1 2 morpholinoethyl 1H pyrazol 4 yl boronic acid 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 benzyloxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 diethoxymethyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 chlorothieno 3 2 b pyridine 5 bromothieno 3 2 b pyridine 4 chloro 3 methyl 1H pyrazolo 3 4 b pyridine 3 iodo 6 nitro 1H indazole 3 iodo 5 nitro 1H indazole 3 bromo 5 nitro 1H indazole 6 chloro 3 iodo 1H indazole 3 bromo 6 chloro 1H indazole 5 bromo 3 iodo 1H indazole 3 bromo 4 chloro 1H indazole 3 bromo 7 chloro 1H indazole 7 bromo 3 chloro 1H indazole 4 fluoro 3 iodo 1H indazole 5 fluoro 3 iodo 1H indazole 3 bromo 5 fluoro 1H indazole 6 fluoro 3 iodo 1H indazole 3 bromo 6 fluoro 1H indazole 7 fluoro 3 iodo 1H indazole 7 bromothieno 2 3 c pyridine 5 trifluoromethyl benzo b thiophene 2 carboxylic acid 7 bromo 3 methylbenzo b thiophene 5 fluoro 3 methylbenzo b thiophene 5 7 dichloro 1H pyrazolo 3 4 c pyridine 4 bromo 1H pyrazolo 3 4 c pyridin 3 amine 7 bromo 1H pyrazolo 3 4 c pyridine 5 trifluoromethyl 1H pyrazolo 3 4 c pyridine

7 trifluoromethyl 1H pyrazolo 3 4 c pyridine 3 bromo 1H pyrazolo 4 3 b pyridine 5 bromo 1H pyrazolo 4 3 b pyridine 6 chloro 1H pyrazolo 4 3 b pyridine 3 bromo 1H pyrazolo 3 4 c pyridine 7 bromo 1H pyrazolo 4 3 c pyridin 3 amine 1H pyrazolo 4 3 c quinolin 3 amine 3 iodo 5 trifluoromethyl 1H indazole 5 iodo 1 methyl 1H pyrazolo 3 4 b pyridin 3 amine 5 bromo 1 methyl 1H pyrazolo 3 4 b pyridine 4 6 dimethyl 1H pyrazolo 3 4 b pyridin 3 amine 5 bromo 6 trifluoromethyl 1H pyrazolo 3 4 b pyridin 3 amine 6 chloro 1H pyrazolo 4 3 c pyridin 3 amine 3 phenyl 1H pyrazolo 4 3 c pyridine 3 bromo 1H pyrazolo 4 3 c pyridine 3 bromo 5 trifluoromethyl 1H indazole 3 chloro 5 trifluoromethyl 1H indazole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methyl acetate 2 chloro 6 methoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 propoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 methyl 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 4 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl morpholine 1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl piperazine 2 piperidin 1 yl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 ethoxy 6 methylpyridin 3 yl boronic acid 2 methoxy 5 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 3 2 b pyridine 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrido 2 3 b pyrazine 2 3 dimethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine

2 amino 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinic acid 3 iodo 6 trifluoromethyl 1H indazole 6 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 5 chloro 3 trifluoromethyl 1H indazole 3 bromo 6 trifluoromethyl 1H indazole 3 methyl 1H indazol 7 amine 4 fluoro 1H indazole 6 carboxylic acid 2 3 4 dimethylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 4 chloro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 4 fluoro 3 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 chloro 6 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 fluoro 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 fluoro 5 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 fluoro 2 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 4 fluoro 3 methylphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 5 chloro 2 methoxymethoxy phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 chloro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl ethanol 2 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenyl ethanol 4 4 5 5 tetramethyl 2 2 3 4 trifluorophenyl 1 3 2 dioxaborolane 2 4 chloro 2 6 difluorophenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 2 fluoro 4 methoxyphenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 fluoro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl phenol 5 fluoro 2 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 2 trifluoromethyl phenol 4 4 5 5 tetramethyl 2 perfluorophenyl 1 3 2 dioxaborolane 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzonitrile 2 4 chloromethyl phenyl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane

3 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 chloro 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl phenol 2 hydroxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzoic acid 3 4 bis methoxycarbonyl phenyl boronic acid 2 3 difluoro 4 methylphenyl boronic acid 2 4 dichloro 6 fluorophenyl boronic acid 4 fluoro 2 methoxyphenyl boronic acid 4 cyano 3 5 difluorophenyl boronic acid 2 chloro 5 methoxyphenyl boronic acid 3 chloro 4 hydroxyphenyl boronic acid 2 hydroxy 5 methoxyphenyl boronic acid 3 fluoro 4 hydroxyphenyl boronic acid 3 5 difluoro 2 hydroxyphenyl boronic acid 4 5 difluoro 2 hydroxyphenyl boronic acid 3 chloro 4 cyanophenyl boronic acid 2 chloro 5 fluorophenyl boronic acid 3 chloro 5 fluoro 4 methoxyphenyl boronic acid 4 hydroxy 2 methylphenyl boronic acid 5 borono 2 hydroxybenzoic acid 4 fluoro 2 hydroxyphenyl boronic acid 2 hydroxy 4 trifluoromethyl phenyl boronic acid 2 hydroxy 5 trifluoromethyl phenyl boronic acid 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isoindolin 1 one 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 2 5 methoxynaphthalen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl indoline 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indole 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole