1 Boc 2 methoxycarbonylmethylpiperazine 3 ethyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 2 Bromo 6 chloropyridine 3 methyl 1H indazol 5 yl boronic acid 3 methyl 1H indazol 6 yl boronic acid 6 fluoro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H indazole 4 amino 2 chloro 3 fluorophenol 1 methyl 1H indazol 4 yl boronic acid 2 Pyrimidinecarboxylic acid 3 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 Chloro 2 iodophenol 1 3 Dichloro 2 methyl 5 nitrobenzene 3 methoxymethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinamide 3 Amino 6 chloropyridazine 3 Methyl 6 nitro 1H indazole 2 Mercapto 5 trifluoromethylpyridine 4 4 5 5 tetramethyl 2 3 methylbenzofuran 5 yl 1 3 2 dioxaborolane 2 6 chlorobenzofuran 5 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Amino 5 Bromo 3 Hydroxymethyl Pyridine 2 7 chlorobenzofuran 6 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 2 Hydroxy 3 nitro 5 trifluoromethyl pyridine 6 Benzylaminopurine 3 Fluoro 4 methylpyridine 6 fluorobenzo b thiophen 7 yl boronic acid 4 Chloro 3 nitropyridine 2 6 Dichloro 3 nitropyridine 3 acetylthiophen 2 yl boronic acid 2 Chloropyridine 5 carbaldehyde

2 2 chlorothiophen 3 yl 4 4 5 5 tetramethyl 1 3 2 dioxaborolane 3 chlorothiophen 2 yl boronic acid 2 Chloropyridine 6 carboxylic acid 4 methoxypicolinaldehyde 4 4 5 5 tetramethyl 2 5 methylthiophen 2 yl 1 3 2 dioxaborolane 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl thiophen 2 yl ethanone 2 Chloro 4 nitropyridine 1 phenyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 5 Bromo 2 pyridinecarboxylic acid 1 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazole 4 Chloro 3 methylpyridine hydrochloride 3 5 Dihydroxybenzoic acid 1 2 tert butyldimethylsilyl oxy ethyl 1H pyrazol 4 yl boronic acid 9 Bromoanthracene 1 phenyl 1H pyrazol 4 yl boronic acid 2 phenyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 3 Dimethylpyrazole 2 4 dichloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 methylthio 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 chloro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 1 Methyl 1H pyrazol 3 amine 4 Iodo 4 methylbiphenyl 2 Amino 6 chloropyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 1H one 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidin 2 amine 2 4 dimethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyrimidine 2 3 4 5 Tetrafluorobenzonitrile 2 chloro 6 methyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 6 trifluoromethyl pyridine

1 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl ethanone 4 4 Dibromobiphenyl 2 hydroxy 3 methylpyridine 4 Fluorobiphenyl 2 isopropyl 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 5 Hydroxy 1 indanone 5 Ethoxy 4 Methyloxazole 2 fluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 6 trifluoromethyl pyridine 2 Adamantanone 2 6 dimethoxypyridin 3 yl boronic acid 2 4 5 Trimethyloxazole 2 6 difluoro 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 chloro 2 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 Mercaptobenzoxazole 2 methoxy 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 Aminoisoxazole 6 methoxy 2 methyl 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 2 chloro 3 methyl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Bromo 2 5 difluoronitrobenzene 2 chloro 3 fluoro 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 fluoro 2 methoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 Trifluoromethylthio aniline 2 5 dichloro 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 Fluoro 2 hydroxybenzaldehyde 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1 8 naphthyridine 2 aminoimidazole sulfate 2 Thenoylacetonitrile 6 Bromoindoline 5 chloro 2 methoxy 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 6 methoxy 5 trifluoromethyl pyridin 3 yl boronic acid

6 Methoxy oxindole 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 3 trifluoromethyl pyridin 2 amine 2 4 5 Trimethoxybenzaldehyde 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl nicotinonitrile 2 ethoxy 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 4 6 Dimethoxysalicylaldehyde 1 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridin 2 yl ethanone 4 Bromooxindole 4 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrazolo 3 4 b pyridine 2 azetidin 1 yl 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl pyridine 3 Bromo 2 methoxy 6 picoline 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl 1H pyrrolo 2 3 b pyridine 5 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl picolinaldehyde 5 Chloro 2 nitrobenzaldehyde 1H pyrazolo 3 4 b pyridin 5 yl boronic acid 3 4 4 5 5 tetramethyl 1 3 2 dioxaborolan 2 yl isonicotinamide 4 bromo 1H indazole 3 carbamoyl 4 chlorophenylboronic acid 1 4 boronobenzoyl piperidine 4 carboxylic acid 5 bromo 3 methyl 1H indazole 3 fluoro 5 isopropoxyphenylboronic acid 4 carbamoyl 3 chlorophenylboronic acid 3 ethylamino phenylboronic acid 4 N Boc amino phenylboronic acid 3 ethylphenylboronic acid 4 isobutylphenylboronic acid 7 Azaindole 4 dipropylcarbamoyl phenylboronic acid 4 3 bromopropylcarbamoyl phenylboronic acid 1 Benzyl 3 piperidone hydrochloride