyridine 4 boronic acid 7 Methyl 1H indazole 4 boronic acid 2 4 ethoxy 3 trifluoromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Piperidin 1 ylmethyl phenylboronic acid pinacol ester 4 Bromo 3 5 dimethylphenylboronic acid 4 Cyano 2 6 dimethylphenylboronic acid 3 Hydroxymethyl 2 methylphenylboronic acid pinacol ester 7 Methoxy 1H indazole 4 boronic acid pinacol ester 4 Methylthio 3 trifluoromethyl phenylboronic acid pinacol ester 4 4 methylpiperazin 1 yl methyl phenylboronic acid 3 CHLORO 2 CYANOPHENYLBORONIC ACID NEOPENTYL GLYCOL ESTER 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzyl pyrrolidine 3 Pyrrolidin 1 ylmethyl phenylboronic acid 2 Fluoro 6 methoxy 4 methylphenylboronic acid 3 Chloro 2 morpholinomethyl phenylboronic acid

3 4 Difluoro 5 formylphenylboronic acid 3 Benzyloxy 5 trifluoromethylphenylboronic acid 4 Piperidin 1 ylmethyl phenylboronic acid hydrochloride 4 Fluoro 3 methoxy 5 methylphenylboronic acid 3 Carboxy 4 chloro 2 fluorophenylboronic acid 4 Carboxy 2 chloro 3 methylphenylboronic acid 2 6 Dimethyl 4 isopropoxyphenylboronic acid 3 5 Dichloro 4 hydroxyphenylboronic acid pinacol ester 3 Fluoro 5 methoxycarbonylpohenylboronic acid pinacol ester 2 Methyl 4 methoxycarbonylphenylboronic acid pinacol ester 4 Methoxycarbonyl 2 methylphenylboronic acid 2 Bromo 6 fluorobenzoic acid methyl ester 6 Propoxynaphthalen 2 yl boronic acid 6 2 Methylpropoxy 2 naphthaleneboronic acid 2 Chloro 5 hydroxyiminomethyl phenylboronic acid 3 5 Difluoro 4 isopropoxyphenylboronic acid 3 5 Difluoro 4 propan 2 yloxy benzoic acid 3 5 Difluoro 4 1 pyrrolidinylcarbonyl phenylboronic acid 3 4 methylpiperazin 1 yl methyl phenylboronic acid 3 Methylaminomethyl phenylboronic acid 2 3 Dichloropyridine 4 boronic acid pinacol ester 2 Fluoro 3 methylpyridine 4 boronic acid 2 6 Difluoro 4 ethoxyphenylboronic acid 4 4 Isobutoxyphenyl phenylboronic acid 2 Ethoxy 4 methylpyridine 5 boronic acid 4 Carbamoyl 2 methoxyphenylboronic acid 4 Methylcarbamoyl 2 methoxyphenylboronic acid 4 Ethylcarbamoyl 2 methoxyphenylboronic acid 6 Bromo 3 chloro 2 fluorophenylboronic acid pinacol ester 4 Carboxy 2 6 difluorophenylboronic acid pinacol ester

8 Ethoxy 5 nitroquinoline 4 Hydroxy 3 trifluoromethyl phenylboronic acid 6 Butoxy 5 methylphenylpyridine 3 boronic acid 4 Chloro 2 fluoro 3 hydroxymethylphenylboronic acid 1 Isopropyl 1H pyrazole 5 boronic acid pinacol ester 2 Chloro 5 methoxymethylphenylboronic acid 2 Methyl 5 propoxyphenylboronic acid 5 Isopropoxy 2 methylphenylboronic acid 2 6 Dichloro 3 nitrophenylboronic acid pinacol ester 7 Methyl 1H indazole 5 boronic acid 4 Bromo 2 trifluoromethyl phenylboronic acid 2 Methoxy 5 methoxycarbonylphenyboronic acid 2 Methoxy 5 morpholinomethyl phenylboronic acid 5 Methylsulfonyl pyridine 3 boronic acid 5 Methylthio pyridine 3 boronic acid 2 5 Difluoro 4 hydroxyphenylboronic acid 3 Bromo 5 ethoxycarbonyl phenylboronic acid 5 Bromo 2 trifluoromethoxy benzoic acid methyl ester 5 Cyclopropylcarbamoyl 2 fluorophenylboronic acid 2 Fluoro 5 morpholine 4 carbonyl phenylboronic acid 2 Fluoro 5 piperidine 1 carbonyl phenylboronic acid 5 Ethylcarbamoyl 2 fluorophenylboronic acid 3 Cyano 5 methylphenylboronic acid 2 Fluoro 3 methoxypyridine 5 boronic acid 5 Benzylcarbamoyl 2 fluorophenylboronic acid 2 Fluoro 5 methoxy methyl carbamoyl phenylboronic acid 5 Diethylcarbamoyl 2 fluorophenylboronic acid 2 Fluoro 5 isopropylcarbamoyl phenylboronic acid 3 Chloro 2 formylphenylboronic acid pinacol ester 4 Chloro 2 fluoro 3 methylphenylboronic acid