1 benzyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 1H one 8 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 3 propylcarbamoyl phenylboronic acid 4 Isopropyl 2 nitrotoluene 3 bromopyrazin 2 amine 6 7 difluorobenzo b thiophene 2 Amino 5 acetylbenzonitrile 4 Bromo 2 fluorobenzylamine 2 3 4 5 Tetrafluoroacetophenone 5 Fluorobenzene 1 3 diol 1 Bromocyclopropane 2 5 Difluoronitrobenzene 4 Methoxy 3 trifluoromethyl acetophenone 2 Chloro 6 fluoro 3 trichloromethyl benzene 4 Amino 2 methoxyphenol 4 Bromo 3 methylbenzamide 2 2 Difluoro 5 aminobenzo d 1 3 dioxole 1 BROMO 2 4 DIMETHOXYBENZENE 3 4 chlorophenyl 3 oxopropanenitrile 3 Chloro 5 fluorobenzonitrile 4 Bromo 2 chlorobenzenesulphonyl chloride 2 Amino 3 bromo 5 methylbenzoic acid 4 Chloro 2 hydroxybenzaldehyde 4 Hydroxy 1 indanone 4 Chloroisatoic anhydride 2 Methoxy 5 pyridineboronic acid 2 6 Dibromo 4 fluoroaniline 3 5 Dimethoxyphenylboronic acid 2 2 Bis 3 4 dimethylphenyl hexafluoropropane 1 3 trifluoromethyl cyclobutyl ethan 1 amine

4 chlorosulfonyl 3 fluorobenzoic acid 4S 5S 5 3 5 bis trifluoromethyl phenyl 4 methyl 1 3 oxazolidin 2 one 8 bromo 2 chloro 6 trifluoromethyl quinazoline 3 acetyl 2 hydroxybenzonitrile 2 chloro 5 trifluoromethyl pyridin 3 ol 2 dimethylamino phenylboronic acid 3 difluoromethoxy azetidine hydrochloride 2 chloro 4 iodo 5 trifluoromethyl pyridine 2 BroMo 3 phenylpyridine 2 3 6 trichlorophenylboronic acid 6 methoxybenzofuran 2 ylboronic acid 7 chloro 1 2 methyl 4 nitrobenzoyl 3 4 dihydro 1H benzo b azepin 5 2H one 2 chloro 3 iodoisonicotinonitrile 2 methyl 7 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 3 methylcarbamoyl phenylboronic acid 3 bromo 2 fluorobenzyl bromide 1 2 Difluoro 4 methylsulfonyl benzene 2 trifluoromethyl pyridin 3 ol 7 bromo 6 fluorobenzo b thiophene 2 Amino 4 Bromo 3 fluorobenzoic acid 2 3 6 Trifluoroacetophenone 5 Fluoro 2 nitrophenol 1 3 trifluoromethyl phenyl ethanone oxime 2 4 Difluoronitrobenzene 4 Methoxy 2 2 2 trifluoroacetophenone 3 Chloro 4 fluorobenzotrifluoride 3 Amino 4 methylphenol 2 Bromo 6 fluorobenzamide 3 3 chlorophenyl 3 oxopropanenitrile 3 Bromobenzenesulfonyl chloride

3 Chloro 4 fluorobenzonitrile 5 Amino 2 bromobenzoic acid 1 BROMO 2 3 6 TRIFLUOROBENZENE 3 4 5 Trifluoropyridine 3 5 Dibromo 2 methylpyridine 4 Nitrobenzoyl chloride 2 Methoxy 3 pyridineboronic acid 1 Boc 2 methoxycarbonylmethylpiperazine 2 Iodo 3 methylbenzoic acid 4 Chloro 2 fluorobenzonitrile 4 Cyanophenylboronic acid 2 methyl 4 heptafluoroisopropylaniline 3 Oxazolidinesulfonyl fluoride 2 oxo 1 3 trifluoromethyl cyclobutyl ethan 1 ol 6 fluoro 5 methoxypyridine 3 carbaldehyde 4R 5R 5 3 5 bis trifluoromethyl phenyl 4 methyl 1 3 oxazolidin 2 one 5 fluoropyrimidin 2 yl methanol 5 fluoropyrimidine 4 carboxylic acid 5 fluoro 3 methyl 1H pyrrolo 2 3 b pyridine 3 difluoromethoxy azetidine 1S 5S 3 methyl 3 6 diazabicyclo 3 2 0 heptane bis trifluoroacetic acid 5 4 4 5 5 tetraMethyl 1 3 2 dioxaborolan 2 yl picolinaMide 6 bromo 5 chloroisoquinoline 4 isopropoxyphenol 2 boronobenzoic acid 2 methoxy 4 6 dimethylphenylboronic acid 2 3 formylphenyl acetic acid 4 chloroquinolin 2 amine 2 fluoro 6 methoxybenzaldehyde 7 chlorothieno 3 2 b pyridine

6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 2 5 difluoro 4 methoxyphenylboronic acid 6 bromo 7 fluorobenzo b thiophene 2 6 Dibromochlorobenzene 3 fluoro 4 iodophenol 4 bromo 2 trifluoromethyl benzyl alcohol 4 Fluoro 2 nitroanisole 4 Chlorobenzotrifluoride 3 Difluoromethoxy nitrobenzene 2 Trifluoromethyl phenylboronic acid 2 3 5 Trifluoroacetophenone 4 Methoxy 3 methylacetophenone 4 Bromo N methoxy N methylbenzamide 2 Amino 3 fluorophenol 3 Chloro 2 fluorobenzonitrile 3 2 chlorophenyl 3 oxopropanenitrile 1 BROMO 2 3 DIFLUOROBENZENE 4 Amino 3 bromobenzoic acid 2 Bromobenzenesulfonyl chloride 4 Chlorophenylboronic acid 2 Chloro 4 fluorobenzonitrile 2 Fluoro 5 trifluoromethyl phenylboronic acid 2 Bromo 6 chloropyridine 2 Nitrophenylboronic acid 1 Bromo 3 chloro 2 5 difluorobenzene 5 4 4 5 5 Tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 1 2 2 trifluorocyclobutyl methanol 2 chloro 5 trifluoromethyl pyridin 4 yl boronic acid 5 fluoropyrimidine 2 carbaldehyde 5 3 5 difluorophenyl methyl 1H indazol 3 amine