4 Methylisoxazole 3 carboxylic acid 3 phenylpyrazin 2 ol 4 6 Pyrimidinedicarboxylic acid 3 Chlorotetrahydrofuran 3 Chloro tetrahydropyran 9 Benzyl 3 9 diaza spiro 5 5 undecane 2 4dione 2 Bromo 6 chloro 4 nitropyridine 4 Benzyl 2 chloromethyl morpholine 1 Boc 3 methylene pyrrolidine 1 Benzhydryl 3 chloroazetidine 4 Bromo 2 3 dimethylanisole 7 Azabicyclo 4 2 0 octan 8 one 6 Bromo 1 2 3 4 tetrahydro 1 1 4 4 tetramethylnaphthalene 2 Methyl 2H 1 4 Benzoxazin 3 4H one 5 Methyl 4 phenyl 3 4 dihydro 2H pyrrole 4 Morpholinecarboxamide N N dimethyl 2 Bromo N tert butoxycarbonyl aniline 3 Iodomethyl oxetane 1 3 5 tris chloromethyl 2 4 dimethylbenzene 6 Chloroisoindolin 1 one 2 4 Dibromofuran 2 Bromo 1 4 bromo 1 1 biphenyl 4 yl ethanone 5 Bromo 2 3H benzofuranone 7 Bromo 3 methoxyquinoline 1 4 Methoxy benzyl piperidine 2 4 dione 3 Bromo 7 chloroquinoline 8 Bromochroman 3 one 8 Oxabicyclo 3 2 1 octan 3 one 1R Dimenthyl succinate 4 Boc 3 2 Oxo ethyl morpholine

2 Cyclohexen 1 one 2 Azabicyclo 2 2 2 octane 2 6 dicarboxylic acid 2 1 1 dimethylethyl 6 methyl ester 1R 4S 6R rel 4 Morpholinocyclohexanone 5 Nitroisatoic anhydride 7 Bromo 2 3 dihydro 1 8 naphthyridin 4 1H one 1 3 4 Dimethylphenyl 2 Phenylethane 1 2 Dione 4 4 Chlorobenzenesulfonyl benzaldehyde 3 Chromanone 1 4 1 3 Dioxolan 2 yl phenyl ethanone 2 Cyclohepten 1 one 1 2H Naphthalenone 3 4 dihydro 7 phenylmethyl 1 Boc 3 5 dioxopyrrolidine 1 Acetamido acetone 8 Methyl 3 oxo 3 4 dihydro 2H benzo b 1 4 oxazine 6 carbaldehyde 3 Hydroxy 5 methoxybenzaldehyde 4 Bromo 3 hydroxybenzaldehyde 9H Fluoren 9 yl methyl 2 oxoethylcarbamate 4 Boronicacid biphenyl 4 carboxylicacid methyl ester 5 Bromo 3 methoxybenzaldehyde 7 Methoxy 4 trifluoromethyl coumarin 5 Boc Amino pyridine 3 boronic acid pinacol ester 3 Pyrrolylboronic acid 3 tert Butoxycarbonyl amino methyl pyridin 4 yl boronic acid 3 4 Chlorobenzoylamino 1 3 chlorobenzyl 6 4 isopropoxyphenyl indole 2 carboxylic acid 1H 1 2 4 Triazole 3 5 diamine N3 4 aminosulfonyl phenyl 1 3 5 dimethyl 2 thienyl carboyl 9CI 1 1H indol 3 yl 2 2 phenylvinyl sulfonyl 1 2 dihydroisoquinoline 1 3 Chlorobenzyl 6 4 isopropoxyphenyl 3 pentanoyl amino indole 2 carboxylic acid 1H 1 2 4 Triazole 3 5 diamine N3 4 2 dimethylamino ethyl mino sulfonyl phenyl 1 3 5 dimethyl 2 thienyl carbonyl 9CI 2 4 2 4 Dioxo 5 thiazolidinyl methyl phenoxy acetic acid 3 Cyclohexyl L alanine hydrate

2S 3R 2 Methyl 3 morpholinecarboxylic acid 1S 3aR 6aS Hexahydro cyclopenta c pyrrole 1 2 dicarboxylic acid 2 tert butyl ester 4S 1 Boc 4 Methyl L proline 1 Amino cyclopentanecarboxylic acid ethyl ester hydrochloride 3 N Boc 3 methylbutane 1 3 diamine HCl 3 Pyridin 4 yl 3 9 diazaspiro 5 5 undecane 1S 3aR 6aS Octahydro cyclopenta c pyrrole 1 carboxylic acid hydrochloride 6aR tert Butyl 6a trifluoromethyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 6aR tert Butyl 6a phenyl hexahydropyrrolo 3 4 c pyrrole 2 1H carboxylate 3aR tert Butyl 3a ethyl hexahydropyrrolo 3 4 c pyrrole 2 3a 1H dicarboxylate 4 Bromophenyl piperidin 4 yl methanone 1 2 3 4 Tetrahydroisoquinolin 4 ol 2 Amino 2 2 pyridyl ethanol 4 4 Acetylpiperazin 1 yl 3 trifluoromethyl aniline 2 Methoxy 1 propanamine 3R 4R 4 4 Fluorophenyl 3 piperidinemethanol 3 Dimethylamino pyrrolidine 1 Cbz 3 aminomethylazetidine 1 Amino 3 buten 2 ol 4 3 nitrophenyl piperidine 2S 5S 2 5 Dimethylmorpholine 3 8 Diazabicyclo 3 2 1 octane 1S 2R 2 Amino cyclohexanol 1S 2R 2 Amino cyclohexanol HCl 1 6 7 dimethoxy 2H benzo d 1 3 dioxolan 5 yl prop 2 ylamine 1S 3R 3 Aminocyclopentanol 1S 3S 3 Aminocyclopentanol 1 Cyclopropylethanamine 1R 3R 3 Aminocyclopentanol 1 Oxa 7 azaspiro 4 5 decane

2 Ethenylmorpholine 6 Oxa 2 aza spiro 4 5 decane 7 Oxa 2 aza spiro 4 5 decane 2 piperidin 2 yl ethanamine 8 Oxa 2 azaspiro 4 5 decane 2 2 Methoxyethyl piperidine hydrochloride 3 2 Pyridyl morpholine 2 2 pyridinyl morpholine 3 2 Thienyl morpholine 3 Thiophen 3 yl morpholine 2 Thiophen 3 yl morpholine 3 Cyclopropylmorpholine 2 Cyclopropylmorpholine 3 Cyclobutylmorpholine 2 Cyclobutylmorpholine 3 Cyclohexylmorpholine 2 Benzylmorpholine 2 Phenyl 2 6 diazaspiro 3 3 heptan 1 one 2 Pyrrolidineacetic acid ethyl ester 1 3 Chloro benzyl 1 2 3 4 tetrahydro quinoxaline 2 Azabicyclo 2 2 1 hept 5 ene 1 Boc 2 Aminomethylazetidine hydrochloride 2 2 Dimethylpyrrolidine 3 Pyrrolidin 3 yl aniline dihydrochloride 1 Boc 4 1 pyrrolidinyl 3 6 dihydro 2H pyridine 6 Aminomethyl 3 morpholinone hydrochloride 4 Ethyl 2 3 methyl 4 nitrophenyl morpholine 3 Amino cyclopentanone 2 Piperidin 4 yl ethylamine dihydrochloride 1 Methyl 2 piperazinemethanamine