1H Pyrazole 3 5 dicarboxylic acid diethyl ester 2 Bromo 4 chlorobenzaldehyde 3 Ethoxy 4 methoxybenzaldehyde 4 Bromo 2 3 difluorobenzaldehyde 2 5 Dibromoanisole 4 Bromobenzyl bromide 5 Amino 2 bromopyridine 5 Chloroisatoic anhydride 2 Bromobenzonitrile 1 1 1 3 3 3 hexafluoroisopropylmethacrylate 2 chloro 6 trifluoromethyl pyrimidin 4 amine 4 4 bromo 3 fluorophenyl methyl 1λ⁶ thiomorpholine 1 1 dione 4 Amino N cyclopropylbenzenemethanamine 3 fluoromethyl 3 methylazetidine 5 fluoropyridin 3 yl methanol 5 1 1 1 trifluoro 2 methylpropan 2 yl 1 2 oxazol 3 amine 1R 2S 2 amino 4 4 difluorocyclopentane 1 carboxylic acid hydrochloride 2 3 fluorocyclobutyl acetyl fluoride 1 4 fluorophenyl cyclobutan 1 amine 4 fluoroazepane hydrochloride 1 tert butyl 2 methyl 2s 4s 4 trifluoromethyl pyrrolidine 1 2 dicarboxylate 6 methylnaphthalen 1 amine 6 chloro 1H benzo d imidazole 2 7 diazaspiro 4 4 nonan 1 one 1 2 4 bromophenoxy ethyl pyrrolidine 3 methoxymethyl phenylboronic acid 5 Fluoro 1 2 3 4 tetrahydroquinoline hydrochloride 3 bromoimidazo 1 2 a pyridine 4 chloro 1H pyrazolo 3 4 c pyridine 4 6 dimethylpyridin 2 1H one

3 isopropoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 4 dimethylphenyl boronic acid 4 bromo N tert butyl pyridin 2 amine 2 ethoxy 6 fluorophenylboronic acid 4 6 dibromopyrimidine 5 carbaldehyde 3 Bromo 4 fluorobenzonitrile 6 Fluoro 2 methylindole 4 4 4 Trifluorobutyric acid 2 chloro 4 iodophenol 4 Bromo 3 ethylaniline 3 5 Bis trifluoromethyl phenyl isothiocyanate 5 Bromo 2 nitrophenol 3 5 Bis trifluoromethyl benzophenone 1 Bromo 2 chloro 5 iodobenzene 5 Amino 2 methylpyridine 2 Fluoro 6 hydroxybenzonitrile 4 Fluoro 2 trifluoromethyl benzyl amine 3 Bromo 5 fluorobenzoic acid 2 4 6 Triisopropylbenzenesulfonyl chloride 2 Bromoisophthalic acid dimethyl ester 2 Amino 4 5 dichlorophenol 2 Iodo 4 methylaniline 2 4 Dihydroxybenzonitrile 3 Trifluoromethylthio bromobenzene 4 Bromobenzoic acid 2 Bromo 5 fluoropyridine 5 Chloroindoline 4 AMINO 5 AZAINDOLE 2 azetidin 3 yl 2 2 difluoroethan 1 ol 4 ​Piperidinone 2 ​methyl ​ 2 ​2 ​2 ​trifluoroacetate 1 1

2 chloro 5 trifluoromethyl pyrimidin 4 amine 3 5 2 cyclopropylpyrimidin 5 yl 1H pyrrolo 2 3 b pyridine 3 carbonyl 2 4 difluoroaniline 1R 2S 2 amino 4 4 difluorocyclopentane 1 carbonitrile 2 3 3 difluorocyclobutyl acetaldehyde 4 fluoroazepane 3 fluoro 4 2H 1 2 3 4 tetrazol 5 yl aniline 6 methyl 1 naphthoic acid 4 methoxymethoxy phenylboronic acid 7 bromo 5 methylbenzo e 1 2 4 triazin 3 amine 2 hydroxypyridin 3 yl boronic acid 8 bromo 2 3 dimethyl 6 trifluoromethyl imidazo 1 2 a pyridine 4 bromo 1H pyrazolo 3 4 c pyridine 6 methyl 2 trifluoromethyl nicotinic acid 5 Fluoroindole 2 carboxylic acid ethyl ester 3 trifluoromethyl benzhydrol 4 dimethoxymethyl pyrimidine 4 bromo N methylpyridin 2 amine 5 ethoxy 2 fluorophenylboronic acid 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl oxy acetonitrile 2 methoxy 3 trifluoromethyl phenyl boronic acid 2 Bromo 3 fluorobenzonitrile 11 Bromoundecanoic acid methyl ester 4 Bromo 2 ethylaniline 3 bromo 2 6 difluorophenol 2 Amino 5 picoline 4 Bromo 3 nitrophenol 3 3 Bis trifluoromethyl benzophenone 1 Bromo 5 chloro 3 fluoro 2 iodobenzene 2 Fluoro 5 trifluoromethyl benzyl amine 4 Trifluoromethyl benzenesulfonyl chloride

2 Fluoro 4 hydroxybenzonitrile 2 Bromo 6 fluorobenzoic acid 3 5 DICHLOROBENZONITRILE 2 Bromo 3 fluoro 5 trifluoromethyl pyridine 2 Phenylpyridine 2 Trifluoromethoxy benzylsulphonyl chloride 2 Amino 2 fluoro 5 nitrobenzophenone 2 Bromobenzoic acid 2 Iodobenzaldehyde dimethyl acetal 4 Bromo 3 trifluoromethyl phenol 4 fluorosulfonyl oxy 3 methoxy Benzaldehyde 3 Bromo 2 chloropyridine 3 difluoromethyl oxetane 3 carboxylic acid 2 2 3 4 4 4 hexafluorobutyl methacrylate 6 6 difluoro 3 azabicyclo 3 1 0 hexane hemioxalate 3 trifluoromethyl pyrrolidin 3 ol hydrochloride 7 fluoro 1H indol 5 amine 2 4 difluoro 3 5 iodo 1H pyrrolo 2 3 b pyridine 3 carbonyl aniline 4 amino 2 chloro 5 fluoropyrimidine 3 5 difluoropyridin 2 yl methanol 6 phenylpyrazin 2 amine 4 N acetylsulfamoyl phenylboronic acid 4 fluoropiperidine hydrochloride 6 6 difluorospiro 3 3 heptan 2 yl methanamine hydrochloride 4 chloro 3 5 methyl 3 4 2 pyrrolidin 1 yl ethoxy phenyl amino benzo e 1 2 4 triazin 7 yl phenol 6 8 dibromo 2 3 dimethylimidazo 1 2 a pyridine 4 chloro 6 methyl 1H pyrazolo 3 4 d pyrimidine 3 dimethylcarbamoyl phenylboronic acid 2 isobutoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 4 6 trimethylnicotinic acid