2 Bromo 1 4 bromo 1 1 biphenyl 4 yl ethanone 5 Bromo 2 3H benzofuranone 3 Bromo 7 chloroquinoline 7 Bromo 3 methoxyquinoline 1 4 Methoxy benzyl piperidine 2 4 dione 8 Bromochroman 3 one 8 Oxabicyclo 3 2 1 octan 3 one 1R Dimenthyl succinate 4 Boc 3 2 Oxo ethyl morpholine 2 Cyclohexen 1 one 4 4 Chlorobenzenesulfonyl benzaldehyde 7 Bromo 2 3 dihydro 1 8 naphthyridin 4 1H one 5 Nitroisatoic anhydride 4 Morpholinocyclohexanone 2 Azabicyclo 2 2 2 octane 2 6 dicarboxylic acid 2 1 1 dimethylethyl 6 methyl ester 1R 4S 6R rel 1 3 4 Dimethylphenyl 2 Phenylethane 1 2 Dione 1 4 1 3 Dioxolan 2 yl phenyl ethanone 3 Chromanone 1 Acetamido acetone 2 Cyclohepten 1 one 1 2H Naphthalenone 3 4 dihydro 7 phenylmethyl 1 Boc 3 5 dioxopyrrolidine 5 Bromo 3 methoxybenzaldehyde 4 Bromo 3 hydroxybenzaldehyde 9H Fluoren 9 yl methyl 2 oxoethylcarbamate 8 Methyl 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 6 carbaldehyde 3 Hydroxy 5 methoxybenzaldehyde 7 Methoxy 4 trifluoromethyl coumarin 4 Boronicacid biphenyl 4 carboxylicacid methyl ester 5 Boc Amino pyridine 3 boronic acid pinacol ester

3 Pyrrolylboronic acid 3 tert Butoxycarbonyl amino methyl pyridin 4 yl boronic acid 1 1H indol 3 yl 2 2 phenylvinyl sulfonyl 1 2 dihydroisoquinoline 1H 1 2 4 Triazole 3 5 diamine N3 4 aminosulfonyl phenyl 1 3 5 dimethyl 2 thienyl carboyl 9CI 1 3 Chlorobenzyl 6 4 isopropoxyphenyl 3 pentanoyl amino indole 2 carboxylic acid 3 4 Chlorobenzoylamino 1 3 chlorobenzyl 6 4 isopropoxyphenyl indole 2 carboxylic acid 1H 1 2 4 Triazole 3 5 diamine N3 4 2 dimethylamino ethyl mino sulfonyl phenyl 1 3 5 dimethyl 2 thienyl carbonyl 9CI 2 4 2 4 Dioxo 5 thiazolidinyl methyl phenoxy acetic acid 3 Cyclohexyl L alanine hydrate 2S 3R 2 Methyl 3 morpholinecarboxylic acid 4S 1 Boc 4 Methyl L proline 1S 3aR 6aS Hexahydro cyclopenta c pyrrole 1 2 dicarboxylic acid 2 tert butyl ester 1 Amino cyclopentanecarboxylic acid ethyl ester hydrochloride 1S 3aR 6aS Octahydro cyclopenta c pyrrole 1 carboxylic acid hydrochloride 3 Pyridin 4 yl 3 9 diazaspiro 5 5 undecane 3 N Boc 3 methylbutane 1 3 diamine HCl 6aR tert Butyl 6a trifluoromethyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 6aR tert Butyl 6a phenyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 3aR tert Butyl 3a ethyl hexahydropyrrolo 3 4 c pyrrole 2 3a 1H dicarboxylate 4 Bromophenyl piperidin 4 yl methanone 1 2 3 4 Tetrahydroisoquinolin 4 ol 2 Amino 2 2 pyridyl ethanol 2 Methoxy 1 propanamine 3R 4R 4 4 Fluorophenyl 3 piperidinemethanol 4 4 Acetylpiperazin 1 yl 3 trifluoromethyl aniline 3 Dimethylamino pyrrolidine 1 Cbz 3 aminomethylazetidine 1 6 7 dimethoxy 2H benzo d 1 3 dioxolan 5 yl prop 2 ylamine 1S 2R 2 Amino cyclohexanol 1S 2R 2 Amino cyclohexanol HCl

3 8 Diazabicyclo 3 2 1 octane 1 Amino 3 buten 2 ol 4 3 nitrophenyl piperidine 2S 5S 2 5 Dimethylmorpholine 1S 3R 3 Aminocyclopentanol 1S 3S 3 Aminocyclopentanol 1 Cyclopropylethanamine 1R 3R 3 Aminocyclopentanol 2 Ethenylmorpholine 1 Oxa 7 azaspiro 4 5 decane 6 Oxa 2 aza spiro 4 5 decane 7 Oxa 2 aza spiro 4 5 decane 8 Oxa 2 azaspiro 4 5 decane 2 piperidin 2 yl ethanamine 2 2 Methoxyethyl piperidine hydrochloride 2 2 pyridinyl morpholine 3 2 Pyridyl morpholine 2 Thiophen 3 yl morpholine 3 2 Thienyl morpholine 3 Thiophen 3 yl morpholine 2 Cyclopropylmorpholine 3 Cyclopropylmorpholine 2 Cyclobutylmorpholine 3 Cyclohexylmorpholine 3 Cyclobutylmorpholine 2 Phenyl 2 6 diazaspiro 3 3 heptan 1 one 2 Benzylmorpholine 1 3 Chloro benzyl 1 2 3 4 tetrahydro quinoxaline 2 Pyrrolidineacetic acid ethyl ester 1 Boc 2 Aminomethylazetidine hydrochloride

2 Azabicyclo 2 2 1 hept 5 ene 3 Pyrrolidin 3 yl aniline dihydrochloride 3 Amino cyclopentanone 1 Boc 4 1 pyrrolidinyl 3 6 dihydro 2H pyridine 6 Aminomethyl 3 morpholinone hydrochloride 2 2 Dimethylpyrrolidine 4 Ethyl 2 3 methyl 4 nitrophenyl morpholine 1 Methyl 2 piperazinemethanamine 2 Piperidin 4 yl ethylamine dihydrochloride 3 Aminotetrahydrofuran 1R 4R 5 Methyl 2 5 diazabicyclo 2 2 1 heptane 3 Aminocyclobutanone hydrochloride 2 N Boc aminomethylmorpholine 3 Maleimidopropionic Acid hydrazide Trifluoroacetic Acid 2 Isopropylmorpholine 1 4 Methoxyphenethyl 4 aminopiperidine 2S 6S 2 6 Dimethyl piperazine 2HCl 7 2 Aminoethyl 2 3 dihydro 1 benzofuran 2 Maleimidoethylamine hydrochloride 1 3 Formylphenyl piperazine 4 Piperidin 3 ylaniline 1 3 Pyrrolidinyl cyclopropanamine 2 Methyl 7 phenylmethyl 2 7 Diazaspiro 3 5 nonane 2S 6S 2 6 diphenyl morpholine 2R 6R 2 6 Dimethylmorpholine 2 Piperazin 1 yl benzaldehyde 5 4 Methylpiperidin 1 yl pyridin 2 amine 2 Chloro 5 hydrazinopyridine 4 4 Boc piperazin 1 yl 3 fluoroaniline 2 Hydrazino 3 fluoropyridine