3 bromopyrazolo 1 5 a pyrimidine 4 4 dimethylamino phenyl 4 oxobutanoic acid 2 2 chloroacetamido N 4 chlorophenyl 4 5 6 7 tetrahydrobenzo b thiophene 3 carboxamide 3R 4S 1 tert butoxy carbonyl 4 3 fluorophenyl pyrrolidine 3 carboxylic acid 3 methyl 3 8 diazabicyclo 4 2 0 octane bis trifluoroacetic acid 8 bromo 6 chloro 3 fluoroimidazo 1 2 b pyridazine 2 3 difluoropyridin 4 ylboronic acid 3 2 bromoethyl 5 fluoro 1H indole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 6 bromo 4 methylquinoline 3 carboxylic acid 2 4 tert butyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 methoxypyrimidin 5 yl boronic acid 2 mercapto 6 trifluoromethyl pyrimidin 4 ol 4 borono 2 methoxybenzoic acid 2 Bromophenyl triflate 4 Chloro 2 5 difluorobenzaldehyde 2 Chloro 4 5 difluorobenzonitrile 2 Fluoro 3 methylbenzenesulfonyl chloride 3 Bromo 4 methylaniline 6 Amino 2H 1 4 benzoxin 3 4H one 2 Bromopyridine 1 Bromo 2 fluoro 4 iodobenzene 3 Iodophenyl isothiocyanate 4 Chloro 5 methyl 2 nitrophenol 4 Chloro 3 methylphenyl methanesulfonate 4 Fluoro 3 trifluoromethyl benzonitrile 4 4 Amino 3 5 dimethylbenzyl 2 6 dimethylaniline 1 3 Dibenzoylbenzene 2 4 6 Trifluorobenzylamine 2 Bromomethyl benzoic acid

1 2 4 5 TETRAKIS BROMOMETHYL BENZENE 3 Nitro 4 iodobenzoic acid 2 Amino 3 5 dibromopyrazine 1 3 Dimethylimidazolidone 2 4 Dichloro 3 nitropyridine 5 Amino 3 bromo 2 chloropyridine 6 Oxa 3 azabicyclo 3 1 0 hexane 3 sulfonyl fluoride 2 3 dimethoxyphenyl boronic acid 4 TERT BUTOXYPHENYLBORONIC ACID PINACOL ESTER 1 bromo 4 fluoro 2 methoxy 5 propan 2 yl benzene 3 fluoro 3 fluoromethyl azetidine 1R 1 4 chloro 3 fluorophenyl ethane 1 2 diol 3 bromomethyl 3 fluorooxetane 2 3 5 bis trifluoromethyl phenyl 2 methylpropanoic acid 3 5 Difluoropyridin 4 yl boronic acid 2 5 fluoro 1H indol 3 yl ethan 1 ol 3 9 9 dimethylacridin 10 9H yl N N dimethylpropan 1 amine 1 benzo b thiophen 4 yl piperazine 3 4 carboxyphenoxy benzoic acid 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 triisopropylsilyl 1H pyrrole 4 5 6 7 tetrahydro 1H pyrazolo 4 3 c pyridine 6 bromo 2 methyl 1H imidazo 4 5 b pyridine 2 chloropyrimidin 5 ol 4 ethoxycarbonyl 3 fluorophenylboronic acid 2 4 chloromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 bis benzyloxy pyrimidin 5 yl boronic acid 4 Acetamido 3 bromobenzotrifluoride 4 fluorobenzo b thiophene 2 carboxylic acid 2 Chloro 3 6 difluorobenzonitrile 4 Ethoxybenzenesulfonyl chloride

3 Bromo 2 fluorobenzoyl chloride 2 Chloro 3 6 difluorobenzaldehyde 2 2 Dibromobutanal 3 Bromo 4 methoxyaniline hydrochloride 5 Bromo 2 nitropyridine 2 Amino 1 3 benzothiazol 1 Bromo 3 fluorobenzene 4 Trifluoromethyl benzophenone 4 Chloro 2 methoxyphenol 4 Fluorophenyl isothiocyanate 3 Fluoro 5 trifluoromethyl benzonitrile 2 Iodobenzenesulphonic acid 4 Bromo 2 methylbenzoic acid 4 methyl 2 3 5 6 tetrafluoro lbenzyl alcohol 2 3 DIFLUORO 4 METHYLBENZONITRILE 2 5 dihydro 1H Pyrrole 1 sulfonyl fluoride 3 Amino 5 bromo 2 chloropyridine 3 Fluoro 2 nitropyridine 2 Bromo 4 nitrotoluene 5 6 Dichloro 1 ethyl 2 methylbenzimidazole 4 Amino 1 Boc piperidine 4 carboxylic acid 4 Bromomethyl biphenyl 6 Chloro 3 fluoropyridine 2 carboxylic acid 5 11 Dihydro 11 chloroacetyl 6h pyrido 2 3 b 1 4 benzodiazepine 6 one 2 6 Difluoropyridin 4 yl boronic acid 1 5 chloro 6 fluoro 1H indol 3 yl ethan 1 ol 1R 2 tert butyldimethylsilyl oxy 1 4 chloro 3 fluorophenyl ethan 1 ol 3 fluorooxetan 3 yl methanamine 2 fluoro 4 methoxy 1 propan 2 yl benzene 3 1 fluoropropyl azetidine

4 Phenoxy 2 6 Diisopropyl Aniline 6 fluoropyridazin 3 amine 2R 3S 3 hydroxypyrrolidine 2 carboxylic acid trifluoroacetic acid 2 chloromethyl oxazolo 5 4 b pyridine 6 bromo 1H imidazo 4 5 b pyridine 2 methylbenzo d oxazol 5 ol 1 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrole 2 methylpropane 1 2 diamine 2 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzaldehyde 4 cyanobenzohydrazide 2 6 difluoropyridin 3 amine 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 chloro 5 cyanophenylboronic acid 7 fluorobenzo b thiophene 2 carboxylic acid 4 fluorobenzofuran 2 carboxylic acid 3 4 Difluorobenzenesulfonyl chloride 2 Bromo 3 methylaniline 2 Chloro 4 5 difluorobenzaldehyde 4 Butyryl benzonitrie 5 Aminobenzimidazole 2 Bromo 6 methylpyridine N oxide 1 Bromo 2 fluorobenzene 2 Trifluoromethyl benzophenone 2 Chloro 4 methoxyphenol 3 Fluorophenyl isothiocyanate 4 Trifluoromethyl benzyl amine 2 Fluoro 6 trifluoromethyl benzonitrile 3 Bromo 5 methylbenzoic acid 4 Bromo 2 3 5 6 tetrafluorobenzaldehyde 5 6 Dihydro 6 oxo 11H pyrido 2 3 b 1 4 benzodiazepine