1 Boc piperidine 4 carboxylic acid ethyl ester 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indole 2 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d 1 2 3 triazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl quinazolin 4 ol 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 6 Chlorobenzo d isoxazol 3 ol 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H benzo d imidazole 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl benzo d oxazol 2 3H one 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 5 Amino 1 2 4 thiadiazole 7 methylimidazo 1 2 a pyridin 6 yl boronic acid 7 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 2 3 dimethyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyrimidine 2 Chloro 4 methoxyphenylacetonitrile 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl imidazo 1 2 a pyridine 3 Amino 5 hydroxypyrazole 1 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 1 methyl 6 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazol 3 amine 1H indazol 5 yl boronic acid 7 Ethyl 10 hydroxycamptothecin 1H indazol 4 yl boronic acid 1H indazol 7 yl boronic acid 2 4 6 Trichloropyridine 5 Methyl 3 2H pyridazinone 4 Nitrobenzyl chloroformate 1 methyl 1H indazol 7 yl boronic acid 3 methylsulfonyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 tert butylbenzenesulfonyl chloride

5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinaldehyde 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl methanol 4 Phenoxybenzoic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl methanol 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 yl ethanone 4 Ethoxybenzoyl chloride 3 butoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 Fluoronaphthalene 3 ethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 4 Cyclohexanedicarboxylic acid 4 4 5 5 tetramethyl 2 3 methylbenzofuran 6 yl 1 3 2 dioxaborolane 3 Chlorobenzaldehyde 2 iodo 4 methoxyaniline 7 methylbenzofuran 5 yl boronic acid 2 7 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Bromo 4 butanolide 2 benzo b thiophen 3 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 Methyl 4 methylthio phenol 3 hydroxymethyl thiophen 2 yl boronic acid 6 Bromopyridine 2 carboxylic acid ethyl ester 3 bromothiophen 2 yl boronic acid 6 Fluoronicotinic acid methyl ester 2 Chloro 6 iodoaniline 4 bromo 5 methylthiophen 2 yl boronic acid 3 methylthiophen 2 yl boronic acid 3 chloro 2 iodoaniline 5 Ethyl 2 methylpyridine 4 4 Methylpiperazino benzoic acid 2 5 chlorothiophen 2 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole

3 Aminopropylphosphate 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiazole 1 Chloro 3 isothiocyanato 2 methylbenzene 1 4 chlorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 Bromo 3 methoxypropanol 4 Benzyloxyphenol 1 4 fluorophenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 1 3 chlorophenyl 1H pyrazol 4 yl boronic acid 1 4 fluorophenyl 1H pyrazol 4 yl boronic acid 5 Amino 4 chloro 2 methylphenol 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 5 Bromo 3 fluoro 2 methoxypyridine 2 Chloro 5 fluoro 4 methylpyridine 2 4 Diaminopyrimidine 5 carbaldehyde 4 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl morpholine 2 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 yl propan 2 ol 2 piperidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 trifluoromethyl biphenyl 4 carboxylic acid 5 4 trifluoromethylphenyl 1H pyrazole 2 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 6 Methyl 5 nitropyridin 2 ol 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 carbonitrile 3 Amino 2 6 dichloropyridine 2 chloro 5 bromobenzaldehyde 4 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 isopropoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 Bromo 2 methylbenzaldehyde 2 ethoxy 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 1 hydroxymethyl cyclopropaneacetonitrile

3 Amino 2 Hydroxyacetophenone 2 chloro 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 chloro 2 fluoropyridin 3 yl boronic acid 3 5 Dichloro 2 Bromopyridine 5 fluoro 2 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Mercapto Thiadiazole 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 ol 3 Bromothiophene 2 carboxylic acid 3 chloro 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 nitro 4 trifluoromethyl aniline 4 Bromo 2 3 difluorobenzaldehyde 2 3 difluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Trifluoromethoxy benzylsulphonyl chloride 1 1 Dimethoxy acetone 2 3 dichloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 5 Dimercapto 1 3 4 thiadiazole 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 amine 2 Methyl 2 propanesulfinamide 2 methoxy 4 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 7 Nitroindole 2 carboxylic acid 5 Bromo 6 hydroxy 3 pyridinecarboxylic acid 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinonitrile 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 3 amine 5 Chloro 2 hydroxy 3 picoline 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Quinoxalinecarboxylic acid 2 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 8 Fluoro 4 chromanone 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 4 trifluoromethyl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine