2 4 chloro 2 6 difluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 chloro 4 6 dimethoxypyrimidin 5 yl boronic acid 4 bromothieno 2 3 b pyridine 1 Bromo 5 fluoro 2 iodobenzene 3 Bromopyridine 4 carboxaldehyde 2 Amino 5 bromo 1 2 4 triazolo 1 5 a pyridin 4 Bromo N methylaniline 2 Chloro 4 6 dimethoxybenzaldehyde 3 Chloro 4 formylbenzonitrile 3 methylbenzenesulfonyl chloride 3 Ethyltoluene 4 bromobenzo b thiophene 3 Hydroxybenzonitrile 4 Benzyloxy aniline 4 Phenoxy phenyl isothiocyanate 2 Chloro 4 methylphenol 2 Benzoylbenzoic acid 4 Bromomethyl benzoic acid 2 Nitrobenzenesulfonyl fluoride 2 METHOXY 5 SULFANYLPHENOL 6 Chloroindole 3 acetonitrile 1 2 Bromoethoxy 4 chlorobenzene 5 Isopropyl 2 methylphenol 4 4 Carboxy phenyl piperidine 1 carboxylic acid tert butyl ester 4 Trifluoromethyl benzoic acid 4 Trifluoromethyl benzoyl chloride 2 4 Dibromobenzoic acid 3 Amino 5 bromo 2 fluoropyridine 2 4 ethynylphenyl 6 fluorosulfonyl oxy 4 Quinolinecarboxylic acid 2 Chloro N 2 6 diisopropylphenyl quinolin 8 amine

5 2 CHLORO PHENYL ISOXAZOLE 3 CARBOXYLIC ACID 3 fluorooxane 4 4 diol 4 trifluoromethyl 1H pyrrolo 3 2 c pyridine 3 carbaldehyde 3 chloro 4 3 fluorophenyl methoxy aniline 2 4 dichloro 7 fluoropyrrolo 2 1 f 1 2 4 triazine 5 fluoro 1H indole 3 carbaldehyde 8 methyl 3 8 diazabicyclo 4 2 0 octane bis trifluoroacetic acid 2 difluoromethyl pyrrolidine hydrochloride 3 bromo 4 5 dichloropyridine 2 5 dibromoisonicotinaldehyde 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoquinoline 4 6 dimethoxypyrimidin 5 yl boronic acid 1 Bromo 3 fluoro 4 iodobenzene 2 Bromopyridine 4 carboxaldehyde 1 Amino 2 bromo 4 hydroxyanthrachinon 4 Bromo 2 methyl 6 nitroaniline 5 Chloro 2 4 difluorobenzaldehyde 3 Chloro 2 6 difluorobenzonitrile 3 Methoxybenzenesulfonyl chloride 3 Fluoropropan 1 ol 6 methylbenzo b thiophene 2 3 difluoro 4 pentyloxy phenylboronic acid 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 3 Benzyloxy aniline 3 Nitrophenyl isothiocyanate 5 Chloro 4 methyl 2 nitrophenol 1 4 Chlorophenyl buten 3 one 5 Fluoro 2 trifluoromethyl benzonitrile 3 Bromomethyl benzoic acid 3 BROMO 2 FLUOROBENZONITRILE

2 4 5 Trifluoro benzoic acid 2 Bromo thiazole 5 carboxylic acid ethyl ester 2 Fluoro 4 methylpyridine 5 boronic 3 Aminopropylphosphonic acid 2 4 Dichloro 5 picoline 3 Amino 2 bromo 5 fluoropyridine 5 1 Methylethyl 2 pyridinamine 2 amino 3 bromo 6 methyl pyridine 1 2 chloromethyl 4 trifluoromethyl phenyl 4 fluoro 2 methoxy 5 propan 2 yl benzene 3 methyl 3 8 diazabicyclo 4 2 0 octane bis trifluoroacetic acid 6 amino 4 fluoro 2 3 dihydro 1H indazol 3 one 3 fluoro 3 iodomethyl oxetane 3 fluoro 4 thiomorpholin 4 yl aniline 8 bromo 6 chloro 3 fluoroimidazo 1 2 b pyridazine 3 2 bromoethyl 5 fluoro 1H indole 2 3 difluoropyridin 4 ylboronic acid 3R 4S 1 tert butoxy carbonyl 4 3 fluorophenyl pyrrolidine 3 carboxylic acid 3 bromopyrazolo 1 5 a pyrimidine 4 4 dimethylamino phenyl 4 oxobutanoic acid 2 2 chloroacetamido N 4 chlorophenyl 4 5 6 7 tetrahydrobenzo b thiophene 3 carboxamide 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 4 4 3 4 dichloro 2 fluorophenyl amino 7 methoxyquinazolin 6 yl oxy piperidin 1 yl prop 2 en 1 one 6 bromo 4 methylquinoline 3 carboxylic acid 2 mercapto 6 trifluoromethyl pyrimidin 4 ol 2 methoxypyrimidin 5 yl boronic acid 2 4 tert butyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 borono 2 methoxybenzoic acid 2 Chloro 4 5 difluorobenzonitrile 2 Bromophenyl triflate 2 Fluoro 3 methylbenzenesulfonyl chloride

4 Chloro 2 5 difluorobenzaldehyde 3 Bromo 4 methylaniline 2 Bromopyridine 6 Amino 2H 1 4 benzoxin 3 4H one 1 Bromo 2 fluoro 4 iodobenzene 1 3 Dibenzoylbenzene 4 Chloro 5 methyl 2 nitrophenol 3 Iodophenyl isothiocyanate 4 4 Amino 3 5 dimethylbenzyl 2 6 dimethylaniline 4 Chloro 3 methylphenyl methanesulfonate 4 Fluoro 3 trifluoromethyl benzonitrile 2 Bromomethyl benzoic acid 1 2 4 5 TETRAKIS BROMOMETHYL BENZENE 2 4 6 Trifluorobenzylamine 3 Nitro 4 iodobenzoic acid 2 Amino 3 5 dibromopyrazine 1 3 Dimethylimidazolidone 5 Amino 3 bromo 2 chloropyridine 2 4 Dichloro 3 nitropyridine 1 bromo 4 fluoro 2 methoxy 5 propan 2 yl benzene 3 fluoro 3 fluoromethyl azetidine 4 TERT BUTOXYPHENYLBORONIC ACID PINACOL ESTER 2 3 dimethoxyphenyl boronic acid 3 5 Difluoropyridin 4 yl boronic acid 2 5 fluoro 1H indol 3 yl ethan 1 ol 6 Oxa 3 azabicyclo 3 1 0 hexane 3 sulfonyl fluoride 2 3 5 bis trifluoromethyl phenyl 2 methylpropanoic acid 3 bromomethyl 3 fluorooxetane 1R 1 4 chloro 3 fluorophenyl ethane 1 2 diol 2 chloropyrimidin 5 ol