2 BROMO 1H INDOLE 3 Chloro 2 methoxybenzaldehyde 3 Amino 1 cyclopentyl 1H pyrazole 4 carbonitrile 3 5 Dibromo N N dimethylpyrazinamine 1 2 BROMOETHOXY 4 FLUOROBENZENE 4 Bromo 1 methoxyisoquinoline 4 8 DIHYDROXYQUINOLINE 5 Fluoro 2 methoxyphenyl methanol 2 Methyl 2H indazol 4 amine 2 tert Butoxycarbonylaminomalonic acid monoethyl ester 3R 3 chloromethyl 1 4 dioxaspiro 4 5 decane 2 Hydroxy 3 6 dimethylbenzaldehyde 5 acetylamido 2 chloroaniline 2 Chloro 5 iodopyrazine 2 Chloro 6 fluoroquinoxaline 5 Methyl L norleucine 6 Methylheptyl 9 octadecenoate 2 Bromo 6 methylpyrazino 2 3 b pyrazine 2 Bromo 4 5 6 7 tetrahydrothiazolo 5 4 c pyridine hydrochloride 2 Amino N N diethylbenzenesulfonamide 2 Amino 6 cyanopyrazine 2 Amino 6 bromopyrazine 2 Amino 5 iodopyrazine 2 methylbutyl 2 methylpropanoate 2 6 Dibromoquinazoline 2 3 Dihydro 2 phenyl 4 1H quinolinone 1 Boc 5 Chloro 6 trifluoromethyl 1H indole 1 Boc 5 6 Dichloro 1H indole 2 boronic acid 1 4 diphenylbutadiyne 2 Aminomethyl benzonitrile

2 Chloro 5 nitrophenol 2 Iodobenzothiazole 5 Methyl 2 nitrophenol 6 Bromo 2 methylisoquinolin 1 2H one 6 Chloro 1 2 3 4 tetrahydropyrido 2 3 b pyrazine 6 Chloro 5 nitroquinoline 2 4 2 Aminobenzenesulfonyl piperazin 1 yl ethanol 1 Boc 1 2 dihydro 5 methoxy 2 oxo spiro 3H indole 3 4 piperidine 5 Bromopyridin 2 yl methyl carbamic acid tert butyl ester 2 4 3 benzo b 1 benzazepin 11 ylpropyl piperazin 1 yl ethanol 3 Iodopicolinic acid 3 Methoxy 4 methyl 2 nitrobenzoic acid 4 Imidazo 1 2 a pyrazin 2 yl 1 2 5 oxadiazol 3 amine 1 Tosyl 1H pyrrolo 2 3 b pyridin 3 ylboronic acid 1 Boc 4 4 Bromo 2 formylphenyl piperazine 1 Boc 5 Fluoro 1 2 dihydro 2 oxo spiro 3H indole 3 4 piperidine 2 Hydroxy 4 5 Dimethoxy Benzoic Acid 1H Indazole 7 carboxamide 1 4 Piperidinyl 2 trifluoromethyl 1H benzimidazole 6 7 dimethoxyquinazoline 2 4 diamine 1 Phenylsulfonyl 1H pyrrolo 2 3 b pyridine 4 Bromothiazol 5 yl methanol 2 Butoxyphenylboronic acid 3 3 Dimethylpiperidin 4 ol 2 Amino 4 iodopyrimidine 2 Chloro 6 nitroquinoline 3S 1 phenylmethoxycarbonyldiazinane 3 carboxylic acid 1 O tert butyl 2 O methyl 2R 4S 4 hydroxypiperidine 1 2 dicarboxylate 6 Bromo 8 chloroimidazo 1 2 a pyrazine 1R 4S N BOC 4 AMINOCYCLOPENT 2 ENECARBOXYLIC ACID

1 3 Benzodioxole 4 carbonylchloride 8 Bromo 2 methylquinoline 1 Methyl 1H pyrazol 4 amine hydrochloride 2 4 Iodophenyl ethanol 8S 13S 14S 13 methyl 1 2 6 7 8 14 15 16 octahydrocyclopenta a phenanthrene 3 17 dione 3R 3 9H fluoren 9 ylmethoxycarbonylamino 4 oxo 4 prop 2 enoxybutanoic acid 2 bromo 1 oxidopyridin 1 ium 2 4 Dibromothiazol 5 yl methanol 4 Chloro 6 iodothieno 3 2 d pyrimidine 3 5 Dichloropicolinamide 2 fluoro 6 trifluoromethyl benzene 1 sulfonyl chloride 2 TRIFLUOROMETHYL THIOPHENOL 2 Cyano 6 fluorobenzoic acid 2 Bromo 4 Trifluoromethoxy benzonitrile 1 Boc pyrazole 3 amino 5 hydroxybenzoic acid 1 IODO 3 5 DIMETHOXYBENZENE 7 Nitro 1 2 3 4 Tetrahydro Isoquinoline Hydrochloride 6 4 methylpiperazin 1 yl pyrimidin 4 amine 8 Bromo 1 chloroisoquinoline 2 2 methoxy 5 nitrophenyl acetic acid 4 Chloro 5 fluoropyrimidine 4 phenylspiro 2 benzofuran 3 2 furan 1 3 dione 5 Methyl 2 piperazin 1 yl thiazole 7 Amino N methyl 1 2 3 4 tetrahydroquinoline hydrochloride 5 bromo 5 chloro 1 3 dimethylimidazolidine 2 4 dione 1 5 Bromopyridin 3 yl N methylmethanamine 3 5 5 dioxophenothiazin 10 yl N N 2 trimethylpropan 1 amine 1 Boc 3 bromopyrrolidine 4 Bromobenzamide

3 5 Dichloronitrobenzene 2 Amino 5 chlorobenzenesulfonic acid 2 2 heptadecyl 2 imidazolin 1 yl ethanol 2 ethylcyclopenta 1 3 diene nickel 2 3 Aminophenylacetic acid methyl ester 2 Chloroethyl 4 methylbenzenesulfonate 4 METHOXY BETA NITROSTYRENE 6R 7R 7 Amino 3 5 methyl 2H tetrazol 2 yl methyl 8 oxo 5 thi a 1 azabicyclo 4 2 0 oct 2 ene 2 carboxylic acid 4 bromophenyl methyl trimethylsilane 4 Nitroisoxazole 1S 4R N BOC 4 AMINOCYCLOPENT 2 ENECARBOXYLIC ACID 6 Chloro 2 methylimidazo 1 2 b pyridazine 3 carboxylic acid 2R 1 4 methylphenyl sulfonylpyrrolidine 2 carboxylic acid 2R 5 amino 5 oxo 2 phenylmethoxycarbonylamino pentanoic acid 2 Methyl 7 phenyl 1H indene 5 chloro N ethyl 4 hydroxy 1 methyl 2 oxo N phenylquinoline 3 carboxamide 5 2 4 Bis S 3 methylmorpholino pyrido 2 3 d pyrimidin 7 yl 2 methoxyphenyl methanol 2S 2 2S 2 2S 2 3 acetamidopropanoylamino 3 1H imidazol 5 yl propanoyl amino 3 hydroxypropanoyl amino 3 1H imidazol 5 yl propanoic acid 2R 3S tert Butyl 6 oxo 2 3 diphenylmorpholine 4 carboxylate 2 6 Dichloro 3 methyl 5 nitropyridine 5 Fluoro 3 Methyl Pyridin 2 Ylamine 3beta 20beta 3 3 Carboxy 1 oxopropoxy 11 oxoolean 12 en 29 oic acid 2 3 4 Dichlorophenyl 1 2 pyrrolidin 1 ylmethyl piperidin 1 yl ethanone hydrochloride 1 Fluoro 2 iodo 3 methoxybenzene 3 4 bis trifluoromethyl phenyl boronic acid 3 Bromo 5 Methylbenzonitrile 3 4 Bis 3 indolyl maleimide 2 Bromomethyl 4 fluoro 1 methoxybenzene 4 Bromoacetyl 3 fluorophenylboronic acid 3 4 Dihydro 8 methoxynaphthalen 1 2H one